122830-14-2
122830-14-2 結構式
物理化學性質
沸點456.4±34.0 °C(Predicted)
密度1.27±0.1 g/cm3(Predicted)
儲存條件-20°C儲存
溶解度溶于二甲基亞砜
酸度系數(shù)(pKa)10.17±0.40(Predicted)
常見問題列表
生物活性
Deriglidole 是外周腎上腺素能受體拮抗劑，對 α2 腎上腺素受體具有高親和力。靶點
Adrenoceptor
體外研究
Deriglidole is a selective α 2 -receptor inhibitor. Deriglidole inhibits [ 3 H]Clonidine and [ 3 H]Idazoxan but not [ 3 H]Prazosin binding to rat cortical and human platelet α 2 -adrenoceptors and is more selective than Idazoxan for peripheral receptors.