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928037-13-2 Basic information More..
Product Name:Golvatinib (E7050)
Synonyms:N-[2-Fluoro-4-[[2-[[[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl]amino]pyridin-4-yl]oxy];E-7050N-[2-Fluoro-4-[[2-[[[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl]amino]pyridin-4-yl]oxy]phenyl]-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide;E-7050;N-[2-Fluoro-4-[[2-[[[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl]amino]pyridin-4-yl]oxy]phenyl]-N'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide;Golvatinib;E-7050 (Golvatinib);Golvatinib (E7050);1,1-Cyclopropanedicarboxamide, N-[2-fluoro-4-[[2-[[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]amino]-4-pyridinyl]oxy]phenyl]-N'-(4-fluorophenyl)-
CAS:928037-13-2
MF:C33H37F2N7O4
MW:633.69
EINECS:
Mol File:928037-13-2.mol
928037-13-2

Use

Golvatinib (E7050) is a dual c-Met and VEGFR-2 inhibitor with IC50 of 14 nM and 16 nM, does not inhibit bFGF-stimulated HUVEC growth (up to 1000 nM). Phase 1/2.

Golvatinib (E7050) manufacturers

  • Golvatinib
  • $61.00
  • 2026-04-22
  • CAS:928037-13-2
  • Purity: 99.50%
  • Supply Ability: 10g
  • Golvatinib (E7050)
  • 2025-04-04
  • CAS:928037-13-2
  • Min. Order: 1KG
  • Purity: 98%
  • Supply Ability: 1Ton
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Products Intro: Product Name: 1-N'-[2-fluoro-4-[2-[[4-(4-methylpiperazin-1-yl)piperidine-1-carbonyl]amino]pyridin-4-yl]oxyphenyl]-1-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide
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