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阻害剤活性化剤

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Structure Chemical Name CAS MF
RNasin Inhibitor (Ribonuclease Inhibitor)) RNasin Inhibitor (Ribonuclease Inhibitor))
ZOTAROLIMUS (MTOR inhibitor) ZOTAROLIMUS (MTOR inhibitor)
SRT 2104 (SIRT1 activator) SRT 2104 (SIRT1 activator)
SPERMIDINE (NNOS inhibitor) SPERMIDINE (NNOS inhibitor)
ROSCOVITINE (SELICICLIB, CYC202) (CDK2 inhibitor) ROSCOVITINE (SELICICLIB, CYC202) (CDK2 inhibitor)
PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist) PURMORPHAMINE (HEDGEHOG/SMOOTHENED agonist)
PONATINIB (SRC-ABL inhibitor) PONATINIB (SRC-ABL inhibitor)
OBATOCLAX MESYLATE (BCL-2 inhibitor) OBATOCLAX MESYLATE (BCL-2 inhibitor)
LEDIPASVIR (HCV PROTEASE INHIBITOR) LEDIPASVIR (HCV PROTEASE INHIBITOR)
FIPI (PLD1/2 inhibitor) FIPI (PLD1/2 inhibitor)
ENMD-2076 (FLT3 inhibitor) ENMD-2076 (FLT3 inhibitor)
DALCETRAPIB (CETP inhibitor) DALCETRAPIB (CETP inhibitor)
CH5183284 (FGFR inhibitor) CH5183284 (FGFR inhibitor)
CAL-101 (PI3K inhibitor) CAL-101 (PI3K inhibitor)
BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist) BREXPIPRAZOLE (DOPAMINE RECEPTOR agonist)
BLU-9931 (FGFR inhibitor) BLU-9931 (FGFR inhibitor)
BEDAQUILINE (anti-tuberculosis mycobacteria) BEDAQUILINE (anti-tuberculosis mycobacteria)
AR-A014418 (GSK-3 inhibitor) AR-A014418 (GSK-3 inhibitor)
YM155 (SURVIVIN inhibitor) YM155 (SURVIVIN inhibitor)
VELIPARIB (ABT-888) (PARP1 inhibitor) VELIPARIB (ABT-888) (PARP1 inhibitor)
TIVOZANIB (VEGFR inhibitor) TIVOZANIB (VEGFR inhibitor)
TG101209 (JAK inhibitor) TG101209 (JAK inhibitor)
SRT 1720 (SIRT1 activator) SRT 1720 (SIRT1 activator)
SEMAGACESTAT (GAMMA - SECRETASE Inhibitor) SEMAGACESTAT (GAMMA - SECRETASE Inhibitor)
RIMONABANT (CANNABINOID RECEPTOR antagonist) RIMONABANT (CANNABINOID RECEPTOR antagonist)
PFI-1 (BET inhibitor) PFI-1 (BET inhibitor)
LEE011 (CDK inhibitor) LEE011 (CDK inhibitor)
ISRIB (PERK inhibitor) ISRIB (PERK inhibitor)
INH1 (MICROTUBULE ASSOCIATED inhibitor) INH1 (MICROTUBULE ASSOCIATED inhibitor)
I-BET-762 (GSK525762) (BET inhibitor) I-BET-762 (GSK525762) (BET inhibitor)
FK-506 (MTOR inhibitor) FK-506 (MTOR inhibitor)
DBEQ (P97 inhibitor) DBEQ (P97 inhibitor)
AZD4547 (FGFR inhibitor) AZD4547 (FGFR inhibitor)
AC480 (BMS-599626) (HER1 inhibitor) AC480 (BMS-599626) (HER1 inhibitor)
[oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate [oxido-(2,3,4,5,6-pentaphosphonatooxycyclohexyl)oxyphosphoryl] phosphate 193743-89-4
EG-011 EG-011 2377113-41-0 C28H26N4O4
(1E,4E)-1,5-ビス(2-メトキシフェニル)-1,4-ペンタジエン-3-オン (1E,4E)-1,5-ビス(2-メトキシフェニル)-1,4-ペンタジエン-3-オン 39777-61-2 C19H18O3
WS3 (IΚB/IKK inhibitor) WS3 (IΚB/IKK inhibitor)
PND-1186 (FAK inhibitor) PND-1186 (FAK inhibitor)
PI-103 (PI3K inhibitor) PI-103 (PI3K inhibitor)
PFI-4 (EPIGENETIC READER DOMAIN inhibitor) PFI-4 (EPIGENETIC READER DOMAIN inhibitor)
PANOBINOSTAT (LBH589) (HDAC inhibitor) PANOBINOSTAT (LBH589) (HDAC inhibitor)
OSELTAMIVIR ACID (NEURAMINIDASE Inhibitor) OSELTAMIVIR ACID (NEURAMINIDASE Inhibitor)
NU-7441 (DNA-PK inhibitor) NU-7441 (DNA-PK inhibitor)
MG-132 (PROTEASOME Inhibitor) MG-132 (PROTEASOME Inhibitor)
MASITINIB (C-KIT inhibitor) MASITINIB (C-KIT inhibitor)
IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor) IXAZEOMIB (MLN2238) (20S PROTEASOME Inhibitor)
ICOTINIB HCL (EGFR inhibitor) ICOTINIB HCL (EGFR inhibitor)
HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride HYDROXYLAMINE HYDROCHLORIDE/Hydroxylamine Hydrochloride Cl2H8N2O2
EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor) EPOTHILONE B (MICROTUBULE ASSOSIATED inhibitor)
E-64 (CYSTEINE PROTEASE inhibitor) E-64 (CYSTEINE PROTEASE inhibitor)
DOCETAXEL (MICROTUBULE ASSOSIATED inhibitor) DOCETAXEL (MICROTUBULE ASSOSIATED inhibitor)
DEGRASYN (BCR-ABL inhibitor) DEGRASYN (BCR-ABL inhibitor)
CC-223 (MTOR inhibitor) CC-223 (MTOR inhibitor)
BI2536 (PLK inhibitor) BI2536 (PLK inhibitor)
A83-01 (ALK5 inhibitor) A83-01 (ALK5 inhibitor)
A-366 (HISTONE METHYLTRANSFERASE Inhibitor) A-366 (HISTONE METHYLTRANSFERASE Inhibitor)
ICA 069673 ICA 069673 582323-16-8 C11H6ClF2N3O
VOLASERTIB (PLK inhibitor) VOLASERTIB (PLK inhibitor)
TUBASTATIN A (HDAC inhibitor) TUBASTATIN A (HDAC inhibitor)
TEDIZOLID (MAO-A inhibitor) TEDIZOLID (MAO-A inhibitor)
SP600125 (JNK inhibitor) SP600125 (JNK inhibitor)
SB203580 (P38 MAPK Inhibitor) SB203580 (P38 MAPK Inhibitor)
SALIRASIB (RHO inhibitor) SALIRASIB (RHO inhibitor)
RG108 (DNA METHYLTRANSFERASE inhibitor) RG108 (DNA METHYLTRANSFERASE inhibitor)
PLERIXAFOR (CXCR inhibitor) PLERIXAFOR (CXCR inhibitor)
PD-173955 (BCR-ABL inhibitor) PD-173955 (BCR-ABL inhibitor)
ODANACATIB (CYSTEINE PROTEASE inhibitor) ODANACATIB (CYSTEINE PROTEASE inhibitor)
MI-2 (HISTONE METHYLTRANSFERASE Inhibitor) MI-2 (HISTONE METHYLTRANSFERASE Inhibitor)
GSK1278863 (HIF inhibitor) GSK1278863 (HIF inhibitor)
DACOMITINIB (EGFR inhibitor) DACOMITINIB (EGFR inhibitor)
BATIMASTAT (MMP inhibitor) BATIMASTAT (MMP inhibitor)
AVASIMIBE (P450 inhibitor) AVASIMIBE (P450 inhibitor)
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