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ChemicalBook CAS DataBase List 1-[5-(Trifluoromethyl)-2-pyridinyl]-(3R)-3-pyrrolidinamine
202267-15-0

1-[5-(Trifluoromethyl)-2-pyridinyl]-(3R)-3-pyrrolidinamine synthesis

2synthesis methods
(R)-N-Boc-1-(5-(trifluoroMethyl)pyridin-2-yl)pyrrolidin-3-aMine

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1-[5-(Trifluoromethyl)-2-pyridinyl]-(3R)-3-pyrrolidinamine

202267-15-0
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Yield:202267-15-0 99 %

Reaction Conditions:

with trifluoroacetic acid in dichloromethane at 20;Inert atmosphere;

References:

Angeli, Andrea;Micheli, Laura;Carta, Fabrizio;Ferraroni, Marta;Pirali, Tracey;Fernandez Carvajal, Asia;Ferrer Montiel, Antonio;Di Cesare Mannelli, Lorenzo;Ghelardini, Carla;Supuran, Claudiu T. [Journal of Medicinal Chemistry,2023,vol. 66,# 2,p. 1616 - 1633]

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