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Postion:Product Catalog >Felcisetrag
Felcisetrag
  • Felcisetrag

Felcisetrag NEW

Price $94 $238 $353
Package 1mg 5mg 10mg
Supply Ability: 10g
Update Time: 2026-04-20

Product Details

Product Name: Felcisetrag CAS No.: 916075-84-8
Purity: 99.99% Supply Ability: 10g
Release date: 2026/04/20

Product Introduction

Bioactivity

NameFelcisetrag
DescriptionFelcisetrag (TD-8954) is a potent and selective orally active 5-HT4 agonist with gastrointestinal prokinetic properties.Felcisetrag shows high affinity for the human recombinant 5-HT4(c) (h5-HT4(c)) receptor with a pKi of 9.4.
In vitroFelcisetrag induces an increase in cAMP levels in HEK-293 cells expressing the h5-HT4(c) receptor (pEC50?=?9.3) and elicits contractions in the guinea pig colonic longitudinal muscle/myenteric plexus preparation (pEC50?=?8.6). In vitro, assays demonstrate that Felcisetrag exhibits moderate intrinsic activity.[1]
In vivoThe administration of Felcisetrag (0.033?mg/kg; s.c.) results in an acceleration of carmine red dye colonic transit, leading to a decrease in excretion time.[1] A dose-dependent relaxation of the esophagus is induced by Felcisetrag (0.03~10?mg/kg; intraduodenal administration).[1] Felcisetrag (10 and 30?μg/kg; p.o) elicits an increase in contractility in the antrum, duodenum, and jejunum.[1]
StoragePowder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature.
Solubility Information10% DMSO+40% PEG300+5% Tween 80+45% Saline : 2 mg/mL (4.39 mM), Sonication is recommended.
DMSO : 45 mg/mL (98.77 mM), Sonication and heating to 60℃ are recommended.
KeywordsFelcisetrag | 5HTReceptor | 5-HT4 | 5HT Receptor
Inhibitors RelatedAlverine citrate | Sevoflurane | Dapoxetine hydrochloride | Cefaclor monohydrate | Clozapine N-Oxide | 1,8-Cineole | Dopamine hydrochloride | Cloperastine hydrochloride | Mianserin hydrochloride | Trazodone hydrochloride | Cinchonidine | Doxepin hydrochloride
Related Compound LibrariesBioactive Compound Library | Pain-Related Compound Library | Neuronal Signaling Compound Library | Membrane Protein-targeted Compound Library | ReFRAME Related Library | Anti-Cancer Clinical Compound Library | Drug Repurposing Compound Library | Bioactive Compounds Library Max | GPCR Compound Library | Anti-Cancer Compound Library | Serotonin Receptor-Targeted Compound Library | Anti-Cancer Drug Library

Company Profile Introduction

Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers. TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.

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  • Address: 36 Washington Street, Wellesley Hill, MA
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