Opipramol NEW
| Price | Get Latest Price |
| Package | 1removed |
| Supply Ability: | 10g |
| Update Time: | 2026-06-11 |
Product Details
| Product Name: Opipramol | CAS No.: 315-72-0 |
| Purity: 99.98% | Supply Ability: 10g |
| Release date: 2026/06/11 |
Product Introduction
Bioactivity
| Name | Opipramol |
| Description | Opipramol (Ensidon) is a compound with antidepressant activity that attenuates cocaine-seeking behavior in a rat model of self-administration.Opipramol is a sigma (σ) receptor agonist with anxiolytic activity and may be used in the study of neurological disorders. |
| In vitro | Opipramol potently binds to the sigma recognition site with a Ki value of 50 nM. Opipramol also inhibits the uptake of [3H] dopamine in crude synaptic preparations with an IC50 value of 5.5 μM. [1] |
| In vivo | Opipramol has been shown to significantly increase dopamine release in vivo by intraperitoneal injection (dose range 5-50 mg/kg). [2] |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | DMSO : 80 mg/mL (220.08 mM), Sonication is recommended. 10% DMSO+40% PEG300+5% Tween 80+45% Saline : 3.3 mg/mL (9.08 mM), Sonication is recommended. |
| Keywords | Sigmareceptor | Sigma receptor |
| Inhibitors Related | Amitriptyline | Cutamesine dihydrochloride | L-693,403 maleate | Noscapine | Oxeladin citrate | Amitriptyline hydrochloride | S1R agonist 2 | 4-PPBP maleate | Glycerol phenylbutyrate | Sigma-1 receptor antagonist 1 | KSK67 | AB21 HCl |
| Related Compound Libraries | FDA-Approved & Pharmacopeia Drug Library | Bioactive Compound Library | Antidepressant Compound Library | Approved Drug Library | Membrane Protein-targeted Compound Library | ReFRAME Related Library | Drug Repurposing Compound Library | Bioactive Compounds Library Max | GPCR Compound Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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