ChemicalBook >> CAS DataBase List >>Melagatran
Melagatran
- CAS No.
- 159776-70-2
- Chemical Name:
- Melagatran
- Synonyms
- H-319/68;Melagatran;Melagatran, 10 mM in DMSO;2-(((R)-2-((S)-2-((4-Carbamimidoylbenzyl)carbamoyl)azetidin-1-yl)-1-cyclohexyl-2-oxoethyl)amino)acetic acid;2-[[(1R)-2-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]azetidin-1-yl]-1-cyclohexyl-2-oxoethyl]amino]acetic acid;N-[(1R)-2-[(2S)-2-[[[[4-(Aminoiminomethyl)phenyl]methyl]amino]carbonyl]-1-azetidinyl]-1-cyclohexyl-2-oxoethyl]glycine;Glycine, N-[(1R)-2-[(2S)-2-[[[[4-(aminoiminomethyl)phenyl]methyl]amino]carbonyl]-1-azetidinyl]-1-cyclohexyl-2-oxoethyl]-
- CBNumber:
- CB41176409
- Molecular Formula:
- C22H31N5O4
- Molecular Weight:
- 429.51
- MDL Number:
- MFCD00945676
- MOL File:
- 159776-70-2.mol
- MSDS File:
- SDS
- TDS File:
- TDS
Last updated:2026-07-11 12:07:37
| Product description | Number | Pack Size | Price |
| Melagatran ≥90% | 9002300 | 1mg | $413 |
| Melagatran >95%(HPLC) | TRC-M208450-5MG | 5mg | $1275 |
| Melagatran >95%(HPLC) | TRC-M208450-1MG | 1mg | $289 |
| Melagatran >95%(HPLC) | TRC-M208450-10MG | 10mg | $2305 |
| Melagatran | 015881 | 1mg | $523 |
| Melting point | 198-200°C |
|---|---|
| Density | 1.41±0.1 g/cm3(Predicted) |
| storage temp. | Hygroscopic, -20°C Freezer, Under Inert Atmosphere |
| solubility | Chloroform (Slightly), DMSO (Slightly), Methanol (Slightly) |
| form | Solid |
| pka | 2.12±0.10(Predicted) |
| color | White to Off-White |
| Stability | Hygroscopic |
| InChIKey | DKWNMCUOEDMMIN-PKOBYXMFSA-N |
| SMILES | C(O)(=O)CN[C@H](C1CCCCC1)C(N1CC[C@H]1C(NCC1=CC=C(C(N)=N)C=C1)=O)=O |
| FDA UNII | 2A9QP32MD4 |
| ATC code | B01AE04 |
SAFETY
Risk and Safety Statements
| Symbol(GHS) |  GHS07 |
|---|---|
| Signal word | Warning |
| Hazard statements | H335-H319-H315 |
| Precautionary statements | P264-P280-P302+P352-P321-P332+P313-P362-P264-P280-P305+P351+P338-P337+P313P |
Melagatran price
| Manufacturer | Product number | Product description | CAS number | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|---|
| Cayman Chemical | 9002300 | Melagatran ≥90% | 159776-70-2 | 1mg | $413 | 2026-04-30 | Buy |
| TRC | TRC-M208450-5MG | Melagatran >95%(HPLC) | 159776-70-2 | 5mg | $1275 | 2026-06-03 | Buy |
| TRC | TRC-M208450-1MG | Melagatran >95%(HPLC) | 159776-70-2 | 1mg | $289 | 2026-06-03 | Buy |
| TRC | TRC-M208450-10MG | Melagatran >95%(HPLC) | 159776-70-2 | 10mg | $2305 | 2026-06-03 | Buy |
| Usbiological | 015881 | Melagatran | 159776-70-2 | 1mg | $523 | 2026-06-03 | Buy |
Melagatran Chemical Properties,Uses,Production
Chemical Properties
White Solid
Uses
Synthetic thrombin inhibitor. Thrombin mutant anticoagulant antagonist. Antithrombotic.
Definition
ChEBI: Melagatran is a member of the class of azetidines that is (2S)-azetidine 2-carboxylic acid in which the carboxylic acid has been converted to the amide corresponding to formal condensation with 4-(aminomethyl)benzenecarboximidamide and in which the hydrogen attached to the azetidine nitrogen is replaced by a (2R)-2-cyclohexyl-2-[(carboxymethyl)amino]acetyl group. It has a role as an anticoagulant, an EC 3.4.21.5 (thrombin) inhibitor and a serine protease inhibitor. It is a carboxamidine, a dicarboxylic acid monoamide, a non-proteinogenic alpha-amino acid, a secondary amino compound and a member of azetidines.
Melagatran Preparation Products And Raw materials
Raw materials
Preparation Products
Melagatran Suppliers
Global( 52)Suppliers
| Supplier | Tel | Country | ProdList | Advantage | |
|---|---|---|---|---|---|
| Alchem Pharmtech,Inc. | 8485655694 | sales@alchempharmtech.com | United States | 63687 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; +17819995354 | marketing@targetmol.com | United States | 32466 | 58 |
| sgtlifesciences pvt ltd | +8617013299288 | dj@sgtlifesciences.com | China | 12373 | 58 |
| TargetMol Chemicals Inc. | +1-781-999-5354; | support@targetmol.com | United States | 39037 | 58 |
| Aladdin Scientific | tp@aladdinsci.com | United States | 52923 | 58 | |
| J & K SCIENTIFIC LTD. | 18210857532; 18210857532 | jkinfo@jkchemical.com | China | 96815 | 76 |
| Chemsky（shanghai）International Co.,Ltd. | 021-50135380 | shchemsky@sina.com | China | 32321 | 50 |
| Sichuan Wei Keqi Biological Technology Co., Ltd. | 028-81700200 18116577057 | 3003855609@qq.com | China | 7750 | 56 |
| Hangzhou Peptidego Biotech Co.,Ltd. | 0571-87213919 | Eric@peptidego.com | China | 7617 | 58 |
| Shanghai Hongye Biotechnology Co. Ltd | 400-9205774 | sales@glpbio.cn | China | 6777 | 58 |
View Lastest Price from Melagatran manufacturers
| Image | Update time | Product | Price | Min. Order | Purity | Supply Ability | Manufacturer | |
|---|---|---|---|---|---|---|---|---|
 |
2026-07-14 | Melagatran
159776-70-2
|
$540.00-1630.00 | 99.83% | 10g | TargetMol Chemicals Inc. | ||
 |
2026-07-14 | Melagatran
159776-70-2
|
$540.00-1630.00 | 99.83% | 10g | TargetMol Chemicals Inc. |
-
- Melagatran
159776-70-2
- $540.00-1630.00
- 99.83%
- TargetMol Chemicals Inc.
-
- Melagatran
159776-70-2
- $540.00-1630.00
- 99.83%
- TargetMol Chemicals Inc.
159776-70-2(Melagatran)Related Search:
H-319/68
Melagatran
N-[(1R)-2-[(2S)-2-[[[[4-(Aminoiminomethyl)phenyl]methyl]amino]carbonyl]-1-azetidinyl]-1-cyclohexyl-2-oxoethyl]glycine
2-(((R)-2-((S)-2-((4-Carbamimidoylbenzyl)carbamoyl)azetidin-1-yl)-1-cyclohexyl-2-oxoethyl)amino)acetic acid
2-[[(1R)-2-[(2S)-2-[(4-carbamimidoylphenyl)methylcarbamoyl]azetidin-1-yl]-1-cyclohexyl-2-oxoethyl]amino]acetic acid
Glycine, N-[(1R)-2-[(2S)-2-[[[[4-(aminoiminomethyl)phenyl]methyl]amino]carbonyl]-1-azetidinyl]-1-cyclohexyl-2-oxoethyl]-
Melagatran, 10 mM in DMSO
159776-70-2
C22H31N5O4
Aromatics
Chiral Reagents
Intermediates & Fine Chemicals
Pharmaceuticals
Aromatics Compounds
