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Epigenetic Reader Domain inhibitors

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Structure Chemical Name CAS MF
(+)-JQ-1 (+)-JQ-1 1268524-70-4 C23H25ClN4O2S
I-BET151 (GSK1210151A) I-BET151 (GSK1210151A) 1300031-49-5 C23H21N5O3
RVX-208 RVX-208 1044870-39-4 C20H22N2O5
PFI-1 PFI-1 1403764-72-6 C16H17N3O4S
GSK 525762A GSK 525762A 1260907-17-2 C22H22ClN5O2
OTX015 OTX015 202590-98-5 C25H22ClN5O2S
SGC-CBP30 SGC-CBP30 1613695-14-9 C28H33ClN4O3
BroMosporine BroMosporine 1619994-69-2 C17H20N6O4S
UNC 669 UNC 669 1314241-44-5 C15H20BrN3O
MS436 MS436 1395084-25-9 C18H17N5O3S
GSK1324726A (I-BET726) GSK1324726A (I-BET726) 1300031-52-0 C25H23ClN2O3
PFI3 PFI3 1819363-80-8 C19H19N3O2
CPI-203 CPI-203 1446144-04-2 C19H18ClN5OS
OF-1 OF-1 919973-83-4 C17H18BrN3O4S
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