| Identification | Back Directory | [Name]
Pyrazolo[4'',3'':3',4']cyclohepta[1',2':4,5]thieno[3,2-d]pyrimidin-10(9H)-one, 8-(2R)-1-azabicyclo[2.2.2]oct-2-yl-2,4,5,6-tetrahydro- | [CAS]
2562329-14-8 | [Synonyms]
Cdc7-IN-18 Pyrazolo[4'',3'':3',4']cyclohepta[1',2':4,5]thieno[3,2-d]pyrimidin-10(9H)-one, 8-(2R)-1-azabicyclo[2.2.2]oct-2-yl-2,4,5,6-tetrahydro- | [Molecular Formula]
C19H21N5OS | [MOL File]
2562329-14-8.mol | [Molecular Weight]
367.47 |
| Hazard Information | Back Directory | [Uses]
Cdc7-IN-18 (compound 1-2) is a potent CDC7 inhibitor with an IC50 of 1.29 nM for Cdc7/DBF4 enzyme. Cdc7-IN-18 shows antiproliferative activities with IC50 of 53.62 nM in COLO205 cells[1]. | [IC 50]
Cdc7: 1.29 nM (IC50) | [References]
[1] Li Gang, et al. Tetracyclic compounds as cdc7 inhibitors. WO2020239107A1. |
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