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Pharmaceutical intermediates

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Structure Chemical Name CAS MF
2-isopropyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-isopropyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2223043-76-1 C13H21BN2O2
2-Methoxy-4-(3-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2-Methoxy-4-(3-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2222997-02-4 C19H30BNO3
2-Methoxy-4-(4-methylimidazol-yl)phenylboronic acid pinacol ester 2-Methoxy-4-(4-methylimidazol-yl)phenylboronic acid pinacol ester 2223031-35-2 C17H23BN2O3
2-Methyl-5-(piperidino)furan-3-boronic acid pinacol ester 2-Methyl-5-(piperidino)furan-3-boronic acid pinacol ester 2223042-98-4 C16H26BNO3
2-Trifluoromethyl-4-(3-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2-Trifluoromethyl-4-(3-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2222996-39-4 C19H27BF3NO2
3-(3-Tolyl)pyridine-2-boronic acid pinacol ester 3-(3-Tolyl)pyridine-2-boronic acid pinacol ester 2223044-59-3 C18H22BNO2
3-(tert-Butoxy)pyridine-2-boronic acid pinacol ester 3-(tert-Butoxy)pyridine-2-boronic acid pinacol ester 2223047-07-0 C15H24BNO3
3-(Trifluoromethyl)-4-(4-tetrahydropyranyl)phenylboronic acid pinacol ester 3-(Trifluoromethyl)-4-(4-tetrahydropyranyl)phenylboronic acid pinacol ester 2223052-48-8 C18H24BF3O3
3,4-DI(PYRIDIN-4-YL)PYRIDINE 3,4-DI(PYRIDIN-4-YL)PYRIDINE 1214336-71-6 C15H11N3
3-Amino-6-(pyrrolidino)pyridine-4-boronic acid pinacol ester 3-Amino-6-(pyrrolidino)pyridine-4-boronic acid pinacol ester 2223042-96-2 C15H24BN3O2
3-Bromo-2-amino-5-(piperidino)pyridine 3-Bromo-2-amino-5-(piperidino)pyridine 1381933-80-7 C10H14BrN3
3-Chloro-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 3-Chloro-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 2223031-97-6 C22H33BClNO4
3-Methyl-4-(2-methylpiperidin-1-yl)phenylboronic acid pinacol ester 3-Methyl-4-(2-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2222996-36-1 C19H30BNO2
3-Trifluoromethyl-4-(2-methylimidazol-1-yl)phenylboronic acid pinacol ester 3-Trifluoromethyl-4-(2-methylimidazol-1-yl)phenylboronic acid pinacol ester 2223050-45-9 C17H20BF3N2O2
4-(2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4-(trifluoromethyl)phenyl)piperidine 4-(2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4-(trifluoromethyl)phenyl)piperidine 2223032-97-9 C18H25BF3NO2
4-(2-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(2-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223049-93-0 C20H30BNO2
4-(2-Methylimidazol-1-yl)thiophene-2-boronic acid pinacol ester 4-(2-Methylimidazol-1-yl)thiophene-2-boronic acid pinacol ester 2223033-41-6 C14H19BN2O2S
4-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethyl)phenyl)piperidine 4-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethyl)phenyl)piperidine 2223043-45-4 C18H25BF3NO2
4-(3-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(3-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223049-94-1 C17H25BFNO2
4-(4-cyclopropyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(4-cyclopropyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223031-93-2 C20H30BNO2
4-(4-Methyl-1H-pyrazol-1-yl)thiophene-2-boronic acid pinacol ester 4-(4-Methyl-1H-pyrazol-1-yl)thiophene-2-boronic acid pinacol ester 2223039-98-1 C14H19BN2O2S
4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl)thiazole 4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl)thiazole 1402166-17-9 C13H16BN3O2S
4-(6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl)thiazole 4-(6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl)thiazole 1402166-18-0 C13H16BN3O2S
4-(Imidazol-1-yl)thiophene-2-boronic acid pinacol ester 4-(Imidazol-1-yl)thiophene-2-boronic acid pinacol ester 2223032-27-5 C13H17BN2O2S
4-(iso-Propyl)pyridine-3-boronic acid pinacol ester 4-(iso-Propyl)pyridine-3-boronic acid pinacol ester 2096342-29-7 C14H22BNO2
4-(tetrahydro-2H-pyran-4-yl)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 4-(tetrahydro-2H-pyran-4-yl)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2223029-97-6 C17H26BNO3
4,4,5,5-tetramethyl-2-(3-(tetrahydro-2H-pyran-3-yl)-4-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(3-(tetrahydro-2H-pyran-3-yl)-4-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 2223003-93-6 C18H24BF3O3
4,4,5,5-tetramethyl-2-(4-methyl-2-(tetrahydro-2H-pyran-3-yl)phenyl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(4-methyl-2-(tetrahydro-2H-pyran-3-yl)phenyl)-1,3,2-dioxaborolane 2223004-36-0 C18H27BO3
4,4,5,5-tetramethyl-2-(5-(tetrahydro-2H-pyran-3-yl)-2-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(5-(tetrahydro-2H-pyran-3-yl)-2-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 2222996-47-4 C18H24BF3O3
4-Amino-2-(1H-pyrazol-1-yl)thiazole 4-Amino-2-(1H-pyrazol-1-yl)thiazole 1314353-38-2 C6H6N4S
4-Amino-2-(iso-propyl)-6-(tert-butoxy)pyrimidine 4-Amino-2-(iso-propyl)-6-(tert-butoxy)pyrimidine 1412956-90-1 C11H19N3O
4-amino-2-cyclopropyl-6-ethylpyrimidine 4-amino-2-cyclopropyl-6-ethylpyrimidine 1247445-04-0 C9H13N3
4-Amino-2-fluoro-6-cyclopropylpyridine 4-Amino-2-fluoro-6-cyclopropylpyridine 1622842-96-9 C8H9FN2
4-amino-6-(3-chlorophenyl)-2-methylpyrimidine 4-amino-6-(3-chlorophenyl)-2-methylpyrimidine 1250795-52-8 C11H10ClN3
4-Bromo-1,2-diethylimidazole 4-Bromo-1,2-diethylimidazole 1622843-94-0 C7H11BrN2
4-Bromo-1-cyclopentyl-2-ethylimidazole 4-Bromo-1-cyclopentyl-2-ethylimidazole 1622840-39-4 C10H15BrN2
4-Bromo-2-(1H-pyridin-2-one)thiazole 4-Bromo-2-(1H-pyridin-2-one)thiazole 959239-58-8 C8H5BrN2OS
4-Bromo-2-(2-furyl)pyrimidine 4-Bromo-2-(2-furyl)pyrimidine 1086381-91-0 C8H5BrN2O
4-Bromo-2-(N,N-diethylamino)pyrimidine 4-Bromo-2-(N,N-diethylamino)pyrimidine 959240-66-5 C8H12BrN3
4-Bromo-2-fluoro-6-(piperidin-3-yl)pyridine 4-Bromo-2-fluoro-6-(piperidin-3-yl)pyridine 1622834-23-4 C10H12BrFN2
4-Bromo-6-(tert-butyl)-2-methylpyrimidine 4-Bromo-6-(tert-butyl)-2-methylpyrimidine 1412954-96-1 C9H13BrN2
4-chloro-2-(1,4-dioxan-2-yl)pyrimidine 4-chloro-2-(1,4-dioxan-2-yl)pyrimidine 1479797-77-7 C8H9ClN2O2
4-Chloro-2-(3-fluorophenyl)pyrimidine 4-Chloro-2-(3-fluorophenyl)pyrimidine 76128-70-6 C10H6ClFN2
4-Chloro-2-cyclopropyl-6-(3-furyl)pyrimidine 4-Chloro-2-cyclopropyl-6-(3-furyl)pyrimidine 1412954-57-4 C11H9ClN2O
4-chloro-2-methyl-6-(1H-imidazol-1-yl)pyrimidine 4-chloro-2-methyl-6-(1H-imidazol-1-yl)pyrimidine 1250182-02-5 C8H7ClN4
4-fluoro-2-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 4-fluoro-2-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2223033-80-3 C12H17BFNO3
4-Iodo-2-chloro-6-fluoropyridine 4-Iodo-2-chloro-6-fluoropyridine 1622843-82-6 C5H2ClFIN
4-methyl-1-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethyl)phenyl)piperidine 4-methyl-1-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethyl)phenyl)piperidine 2223041-05-0 C19H27BF3NO2
4-Methyl-5-(iso-propyl)pyridine-3-boronic acid pinacol ester 4-Methyl-5-(iso-propyl)pyridine-3-boronic acid pinacol ester 2223046-84-0 C15H24BNO2
4-Methyl-6-cyclopropylpyridine-3-boronic acid pinacol ester 4-Methyl-6-cyclopropylpyridine-3-boronic acid pinacol ester 2223036-25-5 C15H22BNO2
5-(2-Aminopyrimidyl)pyridine-2-boronic acid pinacol ester 5-(2-Aminopyrimidyl)pyridine-2-boronic acid pinacol ester 2223047-90-1 C15H19BN4O2
5-(2-Chlorophenyl)pyridine-3-boronic acid pinacol ester 5-(2-Chlorophenyl)pyridine-3-boronic acid pinacol ester 1402227-42-2 C17H19BClNO2
5-(2-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 5-(2-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 2223003-34-5 C16H26BNO2S
5-(3-Methyl-1H-pyrazol-1-yl)furan-2-boronic acid pinacol ester 5-(3-Methyl-1H-pyrazol-1-yl)furan-2-boronic acid pinacol ester 2223046-02-2 C14H19BN2O3
5-(3-Tolyl)-2-hydroxypyrazine 5-(3-Tolyl)-2-hydroxypyrazine 1159818-33-3 C11H10N2O
5-(4-Fluoro-2-methylphenyl)-2-hydroxypyrazine 5-(4-Fluoro-2-methylphenyl)-2-hydroxypyrazine 1159816-55-3 C11H9FN2O
5-(4-Methylpiperidin-1-yl)furan-2-boronic acid pinacol ester 5-(4-Methylpiperidin-1-yl)furan-2-boronic acid pinacol ester 2223054-63-3 C16H26BNO3
5-(N-Methylpiperazin-1-yl)thiophene-2-boronic acid pinacol ester 5-(N-Methylpiperazin-1-yl)thiophene-2-boronic acid pinacol ester 2223033-64-3 C15H25BN2O2S
5-(tetrahydro-2H-pyran-4-yl)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 5-(tetrahydro-2H-pyran-4-yl)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2223054-65-5 C17H26BNO3
5-Amino-2-(1H-pyrazol-1-yl)pyrimidine 5-Amino-2-(1H-pyrazol-1-yl)pyrimidine 1211587-33-5 C7H7N5
5-Amino-2-(3-methylpiperidin-1-yl)thiazole 5-Amino-2-(3-methylpiperidin-1-yl)thiazole 1314354-61-4 C9H15N3S
5-Amino-2-(4-methylpiperidin-1-yl)thiazole 5-Amino-2-(4-methylpiperidin-1-yl)thiazole 1314355-52-6 C9H15N3S
5-Amino-2-(cyclobutyl)pyrimidine 5-Amino-2-(cyclobutyl)pyrimidine 1260833-10-0 C8H11N3
5-Amino-2-(N-methylpiperazin-1-yl)thiazole 5-Amino-2-(N-methylpiperazin-1-yl)thiazole 1314355-58-2 C8H14N4S
5-Amino-2-(pyrrolidino)thiazole 5-Amino-2-(pyrrolidino)thiazole 1314355-61-7 C7H11N3S
5-Bromo-2-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 5-Bromo-2-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2223042-75-7 C15H18BBrN2O2
5-Bromo-2-(3-pyridyl)pyrimidine 5-Bromo-2-(3-pyridyl)pyrimidine 1240594-99-3 C9H6BrN3
5-Bromo-2-(piperidin-4-ol)thiazole 5-Bromo-2-(piperidin-4-ol)thiazole 959239-73-7 C8H11BrN2OS
5-Bromo-6-(2-methylimidazol-1-yl)pyridine-3-boronic acid pinacol ester 5-Bromo-6-(2-methylimidazol-1-yl)pyridine-3-boronic acid pinacol ester 1352574-50-5 C15H19BBrN3O2
5-Bromo-6-(2-trifluoromethylphenyl)pyridine-3-boronic acid pinacol ester 5-Bromo-6-(2-trifluoromethylphenyl)pyridine-3-boronic acid pinacol ester 2223052-29-5 C18H18BBrF3NO2
5-Bromo-6-(iso-propoxy)pyridine-3-boronic acid pinacol ester 5-Bromo-6-(iso-propoxy)pyridine-3-boronic acid pinacol ester 2223054-45-1 C14H21BBrNO3
5-Bromo-6-diethylaminopyridine-3-boronic acid pinacol ester 5-Bromo-6-diethylaminopyridine-3-boronic acid pinacol ester 1352756-86-5 C15H24BBrN2O2
5-Bromo-6-phenylpyridine-3-boronic acid pinacol ester 5-Bromo-6-phenylpyridine-3-boronic acid pinacol ester 2223030-66-6 C17H19BBrNO2
5-Methyl-2-(cyclobutyl)pyridine-4-boronic acid pinacol ester 5-Methyl-2-(cyclobutyl)pyridine-4-boronic acid pinacol ester 2223030-15-5 C16H24BNO2
5-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 5-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 2223033-72-3 C13H17BN2O2
5-Methyl-4-methoxypyridine-3-boronic acid pinacol ester 5-Methyl-4-methoxypyridine-3-boronic acid pinacol ester 2223050-91-5 C13H20BNO3
6-(3-Fluorophenyl)pyrazine-2-boronic acid pinacol ester 6-(3-Fluorophenyl)pyrazine-2-boronic acid pinacol ester 1402172-95-5 C16H18BFN2O2
6-(4-Fluoro-2-methylphenyl)pyrazine-2-boronic acid pinacol ester 6-(4-Fluoro-2-methylphenyl)pyrazine-2-boronic acid pinacol ester 1402227-33-1 C17H20BFN2O2
6-(4-tert-Butylphenyl)pyrazine-2-boronic acid pinacol ester 6-(4-tert-Butylphenyl)pyrazine-2-boronic acid pinacol ester 1402233-49-1 C20H27BN2O2
6-(N,N-Methylethylamino)-2-bromopyridine 6-(N,N-Methylethylamino)-2-bromopyridine 959237-79-7 C8H11BrN2
6-(tert-butyl)-2-fluoro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 6-(tert-butyl)-2-fluoro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2223036-07-3 C15H23BFNO2
6-Bromo-5-methylpyridine-2-boronic acid pinacol ester 6-Bromo-5-methylpyridine-2-boronic acid pinacol ester 2223049-06-5 C12H17BBrNO2
methyl 6-(1-(tert-butoxycarbonyl)piperidin-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate methyl 6-(1-(tert-butoxycarbonyl)piperidin-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 2223009-62-7 C23H35BN2O6
N,N-diethyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-amine N,N-diethyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-amine 1310404-61-5 C14H24BN3O2
tert-butyl (5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl)carbamate tert-butyl (5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl)carbamate 1402227-80-8 C15H24BN3O4
tert-butyl 4-(3-(methoxycarbonyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate tert-butyl 4-(3-(methoxycarbonyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate 2256709-03-0 C24H36BNO6
tert-butyl 4-(3-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate tert-butyl 4-(3-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate 2256708-93-5 C22H33BFNO4
tert-butyl 4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazol-2-yl)piperazine-1-carboxylate tert-butyl 4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazol-2-yl)piperazine-1-carboxylate 1344124-61-3 C18H30BN3O4S
tert-butyl 4-bromo-1H-imidazole-1-carboxylate-2,5-d2 tert-butyl 4-bromo-1H-imidazole-1-carboxylate-2,5-d2 1622844-09-0 C8H11BrN2O2
4-Bromo-5-chloro-1H-pyridin-2-one 4-Bromo-5-chloro-1H-pyridin-2-one 1227587-31-6 C5H3BrClNO
(4-(1H-pyrazol-1-yl-d3)phenyl-2,3,5,6-d4)boronic acid (4-(1H-pyrazol-1-yl-d3)phenyl-2,3,5,6-d4)boronic acid 2256709-40-5 C9H2BD7N2O2
(5-(4-(methyl-d3)piperazin-1-yl-2,2,3,3,5,5,6,6-d8)thiophen-2-yl)boronic acid (5-(4-(methyl-d3)piperazin-1-yl-2,2,3,3,5,5,6,6-d8)thiophen-2-yl)boronic acid 2256709-47-2 C9H4BD11N2O2S
1-(2-(methoxy-d3)phenyl-3,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 1-(2-(methoxy-d3)phenyl-3,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 2256711-05-2 C16H12BD9N2O3
1-(2-bromophenyl)-1H-imidazol-2-amine 1-(2-bromophenyl)-1H-imidazol-2-amine 1695937-66-6 C9H8BrN3
1-(2-bromophenyl)-4-(methyl-d3)-1H-pyrazole-3,5-d2 1-(2-bromophenyl)-4-(methyl-d3)-1H-pyrazole-3,5-d2 2256712-41-9 C10H4BrD5N2
1-(2-fluorophenyl)-1H-imidazol-2-amine 1-(2-fluorophenyl)-1H-imidazol-2-amine 1698842-02-2 C9H8FN3
1-(3-(methoxy-d3)phenyl-2,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-3,5-d2 1-(3-(methoxy-d3)phenyl-2,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-3,5-d2 2256711-09-6 C16H21BN2O3
1-(3-(trifluoromethyl)phenyl)-1,3-dihydro-2H-imidazol-2-one 1-(3-(trifluoromethyl)phenyl)-1,3-dihydro-2H-imidazol-2-one 1526594-45-5 C10H7F3N2O
1-(3-bromo-5-cyclopropylphenyl)piperazine 1-(3-bromo-5-cyclopropylphenyl)piperazine 2222934-83-8 C13H17BrN2
1-(3-bromophenyl)-2-(methyl-d3)-1H-imidazole-4,5-d2 1-(3-bromophenyl)-2-(methyl-d3)-1H-imidazole-4,5-d2 2256712-57-7 C10H4BrD5N2
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