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(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol

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CAS:22972-51-6
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(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol manufacturers

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  • 2026-07-22
  • CAS:22972-51-6
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(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol Basic information
Product Name:(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol
Synonyms:(+)-(1S,4R)-P-MENTHA-2,8-DIEN-1-OL;(1S,4R)-1-methyl-4-prop-1-en-2-ylcyclohex-2-en-1-ol;(1S,4R)-p-Menth-2,8-dien-1-ol;(1S,4R)-1-Methyl-4-(prop-1-en-2-yl)cyclohex-2-eno;(1S,4S)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-en-1-ol;(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-en-1-ol22972-51-6;(1S,4R)-1-Methyl-4-(prop-1-en-2-yl)cyclohex-2-en-1-ol 97+%;(1S,4R)-1-Methyl-4-(1-propen-2-yl)-2-cyclohexenol
CAS:22972-51-6
MF:C10H16O
MW:152.23
EINECS:805-440-4
Product Categories:
Mol File:22972-51-6.mol
(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol Structure
(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol Chemical Properties
Boiling point 69-70 °C(Press: 3 Torr)
density 0.9398
Fp 87.0±19.6 °C
storage temp. 2-8°C
solubility Chloroform (Soluble), Methanol (Soluble)
pka14.66±0.40(Predicted)
form Oil
color Colourless
Optical Rotation-0.11° (C=1.00 g/100ml, CHCL3)
Water Solubility 4.2g/L
Stability:Light Sensitive
InChIInChI=1S/C10H16O/c1-8(2)9-4-6-10(3,11)7-5-9/h4,6,9,11H,1,5,7H2,2-3H3/t9-,10+/m0/s1
InChIKeyMKPMHJQMNACGDI-VHSXEESVSA-N
SMILES[C@@]1(C)(O)CC[C@@H](C(C)=C)C=C1
LogP2.82
Safety Information
HS Code 2906190090
MSDS Information
(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol Usage And Synthesis
Uses (1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol is an acetal reagent used in the synthesis of desoxy cannabidiols and THC (T293202) related psychoactive compounds. It is formed from (+)-Limonene using a photosynthesized O2 transfer.
DefinitionChEBI: (1S,4R)-p-Mentha-2,8-dien-1-ol is a p-menthane monoterpenoid.
Hazard(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol causes skin irritation and serious eye irritation. It may cause respiratory irritation.
Synthesis
Cyclohexanol, 2-(dimethyloxidoamino)-1-methyl-4-(1-methylethenyl)-, (1S,2S,4R)-

1415961-21-5

(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol

22972-51-6

The 1S,2S,5R-N,N,2-trimethyl-2-hydroxy-5-isopropenylcyclohexylamine oxide (1.430 g, 6.7 mmol) was heated in a Kugelrohr oven at 180 °C under 1 mmHg vacuum until the solid residue completely disappeared. The yellow distillate (1.317 g) was collected and purified by fast chromatography (ether:hexane=2:3) to afford the target product (1S,4R)-1-methyl-4-(1-methylethenyl)-2-cyclohexen-1-ol (0.752 g, 74% yield) as a colorless oil. the Rf value was 0.32 (ether:hexane=2:3); the specific optical rotation [α]D26: +60 (c=1.0, CHCl3), consistent with literature value [α]D23: +53.8 (CHCl3); IR spectrum (SeZn) showed absorption peaks: 3354 (medium, broad, O-H), 2967 (medium, C-H), 2935 (medium, CH), 2861 (medium, CH), 1644 (medium, C=C), 1105 (strong, CO), and 888 (strong, C=CH bent), 736 (strong, C=CH bent) cm-1; 1H NMR (500 MHz, CDCl3) chemical shift: δ 5.70 (1H, ddd, 3JH2-H3=10.0 Hz, 4JH2-H4=2.4 Hz, 4JH2-H6=1.4 Hz, H2), 5.65 (1H, ddd. 3JH3-H2=10.0 Hz, 3JH3-H4=2.4 Hz, 4JH3-H5=0.8 Hz, H3), 4.78 (1H, quin, 4JH9b-H10≈4JH9b-H4=1.6 Hz, H9b), 4.74 (1H, quin, 4JH9a-H10≈4JH9a-H4=0.88 Hz, H9a), 2.65 (1H, m, H4), 1.88-1.73 (2H, m, H5eq, H6eq), 1.73 (3H, s, H10), 1.66-1.51 (3H, m, H5ax, H6ax, OH), 1.29 (3H, s, H7) ppm; 13C NMR (125 MHz, CDCl3) chemical shift : 148.3 (C8), 134.1 (C2), 132.3 (C3), 110.7 (C9), 67.6 (C1), 43.6 (C4), 36.9 (C6), 29.6 (C7), 25.0 (C5), 21.0 (C10) ppm; low resolution mass spectra (GC-MS): m/z 152 (M+, 2%), 134 ( [M-H2O]+, 11%), 119 ([M-CH3-H2O]+, 32%), 91 (100%), 79 (37%), 77 (46%); Elemental analysis (C10H16O) Calculated values: C 78.90, H 10.59; Measured values: C 78.25, H 10.59, N < 0.05.

References[1] Tetrahedron Letters, 2013, vol. 54, # 1, p. 52 - 54
Tag:(1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol(22972-51-6) Related Product Information
trans-4-Aminocyclohexanemethanol N,N-DIETHYLBENZAMIDE 2-Methylindole Adenosine 3-METHYLSTYRENE VINYL PROPIONATE Methoxyethene (1R)-(+)-TRANS-ISOLIMONENE (4R)-1-METHYL-4-(1-METHYLETHENYL)-2-CYCLOHEXEN-1-OL (1S,4R)-1-methyl-4-(prop-1-en-2-yl)cyclohex-2-enol