| Identification | Back Directory | [Name]
AC-ARG-CYS-MET-5-AMINOPENTANOYL-ARG-VAL-TYR-5-AMINOPENTANOYL-CYS-NH2, (DISULFIDE BOND) TRIFLUOROACETATE | [CAS]
353487-64-6 | [Synonyms]
Ac-Arg-Cys-Met-Ava-Arg-Val-Tyr-Ava-Cys-NH2|(Disulfide bond)
Ac-Arg-Cys-Met-5-aminopentanoyl-Arg-Val-Tyr-5-aminopentanoyl-Cys-NH2, (Disulfide bond)
AC-ARG-CYS-MET-5-AMINOPENTANOYL-ARG-VAL-TYR-5-AMINOPENTANOYL-CYS-NH2, (DISULFIDE BOND) TRIFLUOROACETATE
Ac-Arg-Cys-Met-5-aminopentanoyl-Arg-Val-Tyr-5-aminopentanoyl-Cys-NH2 trifluoroacetate salt (Disulfide bond)
L-Cysteinamide, N2-acetyl-L-arginyl-L-cysteinyl-L-methionyl-5-aminopentanoyl-L-arginyl-L-valyl-L-tyrosyl-5-aminopentanoyl-, cyclic (2→9)-disulfide | [Molecular Formula]
C49H82N16O11S3 | [MDL Number]
MFCD09037404 | [MOL File]
353487-64-6.mol | [Molecular Weight]
1167.47 |
| Hazard Information | Back Directory | [Uses]
hMCH-1R antagonist 1 (Compound 30) is an effective and selective antagonist of human melanin-concentrating hormone receptor 1 (hMCHR1) with an KB value of 3.6 nM. HMCH-1R antagonist 1 can bind to hMCHR1 and hMCHR2 with IC50 values of 65 nM and 49 nM, respectively. HMCH-1R antagonistist 1 can be used for metabolic research[1]. | [References]
[1] Bednarek MA, et al. Synthesis and biological evaluation in vitro of selective, high affinity peptide antagonists of human melanin-concentrating hormone action at human melanin-concentrating hormone receptor 1. Biochemistry. 2002 May 21;41(20):6383-90. DOI:10.1021/bi0200514 |
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