N2-[2-Methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-1,3,5-triazine-2,4-diamine
![N2-[2-Methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-1,3,5-triazine-2,4-diamine price.](/CAS/GIF/1097917-15-1.gif)
|
- $10 - $12210
- Product name: N2-[2-Methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-1,3,5-triazine-2,4-diamine
- CAS: 1097917-15-1
- MF: C29H40N8O3S
- MW: 580.74
- EINECS:200-258-5
- MDL Number:MFCD21609265
- Synonyms:ASP3026;ASP 3026;ASP-3026;N2-[2-Methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfon;ASP 3026;N2-[2-Methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-1,3,5-triazine-2,4-diamine;1,3,5-Triazine-2,4-diamine, N2-[2-methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-;N2-[2-Methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-1,3,5-triazine-2,4-diamine ASP 3026;ASP 3026; ASP-3026;CS-286
79 prices
Selected condition：
Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Axon Medchem
- Biorbyt Ltd
- Biosynth
- Cayman Chemical
- ChemScene
- Crysdot
- DC Chemicals
- Matrix Scientific
- Tocris
- TRC
- Usbiological
Package
- 2mg
- 10mM*1mLinDMSO
- 50
- 1g
- 1000mg
- 5g
- 100.00g
- 250.00g
- 50.00g
- 10
- 10mM*1mLinDMSO(Solid+Solvent)
- 1mg
- 10mM(in1mLDMSO)
- 5mg
- 10mg
- 25mg
- 50mg
- 200mg
- 250MG
- 100mg
- 10mM*1mLinDMSO(Solution)
- Manufactureraablocks
- Product numberAA008TAR
- Product descriptionASP3026 ≥98%
- Packaging1mg
- Price$10
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA008TAR
- Product descriptionASP3026 ≥98%
- Packaging5mg
- Price$17
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA008TAR
- Product descriptionASP3026 ≥98%
- Packaging25mg
- Price$62
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA008TAR
- Product descriptionASP3026 98+%
- Packaging50mg
- Price$99
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA008TAR
- Product descriptionASP3026
- Packaging100mg
- Price$178
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA008TAR
- Product descriptionASP3026
- Packaging200mg
- Price$254
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberT94562
- Product descriptionASP3026 98%
- Packaging100MG
- Price$235
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberT94562
- Product descriptionASP3026 98%
- Packaging100MG
- Price$235
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberT94562
- Product descriptionASP3026 98%
- Packaging250MG
- Price$470
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberT94562
- Product descriptionASP3026 98%
- Packaging250MG
- Price$470
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product numberSYN5648
- Product descriptionASP3026
- Packaging10mg
- Price$160
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0001435
- Product descriptionASP-3026 95.00%
- Packaging1MG
- Price$480
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0001435
- Product descriptionASP-3026 95.00%
- Packaging5MG
- Price$786.5
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0001435
- Product descriptionASP-3026 95.00%
- Packaging10MG
- Price$866.25
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0001435
- Product descriptionASP-3026 95.00%
- Packaging50MG
- Price$1374.45
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA3193
- Product descriptionASP3026
- Packaging50mg
- Price$300
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA008TAR | ASP3026 ≥98% | 1mg | $10 | 2026-05-28 | Buy |
| aablocks | AA008TAR | ASP3026 ≥98% | 5mg | $17 | 2026-05-28 | Buy |
| aablocks | AA008TAR | ASP3026 ≥98% | 25mg | $62 | 2026-05-28 | Buy |
| aablocks | AA008TAR | ASP3026 98+% | 50mg | $99 | 2026-05-28 | Buy |
| aablocks | AA008TAR | ASP3026 | 100mg | $178 | 2026-05-28 | Buy |
| aablocks | AA008TAR | ASP3026 | 200mg | $254 | 2026-05-28 | Buy |
| ACHEMBLOCK | T94562 | ASP3026 98% | 100MG | $235 | 2026-05-25 | Buy |
| ACHEMBLOCK | T94562 | ASP3026 98% | 100MG | $235 | 2026-05-27 | Buy |
| ACHEMBLOCK | T94562 | ASP3026 98% | 250MG | $470 | 2026-05-25 | Buy |
| ACHEMBLOCK | T94562 | ASP3026 98% | 250MG | $470 | 2026-05-27 | Buy |
| AK Scientific | SYN5648 | ASP3026 | 10mg | $160 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0001435 | ASP-3026 95.00% | 1MG | $480 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0001435 | ASP-3026 95.00% | 5MG | $786.5 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0001435 | ASP-3026 95.00% | 10MG | $866.25 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0001435 | ASP-3026 95.00% | 50MG | $1374.45 | 2021-12-16 | Buy |
| ApexBio Technology | A3193 | ASP3026 | 50mg | $300 | 2021-12-16 | Buy |
Properties
Boiling point :794.3±70.0 °C(Predicted)
Density :1.276
storage temp. :Store at -20°C
solubility :insoluble in H2O; ≥14.53 mg/mL in DMSO; ≥4.9 mg/mL in EtOH with gentle warming and ultrasonic
form :solid
pka :8.14±0.42(Predicted)
color :White to off-white
Density :1.276
storage temp. :Store at -20°C
solubility :insoluble in H2O; ≥14.53 mg/mL in DMSO; ≥4.9 mg/mL in EtOH with gentle warming and ultrasonic
form :solid
pka :8.14±0.42(Predicted)
color :White to off-white
Safety Information
| Symbol(GHS): |
|
|||||||
|---|---|---|---|---|---|---|---|---|
| Signal word: | Warning | |||||||
| Hazard statements: |
|
|||||||
| Precautionary statements: |
|
Description
ASP3026 is an ATP-competitive, second-generation ALK inhibitor (IC50 = 3.5 nM) that also inhibits ROS (IC50 = 8.9 nM) and ACK (IC50 = 5.8 nM). It inhibits neuroblastoma-activating ALK mutants F1174L (IC50 = 10 nM) and R1275Q (IC50 = 5.4 nM) and demonstrates antitumor activity in xenograft mouse models. ASP3026 has been shown to overcome crizotinib resistance in non-small cell lung cancer, and is currently being evaluated in clinical trials of patients with ALK-positive solid tumors.More related product prices
PF-06463922 Crizotinib AP26113 ALK/IGF1R inhibitor 1256580-46-7 Ceritinib (LDK378) 936091-14-4 ASP-2215 SGI 7079 XL 228 UNC 0631 AGI6780 ABX-1431Related product price
-
PF-06463922
$12-2822 -
Crizotinib
$5-1963.5 -
AP26113
$8-1200
![N2-[2-Methoxy-4-[4-(4-methyl-1-piperazinyl)-1-piperidinyl]phenyl]-N4-[2-[(1-methylethyl)sulfonyl]phenyl]-1,3,5-triazine-2,4-diamine](https://img.chemicalbook.com/ProductImageEN/2019-12/small/14b936d0-093b-4cf8-8442-2e050c2f0f67.png){kind=small}
