CHK1-IN-3 NEW
| Price | $257 | $413 | $621 |
| Package | 2mg | 5mg | 10mg |
| Supply Ability: | 10g |
| Update Time: | 2026-07-17 |
Product Details
| Product Name: CHK1-IN-3 | CAS No.: 2097252-39-4 |
| Purity: 98.78% | Supply Ability: 10g |
| Release date: 2026/07/17 |
Product Introduction
Bioactivity
| Name | CHK1-IN-3 |
| Description | CHK1-IN-3 is an inhibitor of checkpoint kinase 1 (CHK1; IC50: 0.4 nM). |
| In vitro | CHK1-IN-3 displays a low affinity for hERG (IC50 > 40 μM). CHK1-IN-3 effectively inhibits the growth of malignant hematopathy cell lines especially Z-138 (IC50: 0.013 μM)[1]. |
| In vivo | In the Z-138 cell inoculated xenograft model, CHK1-IN-3 significantly suppresses the tumor growth as a single agent with bodyweight unaffected[1]. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | 10% DMSO+40% PEG300+5% Tween 80+45% Saline : 10 mg/mL (24.66 mM), Solution. DMSO : 150 mg/mL (369.95 mM), Sonication is recommended. 10% DMSO+90% Saline : < 10 mg/mL (24.66 mM), Lower concentrations may be soluble, but exact solubility limit is unknown. |
| Keywords | CHK1-IN-3 | CHK-1-IN-3 | CHK1IN3 | CHK1 IN 3 | Chk1 |
| Inhibitors Related | Rabusertib | CCT245737 | Tuvusertib | WAY-230563 | Prexasertib | PD0166285 | CHK1-IN-4 hydrochloride | Protein kinase inhibitor 6 | Prexasertib dihydrochloride | ANI-7 | BX795 | M2I-1 |
| Related Compound Libraries | Bioactive Compound Library | Kinase Inhibitor Library | Post-Translational Modification Compound Library | Inhibitor Library | Bioactive Compounds Library Max | Covalent Inhibitor Library | Cell Cycle Compound Library | Anti-Cancer Compound Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, USA
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