| Company Name: |
TargetMol Chemicals Inc.
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| Tel: |
15002134094 |
| Email: |
marketing@targetmol.cn |
| Products Intro: |
Product Name:HSP90-IN-13 CAS:2446055-29-2 Package:25mg/RMB 10600;50mg/RMB 13800;100mg/RMB 17500
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Benzoic acid, 3-[4-[[[3,4-dihydro-6-methyl-4-oxo-3-(phenylmethyl)-2-quinazolinyl]thio]methyl]-1H-1,2,3-triazol-1-yl]- manufacturers
- HSP90-IN-13
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- $1520.00
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2026-07-27
- CAS:2446055-29-2
- Purity:
- Supply Ability: 10g
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| | Benzoic acid, 3-[4-[[[3,4-dihydro-6-methyl-4-oxo-3-(phenylmethyl)-2-quinazolinyl]thio]methyl]-1H-1,2,3-triazol-1-yl]- Basic information |
| | Benzoic acid, 3-[4-[[[3,4-dihydro-6-methyl-4-oxo-3-(phenylmethyl)-2-quinazolinyl]thio]methyl]-1H-1,2,3-triazol-1-yl]- Chemical Properties |
| Boiling point | 768.6±70.0 °C(Predicted) | | density | 1.38±0.1 g/cm3(Predicted) | | pka | 3.75±0.10(Predicted) |
| | Benzoic acid, 3-[4-[[[3,4-dihydro-6-methyl-4-oxo-3-(phenylmethyl)-2-quinazolinyl]thio]methyl]-1H-1,2,3-triazol-1-yl]- Usage And Synthesis |
| Uses | HSP90-IN-13 (compound 5k) is a highly potent HSP90 pan inhibitor with an IC50 value of 25.07 nM. HSP90-IN-13 has multi-target activity against EGFR, VEGFR-2 and Topoisomerase-2. HSP90-IN-13 causes cell cycle arrest at G2/M phase and induces apoptosis of MCF-7 cells through mitochondrial-mediated pathway[1]. | | IC 50 | HSP90: 25.07 nM (IC50); Topoisomerase-2: 25.85 nM (IC50); EGFR: 38.5 nM (IC50); VEGFR-2: 126.95 nM (IC50) | | References | [1] El-Shafey HW, et al. Synthetic approaches, anticancer potential, HSP90 inhibition, multitarget evaluation, molecular modeling and apoptosis mechanistic study of thioquinazolinone skeleton: Promising antibreast cancer agent. Bioorg Chem. 2020 Aug;101:10398 DOI:10.1016/j.bioorg.2020.103987 |
| | Benzoic acid, 3-[4-[[[3,4-dihydro-6-methyl-4-oxo-3-(phenylmethyl)-2-quinazolinyl]thio]methyl]-1H-1,2,3-triazol-1-yl]- Preparation Products And Raw materials |
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