| Company Name: |
Beijing Jin Ming Biotechnology Co., Ltd.
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| Tel: |
010-60605840 18892239720 |
| Email: |
psaitong@jm-bio.com |
| Products Intro: |
Product Name:Cyclooctyne-O-amido-PEG3-PFP ester CAS:2101206-33-9 Package:100mg;250mg;500mg
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| Company Name: |
MedChemExpress
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| Tel: |
021-58955995 |
| Email: |
sales@medchemexpress.com |
| Products Intro: |
Product Name:Cyclooctyne-O-amido-PEG3-PFP ester CAS:2101206-33-9
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| | Propanoic acid, 3-[2-[2-[2-[[2-(2-cyclooctyn-1-yloxy)acetyl]amino]ethoxy]ethoxy]ethoxy]-, 2,3,4,5,6-pentafluorophenyl ester Basic information |
| Product Name: | Propanoic acid, 3-[2-[2-[2-[[2-(2-cyclooctyn-1-yloxy)acetyl]amino]ethoxy]ethoxy]ethoxy]-, 2,3,4,5,6-pentafluorophenyl ester | | Synonyms: | Propanoic acid, 3-[2-[2-[2-[[2-(2-cyclooctyn-1-yloxy)acetyl]amino]ethoxy]ethoxy]ethoxy]-, 2,3,4,5,6-pentafluorophenyl ester;Cyclooctyne-O-amido-PEG3-PFP ester | | CAS: | 2101206-33-9 | | MF: | C25H30F5NO7 | | MW: | 551.5 | | EINECS: | | | Product Categories: | | | Mol File: | 2101206-33-9.mol | ![Propanoic acid, 3-[2-[2-[2-[[2-(2-cyclooctyn-1-yloxy)acetyl]amino]ethoxy]ethoxy]ethoxy]-, 2,3,4,5,6-pentafluorophenyl ester Structure](CAS/20210111/GIF/2101206-33-9.gif) |
| | Propanoic acid, 3-[2-[2-[2-[[2-(2-cyclooctyn-1-yloxy)acetyl]amino]ethoxy]ethoxy]ethoxy]-, 2,3,4,5,6-pentafluorophenyl ester Chemical Properties |
| Boiling point | 640.5±55.0 °C(Predicted) | | density | 1.31±0.1 g/cm3(Predicted) | | pka | 14.02±0.46(Predicted) |
| | Propanoic acid, 3-[2-[2-[2-[[2-(2-cyclooctyn-1-yloxy)acetyl]amino]ethoxy]ethoxy]ethoxy]-, 2,3,4,5,6-pentafluorophenyl ester Usage And Synthesis |
| Uses | Cyclooctyne-O-amido-PEG3-PFP ester is a non-cleavable 3 unit PEG ADC linker used in the synthesis of antibody-drug conjugates (ADCs)[1]. Cyclooctyne-O-amido-PEG3-PFP ester is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups. | | IC 50 | Non-cleavable Linker | | References | [1] Beck A, et al. Strategies and challenges for the next generation of antibody-drug conjugates. Nat Rev Drug Discov. 2017 May;16(5):315-337. DOI:10.1038/nrd.2016.268 |
| | Propanoic acid, 3-[2-[2-[2-[[2-(2-cyclooctyn-1-yloxy)acetyl]amino]ethoxy]ethoxy]ethoxy]-, 2,3,4,5,6-pentafluorophenyl ester Preparation Products And Raw materials |
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