864082-35-9
864082-35-9 結(jié)構(gòu)式
物理化學(xué)性質(zhì)
沸點(diǎn)739.3±60.0 °C(Predicted)
密度1.479±0.06 g/cm3(Predicted)
酸度系數(shù)(pKa)12.73±0.40(Predicted)
應(yīng)用領(lǐng)域
用途一
GSK299115A is a G-Protein-Coupled Receptor Kinase 2 (GRK2) Inhibitor (GRK2 inhibitor). G-protein-coupled receptor kinase 2 (GRK2) is a G-protein-coupled receptor kinase that is ubiquitously expressed in many tissues and regulates various intracellular mechanisms. GRK2 plays an important role in the maintenance of heart structure and function; thus, this kinase is involved in many cardiovascular diseases.