JMS-17-2 HYDROCHLORIDE
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- CAS號(hào):
- 2341841-07-2
- 英文名:
- JMS 17-2 hydrochloride
- 英文別名:
- JMS 17-2 hydrochloride
- 中文名:
- JMS-17-2 HYDROCHLORIDE
- 中文別名:
- CBNumber:
- CB28202884
- 分子式:
- C25H27Cl2N3O
- 分子量:
- 456.41
- MOL File:
- 2341841-07-2.mol
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JMS-17-2 HYDROCHLORIDE化學(xué)性質(zhì)
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溶解度:
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Soluble to 100 mM in DMSO and to 50 mM in ethanol
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JMS-17-2 HYDROCHLORIDE性質(zhì)、用途與生產(chǎn)工藝
JMS-17-2 hydrochloride 是一種有效的選擇性 CX3CR1 拮抗劑,IC50 為 0.32 nM。JMS-17-2 hydrochloride 降低乳腺癌細(xì)胞的轉(zhuǎn)移和定植。
JMS-17-2 (10 mg/kg; aministered i.p.; twice a day for three weeks) causes a dramatic reduction of tumors in both skeleton and visceral organs in SCID mice.
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Animal Model:
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SCID mice (~25g) with MDA-231 xenograft
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Dosage:
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10 mg/kg
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Administration:
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Aministered i.p.; twice a day for three weeks
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Result:
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Caused a dramatic reduction of tumors in both skeleton and visceral organs.
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JMS-17-2 HYDROCHLORIDE
上下游產(chǎn)品信息
上游原料
下游產(chǎn)品
JMS-17-2 HYDROCHLORIDE
生產(chǎn)廠家
2341841-07-2, JMS-17-2 HYDROCHLORIDE 相關(guān)搜索:
- 抑制劑
- 2341841-07-2
- JMS 17-2 hydrochloride