4-Amino-5-chloro-N-(1-((4-fluorophenyl)methyl)-4-piperidinyl)-2-methox ybenzamide
- CAS No.
- 154540-49-5
- Chemical Name:
- 4-Amino-5-chloro-N-(1-((4-fluorophenyl)methyl)-4-piperidinyl)-2-methox ybenzamide
- Synonyms
- fluoroclebopride;Fluoroclebopride, 10 mM in DMSO;Abmole M4962-10mg fluoroclebopride 154540-49-5;Abmole M4962-50mg fluoroclebopride 154540-49-5;Inhibitor,inhibit,Fluoroclebopride,Dopamine Receptor;4-Amino-5-chloro-N-(1-((4-fluorophenyl)methyl)-4-piperidinyl)-2-methox ybenzamide;Benzamide,4-amino-5-chloro-N-[1-[(4-fluorophenyl)methyl]-4-piperidinyl]-2-methoxy-
- CBNumber:
- CB11242925
- Molecular Formula:
- C20H23ClFN3O2
- Molecular Weight:
- 391.87
- MDL Number:
- MOL File:
- 154540-49-5.mol
- MSDS File:
- SDS
- TDS File:
- TDS
| Product description | Number | Pack Size | Price |
| Fluoroclebopride ≥98% | 23447 | 1mg | $41 |
| Fluoroclebopride ≥98% | 23447 | 5mg | $178 |
| Fluoroclebopride ≥98% | 23447 | 10mg | $312 |
| Fluoroclebopride ≥98% | 23447 | 1mg | $37 |
| Fluoroclebopride ≥98% | 23447 | 5mg | $161 |
| More product size | |||
| Boiling point | 518.2±50.0 °C(Predicted) |
|---|---|
| Density | 1.31±0.1 g/cm3(Predicted) |
| storage temp. | Store at -20°C |
| solubility | DMF: 20 mg/ml; DMF:PBS (pH 7.2) (1:9): 0.1 mg/ml; DMSO: 10 mg/ml; Ethanol: 10 mg/ml |
| form | A crystalline solid |
| pka | 13.62±0.20(Predicted) |
| color | White to off-white |
4-Amino-5-chloro-N-(1-((4-fluorophenyl)methyl)-4-piperidinyl)-2-methox ybenzamide price More Price(35)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Cayman Chemical | 23447 | Fluoroclebopride ≥98% | 154540-49-5 | 1mg | $41 | 2026-04-30 | Buy |
| Cayman Chemical | 23447 | Fluoroclebopride ≥98% | 154540-49-5 | 5mg | $178 | 2026-04-30 | Buy |
| Cayman Chemical | 23447 | Fluoroclebopride ≥98% | 154540-49-5 | 10mg | $312 | 2026-04-30 | Buy |
| Cayman Chemical | 23447 | Fluoroclebopride ≥98% | 154540-49-5 | 1mg | $37 | 2024-03-01 | Buy |
| Cayman Chemical | 23447 | Fluoroclebopride ≥98% | 154540-49-5 | 5mg | $161 | 2024-03-01 | Buy |
4-Amino-5-chloro-N-(1-((4-fluorophenyl)methyl)-4-piperidinyl)-2-methox ybenzamide Chemical Properties,Uses,Production
Description
Fluoroclebopride is a benzamide analog that is used in positron emission tomography (PET) applications. It binds reversibly to dopamine receptors (Kis = 0.95, 5.7, 5.46, and 144 nM for D2-like, D2(long), D3, and D4 receptors, respectively, in radioligand binding assays). It is selective for these receptors over D1, serotonin 5-HT2, and α2-adrenergic receptors (Kis = >10,000, 283, and 1,300 nM, respectively). A fluorine-18 moiety has been used to label this compound for use as a probe for studying D2/D3 receptor availability via PET in various monkey models.
Uses
Fluoroclebopride binds reversibly to dopamine receptors. 18F labeled fluoroclebopride has been used as a probe for studying D2/D3 receptor availability via PET in various monkey models[1][2].
References
[1] Nader MA, Czoty PW. PET imaging of dopamine D2 receptors in monkey models of cocaine abuse: genetic predisposition versus environmental modulation. Am J Psychiatry. 2005 Aug;162(8):1473-82. DOI:10.1176/appi.ajp.162.8.1473
[2] Czoty PW, et al. Effects of repeated treatment with the dopamine D2/D3 receptor partial agonist aripiprazole on striatal D2/D3 receptor availability in monkeys. Psychopharmacology (Berl). 2013 Sep 29:10.1007/s00213-013-3274-7. DOI:10.1007/s00213-013-3274-7. doi: 10.1007/s00213-013-3274-7
4-Amino-5-chloro-N-(1-((4-fluorophenyl)methyl)-4-piperidinyl)-2-methox ybenzamide Preparation Products And Raw materials
Raw materials
Preparation Products
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| ATK CHEMICAL COMPANY LIMITED | +undefined-21-51877795 | ivan@atkchemical.com | China | 33024 | 60 |
| TargetMol Chemicals Inc. | +1-781-999-5354; +17819995354 | marketing@targetmol.com | United States | 32466 | 58 |
| HANGZHOU CLAP TECHNOLOGY CO.,LTD | 86-571-88216897,88216896 13588875226 | sales@hzclap.com | CHINA | 6312 | 58 |
| BOC Sciences | 16314854226; +16314854226 | inquiry@bocsci.com | United States | 19853 | 58 |
| Zhejiang J&C Biological Technology Co.,Limited | +1-2135480471 +1-2135480471; | sales@sarms4muscle.com | China | 10473 | 58 |
| InvivoChem | +1-708-310-1919 +1-13798911105 | sales@invivochem.cn | United States | 6391 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; | support@targetmol.com | United States | 39039 | 58 |
| ShenZhen Trendseen Biological Technology Co.,Ltd. | 13417589054 | trendseenbio@gmail.com | China | 11681 | 58 |
| Zibo Hangyu Biotechnology Development Co., Ltd | +86-0533-2185556 +8615965530500 | nickzhang@hangyubiotech.com | China | 9949 | 58 |
| Aladdin Scientific | tp@aladdinsci.com | United States | 52923 | 58 |
View Lastest Price from 4-Amino-5-chloro-N-(1-((4-fluorophenyl)methyl)-4-piperidinyl)-2-methox ybenzamide manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2026-05-26 | Fluoroclebopride
154540-49-5
|
$68.00-162.00 | 99.80% | 10g | TargetMol Chemicals Inc. |
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- Fluoroclebopride
154540-49-5
- $68.00-162.00
- 99.80%
- TargetMol Chemicals Inc.
