720690-73-3
中文名稱
6-(3-CYCLOBUTYL-2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPIN-7-YLOXY)-N-METHYLNICOTINAMIDE
英文名稱
GSK 189254A
CAS
720690-73-3
分子式
C21H25N3O2
分子量
351.44
MOL 文件
720690-73-3.mol
更新日期
2026/05/14 08:26:11
720690-73-3 結(jié)構(gòu)式
基本信息
中文別名
化合物GSK189254A 英文別名
CS-2905GSK 189254A
histamine H3 receptor antagonist GS189254A
Histamine Receptor,GSK-189254,GSK 189254,GSK-189254A,inhibit,GSK189254A,Inhibitor
6-(3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-yloxy)-N-MethylnicotinaMide
N-(4-METHOXYBENZYL)-1-[(4-METHYLPHENYL)SULFONYL]-1H-PYRROLO[2,3-B
6-[(3-cyclobutyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)oxy]-N-methylpyridine-3-carboxamide
3-Pyridinecarboxamide, 6-[(3-cyclobutyl-2,3,4,5-tetrahydro-1H-3-benzazepin-7-yl)oxy]-N-methyl-
所屬類別
生物化工：激動劑抑制劑物理化學(xué)性質(zhì)
沸點545.0±50.0 °C(Predicted)
密度1.195±0.06 g/cm3(Predicted)
儲存條件-20°C儲存
溶解度DMSO:25.0(Max Conc. mg/mL);71.13(Max Conc. mM)
酸度系數(shù)(pKa)14.26±0.46(Predicted)
形態(tài)固體
顏色White to off-white
常見問題列表
概述
GSK189254A (GSK189254 free base)是一個新穎高效有選擇性的H3受體拮抗劑，對人類和大鼠H3的pKi值分別為9.59-9.90 and 8.51-9.17。6-(3-CYCLOBUTYL-2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPIN-7-YLOXY)-N-METHYLNICOTINAMIDE價格(試劑級)
| 報價日期 | 產(chǎn)品編號 | 產(chǎn)品名稱 | CAS號 | 包裝 | 價格 |
| 2025/12/22 | HY-14111 | 6-(3-CYCLOBUTYL-2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPIN-7-YLOXY)-N-METHYLNICOTINAMIDE GSK189254A | 720690-73-3 | 1mg | 600元 |
| 2025/12/22 | HY-14111 | 6-(3-CYCLOBUTYL-2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPIN-7-YLOXY)-N-METHYLNICOTINAMIDE GSK189254A | 720690-73-3 | 10mM * 1mLin DMSO | 773元 |
| 2025/12/22 | HY-14111 | 6-(3-CYCLOBUTYL-2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPIN-7-YLOXY)-N-METHYLNICOTINAMIDE GSK189254A | 720690-73-3 | 5mg | 1000元 |