| Identification | Back Directory | [Name]
5-Oxaspiro[3.4]octane-7,8-diol, 6-(6-amino-9H-purin-9-yl)-1-(hydroxymethyl)-, (1R,4R,6R,7R,8S)- | [CAS]
2567564-33-2 | [Synonyms]
PRMT5-IN-11 5-Oxaspiro[3.4]octane-7,8-diol, 6-(6-amino-9H-purin-9-yl)-1-(hydroxymethyl)-, (1R,4R,6R,7R,8S)- | [Molecular Formula]
C13H17N5O4 | [MOL File]
2567564-33-2.mol | [Molecular Weight]
307.31 |
| Hazard Information | Back Directory | [Uses]
PRMT5-IN-11 is a promising structure-dependent inhibition of the protein methyltransferase PRMT5:MEP50 complex in the (sub)micromolar range. | [References]
[1] Jouffroy L, et al. Regio- and Stereoselective Synthesis of C-4' Spirocyclobutyl Ribofuranose Scaffolds and Their Use as Biologically Active Nucleoside Analogues. Org Lett. 2021 Nov 19;23(22):8828-8833. DOI:10.1021/acs.orglett.1c03334 |
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