| Identification | Back Directory | [Name]
1H-Purine-2,6-dione, 8-[(acetyloxy)methyl]-7-[(3-bromophenyl)methyl]-3,7-dihydro-3-methyl- | [CAS]
2761321-18-8 | [Synonyms]
BRD4-BD1-IN-1 1H-Purine-2,6-dione, 8-[(acetyloxy)methyl]-7-[(3-bromophenyl)methyl]-3,7-dihydro-3-methyl- | [Molecular Formula]
C16H15BrN4O4 | [MOL File]
2761321-18-8.mol | [Molecular Weight]
407.22 |
| Hazard Information | Back Directory | [Uses]
BRD4-BD1-IN-1 (Compound 9a) is a BRD4-BD1 inhibitor with an IC50 of 38.20 μM[1]. | [IC 50]
BRD4 BD1: 38.20 μM (IC50) | [References]
[1] Chang Y, et al. Design, synthesis, biological evaluation, and molecular docking of 1, 7-dibenzyl-substituted theophylline derivatives as novel BRD4-BD1-selective inhibitors. Medicinal Chemistry Research, 2021, 30(8): 1453-1468. |
|
|