XMD17 109性質(zhì)、用途與生產(chǎn)工藝

生物活性

靶點(diǎn)

體外研究

ERK5-IN-1可有效抑制ERK5的生物化學(xué)性質(zhì)，其IC50值為162 nM，在細(xì)胞水平可抑制內(nèi)皮生長(zhǎng)因子誘導(dǎo)的ERK5自磷酸化，其EC50值為90 nM。

XMD17 109 上下游產(chǎn)品信息

上游原料

下游產(chǎn)品

XMD17 109 生產(chǎn)廠家

XMD17 109 圖譜信息:

1435488-37-1, XMD17 109 相關(guān)搜索:

• MAPK
• Inhibitors
• 抑制劑
• 天然產(chǎn)物
• 細(xì)胞生物學(xué)試劑
• 小分子抑制劑，天然產(chǎn)物
• 小分子抑制劑
• C36H46N8O3
• 化合物XMD17-109,10 MM DMSO 溶液
• 11-環(huán)戊基-2-[[2-乙氧基-4-[[4-(4-甲基-1-哌嗪基)-1-哌啶基]羰基]苯基]氨基]-5,11-二氫-5-甲基-6H-嘧啶并[4,5-B][1,4]苯并二氮雜環(huán)庚烷-6-酮
• 11-環(huán)戊基-2-((2-乙氧基-4-(4-(4-甲基哌嗪-1-基)哌啶-1-羰基-1-羰基)苯基)氨基)-5-甲基-5H-苯并[E]嘧啶并[5,4-B][1,4]二氮雜卓-6(11H)-酮
• ERK-5抑制劑(XMD17-109)
• 11-環(huán)戊基-2-[[2-乙氧基-4-[[4-(4-甲基-1-哌嗪基)-1-哌啶基]羰基]苯基]氨基]-5,11-二氫-5-甲基-6H-嘧啶并[4,5-B][1,4]苯并二氮雜卓-6-酮
• 1435488-37-1
• XMD17-109
• 11-Cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-piperazin-1-yl)piperidin-1-yl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one
• XMD17-109, 10 mM in DMSO
• 11-Cyclopentyl-2-[2-ethoxy-4-[4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]anilino]-5-methylpyrimido[4,5-b][1,4]benzodiazepin-6-one
• 6H-Pyrimido[4,5-b][1,4]benzodiazepin-6-one, 11-cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-
• CS-1288
• XMD17 109;XMD17109
• 11-Cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one XMD17-109
• 11-Cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-6H-pyrimido[4,5-b][1,4]benzodiazepin-6-one
• XMD17 109