ChemicalBook >> CAS DataBase List >>1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE
1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE
![1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE Structure](CAS/GIF/4789-68-8.gif)
- CAS No.
- 4789-68-8
- Chemical Name:
- 1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE
- Synonyms
- vufb-6281;octoclothepinemaleate;OCTOCLOTHEPIN MALEATE;OCTOCLOTHEPIN MALEATE SALT;OCTOCLOTHEPIN MALEATE D2 DOPAMINE ANTAGO NIS;8-chloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo(b,f)thiepinmaleate;1-(8-chloro-10,11-dihydrodibenzo(b,f)thiepin-10-yl)-4-methyl-piperazinmale;d,l-8-chloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo(b,f)thiepinmaleate;1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE;Piperazine, 1-(8-chloro-10,11-dihydrodibenzo(B,F)thiepin-10-yl)-4-methyl-, maleate
- CBNumber:
- CB6143736
- Molecular Formula:
- C23H25ClN2O4S
- Molecular Weight:
- 460.97
- MDL Number:
- MFCD00153855
- MOL File:
- 4789-68-8.mol
- MSDS File:
- SDS
- TDS File:
- TDS
Last updated:2026-05-28 02:10:43
| Product description | Number | Pack Size | Price |
| Octoclothepin maleate salt solid | O111 | 25mg | $108 |
| Octoclothepin maleate salt 99.14% | CS-0134312 | 5mg | $89 |
| Octoclothepin maleate salt 99.14% | CS-0134312 | 10mg | $141 |
| Octoclothepin maleate salt 99.14% | CS-0134312 | 25mg | $253 |
| Octoclothepin maleate salt 99.14% | CS-0134312 | 5mg | $89 |
| solubility | 45% (w/v) aq 2-hydroxypropyl-β-cyclodextrin: >21 mg/mL |
|---|---|
| form | solid |
| color | white |
| InChI | 1S/C19H21ClN2S.C4H4O4/c1-21-8-10-22(11-9-21)17-12-14-4-2-3-5-18(14)23-19-7-6-15(20)13-16(17)19;5-3(6)1-2-4(7)8/h2-7,13,17H,8-12H2,1H3;1-2H,(H,5,6)(H,7,8)/b;2-1- |
| InChIKey | GWKBZIADWSOIQV-BTJKTKAUSA-N |
| SMILES | [H]\C(=C(/[H])C(O)=O)C(O)=O.CN1CCN(CC1)C2Cc3ccccc3Sc4ccc(Cl)cc24 |
| EWG's Food Scores | 1 |
| FDA UNII | M5Z1H0WN1S |
| UNSPSC Code | 12352200 |
| NACRES | NA.77 |
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS06 |
|---|---|
| Signal word | Danger |
| Hazard statements | H301 |
| Precautionary statements | P301+P310 |
| PPE | Eyeshields, Faceshields, Gloves, type P2 (EN 143) respirator cartridges |
| Hazard Codes | T |
| Risk Statements | 25 |
| Safety Statements | 36/37/39-45 |
| RIDADR | UN 2811 6.1/PG 3 |
| WGK Germany | 3 |
| RTECS | TL1575000 |
| Storage Class | 6.1C - Combustible acute toxic Cat.3 toxic compounds or compounds which causing chronic effects |
| Hazard Classifications | Acute Tox. 3 Oral |
1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE price More Price(11)
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Sigma-Aldrich | O111 | Octoclothepin maleate salt solid | 4789-68-8 | 25mg | $108 | 2026-04-30 | Buy |
| ChemScene | CS-0134312 | Octoclothepin maleate salt 99.14% | 4789-68-8 | 5mg | $89 | 2026-06-04 | Buy |
| ChemScene | CS-0134312 | Octoclothepin maleate salt 99.14% | 4789-68-8 | 10mg | $141 | 2026-06-04 | Buy |
| ChemScene | CS-0134312 | Octoclothepin maleate salt 99.14% | 4789-68-8 | 25mg | $253 | 2026-06-04 | Buy |
| ChemScene | CS-0134312 | Octoclothepin maleate salt 99.14% | 4789-68-8 | 5mg | $89 | 2026-06-04 | Buy |
1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE Chemical Properties,Uses,Production
Uses
Octoclothepin Maleate Salt is an SR-2A inhibitor as well as a D2DR inhibitor.
Biological Activity
D2 dopamine receptor antagonist; 5-HT2 serotonin receptor antagonist.
in vivo
Octoclothepin possesses high cataleptogenic and anti-apomorphine activities in rats; it is able to exert full protection against apomorphine-induced emesis in dogs after the dose of 0.1 mg/kg s.c.[1].
Octoclothepin in doses of 0.5 and 1.5 mg/kg s.c. reduces the DA level and raises the HVA and DOPAC levels significantly[1].
1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE Preparation Products And Raw materials
Raw materials
Preparation Products
1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE Suppliers
Global( 13)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| TargetMol Chemicals Inc. | +17819995354 | marketing@targetmol.com | United States | 19956 | 58 |
| Energy Chemical | 021-58432009 400-005-6266 | marketing@energy-chemical.com | China | 44918 | 58 |
| TargetMol Chemicals Inc. | 15002134094 | marketing@targetmol.cn | China | 29845 | 58 |
| Merck KGaA | -- | ordercn@merckgroup.com | China | 6394 | 58 |
| Santa Cruz Biotechnology Inc | -- | scbt@scbt.com | China | 6594 | 58 |
| Supplier | Advantage |
|---|---|
| TargetMol Chemicals Inc. | 58 |
| Energy Chemical | 58 |
| TargetMol Chemicals Inc. | 58 |
| Merck KGaA | 58 |
| Santa Cruz Biotechnology Inc | 58 |
View Lastest Price from 1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2026-05-11 | Octoclothepin maleate salt
4789-68-8
|
$1520.00-2500.00 | 10g | TargetMol Chemicals Inc. |
-
- Octoclothepin maleate salt
4789-68-8
- $1520.00-2500.00
- TargetMol Chemicals Inc.
4789-68-8(1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE)Related Search:
2-Chloro-11-(4-(2-mandeloyloxyethyl)piperazino)-10,11-dihydrodibenzo(b ,f)thiepin bis(maleate)
4-(8-Chloro-10,11-dihydrodibenzo(b,f)thiepin-10-yl)-1-piperazinebutano l dimaleate
1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE
1-Piperazinebutanol, 4-(8-chloro-10,11-dihydrodibenzo(b,f)thiepin-10-y l)-alpha-methyl-, (Z)-2-butenedioate (1:2)
Piperazine, 1-(8-chloro-10,11-dihydrodibenzo(b,f)thiepin-10-yl)-4-meth yl-, S-oxide, (Z)-2-butenedioate (1:1)
1-(8-chloro-10,11-dihydrodibenzo(b,f)thiepin-10-yl)-4-methyl-piperazinmale
8-chloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo(b,f)thiepinmaleate
d,l-8-chloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo(b,f)thiepinmaleate
octoclothepinemaleate
vufb-6281
OCTOCLOTHEPIN MALEATE
OCTOCLOTHEPIN MALEATE SALT
1-(8-CHLORO-10,11-DIHYDRODIBENZO[B,F]THIEPIN-10-YL)-4-METHYL-PIPERAZINE MALEATE
OCTOCLOTHEPIN MALEATE D2 DOPAMINE ANTAGO NIS
Piperazine, 1-(8-chloro-10,11-dihydrodibenzo(B,F)thiepin-10-yl)-4-methyl-, maleate
1-(8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl)-4-methyl-piperazine maleate salt
4789-68-8
C23H25ClN2O4S
C19H21ClN2SC4H4O4
C19H21ClN2OSC4H4O4
