Paliperidone
|
- $5 - $9000
- Product name: Paliperidone
- CAS: 144598-75-4
- MF: C23H27FN4O3
- MW: 426.48
- EINECS:620-493-1
- MDL Number:MFCD00871802
- Synonyms:3-[2-[4-(6-Fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-9-hydroxy-2-Methyl-;Risperidone EP IMpurity C;Paliperidone 9-Hydroxyrisperidone;9-Hydroxyrisperidone solution;Racemic Paliperidone;4h-pyrido(2,1-a)pyrimidin-4-one,6,7,8,9-tetrahydro-3-(2-(4-(6-fluro-1,2-benzis ;oxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl- ;r76477
104 prices
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Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- Ambeed
- ApexBio Technology
- Arctom
- AvaChem
- Biosynth
- Cayman Chemical
- Chemcia Scientific
- Chem-Impex
- ChemScene
- Chemtos
- Crysdot
- DC Chemicals
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TCI Chemical
- Thermo Scientific Chemicals
- Tocris
- TRC
- Usbiological
Package
- 1mg
- 2.5mg
- 5mg
- 10mg
- 1ml of 1mg
- 25mg
- 50mg
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- 250mg
- 10
- 1mL
- 500mg
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- 1g
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- 2G
- 5g
- 5000mg
- 10g
- 25g
- 100000mg
- 1 g
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98%
- Packaging10mg
- Price$10
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98%
- Packaging50mg
- Price$14
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98%
- Packaging250mg
- Price$30
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98%
- Packaging1g
- Price$68
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98%
- Packaging5g
- Price$224
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA001JQR
- Product description6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98%
- Packaging25g
- Price$863
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product number10483
- Product descriptionPaliperidone 98%
- Packaging25G
- Price$640
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product number10483
- Product descriptionPaliperidone 98%
- Packaging5G
- Price$155
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product numberS451
- Product descriptionPaliperidone
- Packaging5g
- Price$645
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product numberJ10457
- Product descriptionPaliperidone >98%(HPLC),powder
- Packaging1g
- Price$642
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberS451
- Product descriptionPaliperidone 98%(HPLC)
- Packaging5g
- Price$665
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ98586
- Product descriptionPaliperidone 95%
- Packaging5g
- Price$498
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberS451
- Product descriptionPaliperidone 98%(HPLC)
- Packaging1g
- Price$243
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ98586
- Product descriptionPaliperidone 95%
- Packaging1g
- Price$166
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10457
- Product descriptionPaliperidone >98%(HPLC),powder
- Packaging100mg
- Price$195
- Updated2026-06-04
- Buy
- ManufacturerAK Scientific
- Product numberJ10457
- Product descriptionPaliperidone >98%(HPLC),powder
- Packaging25mg
- Price$62
- Updated2026-06-04
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98% | 10mg | $10 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98% | 50mg | $14 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one ≥98% | 250mg | $30 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98% | 1g | $68 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98% | 5g | $224 | 2026-05-28 | Buy |
| aablocks | AA001JQR | 6,7,8,9-Tetrahydro-3-(2-(4-(6-fluro-1,2-benzisoxazol-3-yl)-1-piperidinyl)ethyl)-9-hydroxy-2-methyl-4H-pyrido[2,1-a]pyrimidin-4-one 98% | 25g | $863 | 2026-05-28 | Buy |
| ACHEMBLOCK | 10483 | Paliperidone 98% | 25G | $640 | 2026-05-27 | Buy |
| ACHEMBLOCK | 10483 | Paliperidone 98% | 5G | $155 | 2026-05-27 | Buy |
| AK Scientific | S451 | Paliperidone | 5g | $645 | 2021-12-16 | Buy |
| AK Scientific | J10457 | Paliperidone >98%(HPLC),powder | 1g | $642 | 2026-06-04 | Buy |
| AK Scientific | S451 | Paliperidone 98%(HPLC) | 5g | $665 | 2026-06-04 | Buy |
| AK Scientific | J98586 | Paliperidone 95% | 5g | $498 | 2026-06-04 | Buy |
| AK Scientific | S451 | Paliperidone 98%(HPLC) | 1g | $243 | 2026-06-04 | Buy |
| AK Scientific | J98586 | Paliperidone 95% | 1g | $166 | 2026-06-04 | Buy |
| AK Scientific | J10457 | Paliperidone >98%(HPLC),powder | 100mg | $195 | 2026-06-04 | Buy |
| AK Scientific | J10457 | Paliperidone >98%(HPLC),powder | 25mg | $62 | 2026-06-04 | Buy |
Properties
Melting point :158-160°C
Boiling point :612.3±65.0 °C(Predicted)
Density :1.45±0.1 g/cm3(Predicted)
Flash point :9℃
storage temp. :2-8°C
solubility :DMSO: soluble2mg/mL, clear (warmed)
pka :13.00±0.60(Predicted)
form :powder
color :white to brown
Henry's Law Constant :1.2×1015 mol/(m3Pa) at 25℃, HSDB (2015)
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.
InChI :InChI=1S/C23H27FN4O3/c1-14-17(23(30)28-9-2-3-19(29)22(28)25-14)8-12-27-10-6-15(7-11-27)21-18-5-4-16(24)13-20(18)31-26-21/h4-5,13,15,19,29H,2-3,6-12H2,1H3
InChIKey :PMXMIIMHBWHSKN-UHFFFAOYSA-N
SMILES :C12C(O)CCCN1C(=O)C(CCN1CCC(C3C4=C(ON=3)C=C(F)C=C4)CC1)=C(C)N=2
CAS DataBase Reference :144598-75-4(CAS DataBase Reference)
Boiling point :612.3±65.0 °C(Predicted)
Density :1.45±0.1 g/cm3(Predicted)
Flash point :9℃
storage temp. :2-8°C
solubility :DMSO: soluble2mg/mL, clear (warmed)
pka :13.00±0.60(Predicted)
form :powder
color :white to brown
Henry's Law Constant :1.2×1015 mol/(m3Pa) at 25℃, HSDB (2015)
Stability :Stable for 2 years from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 2 months.
InChI :InChI=1S/C23H27FN4O3/c1-14-17(23(30)28-9-2-3-19(29)22(28)25-14)8-12-27-10-6-15(7-11-27)21-18-5-4-16(24)13-20(18)31-26-21/h4-5,13,15,19,29H,2-3,6-12H2,1H3
InChIKey :PMXMIIMHBWHSKN-UHFFFAOYSA-N
SMILES :C12C(O)CCCN1C(=O)C(CCN1CCC(C3C4=C(ON=3)C=C(F)C=C4)CC1)=C(C)N=2
CAS DataBase Reference :144598-75-4(CAS DataBase Reference)
Safety Information
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| Signal word: | Danger | ||||||||||||||
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Description
Paliperidone is a potent antagonist of dopamine receptors (IC50s = 1.0 and 0.9 nM for D2 and D3, respectively). It also avidly binds α1- and α2-adrenergic receptors, histamine H1 receptor, and serotonin (5-HT) receptors 5-HT1D and 5-HT2A (Kis = 10, 80, 3.4, 19, 1.2 nM, respectively). Paliperidone is also known as 9-hydroxy risperidone and is the major metabolite of the antipsychotic medication risperidone .Related product price
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Suppliers and manufacturers
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Sinoway Industrial co., ltd.
Aceschem Inc.
Capot Chemical Co.,Ltd.
Henan Tianfu Chemical Co.,Ltd.
Nanjing ChemLin Chemical Industry Co., Ltd.
Lianyungang happen teng technology co., LTD
Tianjin Huiren Chemtech Co., Ltd
Paliperidone
CAS:144598-75-4
