| 價格 | ¥3520 | ¥812 | ¥4930 |
| 包裝 | 5mg | 1mg | 10mg |
| 最小起訂量 | 1mg |
| 發(fā)貨地 | 上海 |
| 更新日期 | 2026-06-29 |
| 中文名稱:化合物 B-HT 933 dihydrochloride | 英文名稱:B-HT 933 dihydrochloride |
| CAS:36067-72-8 | 品牌: TargetMol |
| 產地: 美國 | 保存條件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |
| 產品類別: 抑制劑 | |
| 貨號: T21787 |
| 名稱 | B-HT 933 dihydrochloride |
| 描述 | Azepexole dihydrochloride (B-HT 933), a potent and selective alpha 2-adrenoceptor agonist, exhibits affinity for α2A-, α2B-, and α2C-adrenoceptor subtypes with pKis of 8.3, 7.6, and 7.5, respectively [1]. It elicits a concentration-dependent inhibition of peristaltic contractions, evidenced by an IC50 of 78.72 nM. |
| 體外活性 | In normoglycemic rats, the sympathetically-induced vasopressor responses are dose-dependently inhibited by 1 and 3 μg/kg.min (i.v.) Azepexole dihydrochloride, with 10 and 30 μg/kg.min Azepexole dihydrochloride do not produce further inhibition. In diabetic rats, the electrically-induced vasopressor responses are: (i) unchanged by 1 and 3 μg/kg.min Azepexole dihydrochloride; (ii) significantly inhibited at all frequencies of stimulation by 10 μg/kg.min B-HT 933 dihydrochloride; and (iii) similarly inhibited (i.e. supramaximal inhibition) by 30 μg/kg.min Azepexole dihydrochloride [1]. |
| 存儲條件 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |
| 關鍵字 | B-HT-933 Dihydrochloride | B-HT933 Dihydrochloride | B-HT-933 | B-HT933 | B-HT 933 Dihydrochloride | BHT 933 dihydrochloride | B-HT 933 | B HT 933 dihydrochloride |
| 相關產品 | Trifluoperazine dihydrochloride | Buflomedil hydrochloride | Mirtazapine | Mianserin hydrochloride | Trazodone hydrochloride | Gemfibrozil | Doxepin hydrochloride | D-Mannitol | Octopamine hydrochloride | Tolazoline hydrochloride | Isoprenaline hydrochloride | Dexmedetomidine hydrochloride |
| 成立日期 | 2013-04-18 (14年) | 注冊資本 | 566.265100萬人民幣 |
| 員工人數(shù) | 100-500人 | 年營業(yè)額 | ¥ 1億以上 |
| 主營行業(yè) | 天然產物,生化試劑,分子生物學,分子砌塊,生物技術服務 | 經營模式 | 貿易,工廠,試劑,定制,服務 |
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