GSK 525768A NEW
| Price | $198 | $347 | $1170 |
| Package | 2mg | 5mg | 25mg |
| Supply Ability: | 10g |
| Update Time: | 2026-05-11 |
Product Details
| Product Name: GSK 525768A | CAS No.: 1260530-25-3 |
| Supply Ability: 10g | Release date: 2026/05/11 |
Product Introduction
Bioactivity
| Name | GSK 525768A |
| Description | GSK 525768A, the inactive enantiomer of GSK525762A, exhibits no activity towards BET. |
| In vitro | GSK 525768A interacts with the protein's module by establishing hydrogen bonds with the conserved asparagine residue, effectively mimicking the acetylated lysine's binding mechanism. This interaction leads to the compound's binding deeper within the acetylated lysine's binding site, all the while preserving the position of conserved water molecules in the acetyl-lysine binding cavity's base. GSK 525768A exhibits no activity towards BET and is identified as the (R)-enantiomer of GSK525762A. Contrasting its counterpart, GSK525762A, which influences the regulation of apolipoprotein A1 (APOA1) levels in liver cell assays, GSK 525768A does not impact APOA1 release, highlighting a distinctive functional divergence between the two enantiomers. |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |
| Solubility Information | 10% DMSO+40% PEG300+5% Tween-80+45% Saline : 3.3 mg/mL (7.78 mM), Sonication is recommended. DMSO : 100 mg/mL (235.9 mM), Sonication is recommended. |
| Keywords | GSK 525768A |
| Inhibitors Related | ABBV-744 | SNDX-5613 | CeMMEC1 | 3-methyl-1,2,3,4-tetrahydroquinazolin-2-one | (+)-JQ-1 | J-147 | 5-Ph-IAA | Curcumin | dBET6 | Naphthol AS-E | JQ-1 (carboxylic acid) | Bisdemethoxycurcumin |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, USA
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