| Identification | Back Directory | [Name]
MAK-683 hyrochloride | [CAS]
2170606-94-5 | [Synonyms]
MAK-683 hyrochloride MAK-683 hydrochloride EED inhibitor,MAK 683 hyrochloride,embryonic ectoderm development,Histone Methyltransferase,MAK 683,inhibit,MAK-683,MAK683,MAK683 hyrochloride,Inhibitor | [Molecular Formula]
C20H18ClFN6O | [MOL File]
2170606-94-5.mol | [Molecular Weight]
412.85 |
| Hazard Information | Back Directory | [Uses]
MAK683 hydrochloride is an embryonic ectoderm development (EED) inhibitor extracted from patent US20160176882 A1, compound example 2. MAK683 exhibits IC50s of 59, 89, 26 nM in EED Alphascreen binding, LC-MS and ELISA assay[1][2]. | [References]
[1] Chan, Ho Man, et al. TRIAZOLOPYRIMIDINE COMPOUNDS AND USES THEREOF. US20160176882 A1. [2] Huang D, et al. Binding Modes of Small-Molecule Inhibitors to the EED Pocket of PRC2. Chemphyschem. 2020 Feb 4;21(3):263-271. DOI:10.1002/cphc.201900903 |
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