Omarigliptin (MK-3102)
|
- $11 - $5576
- Product name: Omarigliptin (MK-3102)
- CAS: 1226781-44-7
- MF: C17H20F2N4O3S
- MW: 398.43
- EINECS:682-558-0
- MDL Number:MFCD22573261
- Synonyms:(2R,3S,5R)-2-(2,5-difluorophenyl)-5-(2-(Methylsulfonyl)pyrrolo[3,4-c]pyrazol-5(2H,4H,6H)-yl)tetrahydro-2H-pyran-3-aMine;MK-3012;(2S,3R,5S)-2-(2,5-Difluorophenyl)-5-[2-(Methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-2H-pyran-3-aMine (MK-3102 enantioMer);(2R,3S,5R)-2-(2,5-Difluorophenyl)-5-[2-(methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-2H-pyran-3-amine;OMarigliptin (MK-3102);2R,3S,5R)-2-(2,5-Difluorophenyl)-5-[2-(methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]pyrazol-5(4H)-yl]tetrahydro-2H-pyran-3-amine MK3102;MK-3102 - M10588;MK-3102, >=98%
88 prices
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Brand
- aablocks
- ACHEMBLOCK
- AK Scientific
- Ambeed
- ApexBio Technology
- Arctom
- Biorbyt Ltd
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Matrix Scientific
- Medical Isotopes, Inc.
- TRC
- Usbiological
Package
- 25mg
- 10mM(1mLinDMSO)
- 1mg
- 10mM*1mLinDMSO(Solid+Solvent)
- 100.00mg
- 1.00g
- 1000mg
- 250.00mg
- 10mM*1mLinDMSO
- 10mM*1mLinDMSO(Solution)
- 2mg
- 5mg
- 10mg
- 50mg
- 100mg
- 250mg
- 1g
- 5g
- 10mM(in1mLDMSO)
- Manufactureraablocks
- Product numberAA0017JR
- Product descriptionOmarigliptin 98%
- Packaging5mg
- Price$11
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0017JR
- Product descriptionOmarigliptin 98%
- Packaging10mg
- Price$14
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0017JR
- Product descriptionOmarigliptin 98%
- Packaging50mg
- Price$34
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0017JR
- Product descriptionOmarigliptin 98%
- Packaging100mg
- Price$48
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0017JR
- Product descriptionOmarigliptin 98%
- Packaging250mg
- Price$95
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0017JR
- Product descriptionOmarigliptin 95%
- Packaging1g
- Price$335
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA0017JR
- Product descriptionOmarigliptin 95%
- Packaging5g
- Price$1096
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberG-6852
- Product descriptionMK-3102 98%
- Packaging5G
- Price$870
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberG-6852
- Product descriptionMK-3102 98%
- Packaging5G
- Price$870
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberG-6852
- Product descriptionMK-3102 98%
- Packaging100MG
- Price$55
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberG-6852
- Product descriptionMK-3102 98%
- Packaging100MG
- Price$55
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberG-6852
- Product descriptionMK-3102 98%
- Packaging1G
- Price$255
- Updated2026-05-25
- Buy
- ManufacturerACHEMBLOCK
- Product numberG-6852
- Product descriptionMK-3102 98%
- Packaging1G
- Price$255
- Updated2026-05-27
- Buy
- ManufacturerAK Scientific
- Product number9051AF
- Product descriptionOmarigliptin
- Packaging2mg
- Price$158
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA115550
- Product descriptionOmarigliptin 98+%
- Packaging5mg
- Price$149
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA115550
- Product descriptionOmarigliptin 98+%
- Packaging10mg
- Price$194
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA0017JR | Omarigliptin 98% | 5mg | $11 | 2026-05-28 | Buy |
| aablocks | AA0017JR | Omarigliptin 98% | 10mg | $14 | 2026-05-28 | Buy |
| aablocks | AA0017JR | Omarigliptin 98% | 50mg | $34 | 2026-05-28 | Buy |
| aablocks | AA0017JR | Omarigliptin 98% | 100mg | $48 | 2026-05-28 | Buy |
| aablocks | AA0017JR | Omarigliptin 98% | 250mg | $95 | 2026-05-28 | Buy |
| aablocks | AA0017JR | Omarigliptin 95% | 1g | $335 | 2026-05-28 | Buy |
| aablocks | AA0017JR | Omarigliptin 95% | 5g | $1096 | 2026-05-28 | Buy |
| ACHEMBLOCK | G-6852 | MK-3102 98% | 5G | $870 | 2026-05-25 | Buy |
| ACHEMBLOCK | G-6852 | MK-3102 98% | 5G | $870 | 2026-05-27 | Buy |
| ACHEMBLOCK | G-6852 | MK-3102 98% | 100MG | $55 | 2026-05-25 | Buy |
| ACHEMBLOCK | G-6852 | MK-3102 98% | 100MG | $55 | 2026-05-27 | Buy |
| ACHEMBLOCK | G-6852 | MK-3102 98% | 1G | $255 | 2026-05-25 | Buy |
| ACHEMBLOCK | G-6852 | MK-3102 98% | 1G | $255 | 2026-05-27 | Buy |
| AK Scientific | 9051AF | Omarigliptin | 2mg | $158 | 2021-12-16 | Buy |
| Ambeed | A115550 | Omarigliptin 98+% | 5mg | $149 | 2021-12-16 | Buy |
| Ambeed | A115550 | Omarigliptin 98+% | 10mg | $194 | 2021-12-16 | Buy |
Properties
Boiling point :529.4±60.0 °C(Predicted)
Density :1.61±0.1 g/cm3(Predicted)
storage temp. :2-8°C(protect from light)
solubility :insoluble in EtOH; insoluble in H2O; ≥17.15 mg/mL in DMSO
form :solid
pka :9.11±0.60(Predicted)
color :White to off-white
InChI :InChI=1S/C17H20F2N4O3S/c1-27(24,25)23-7-10-6-22(8-16(10)21-23)12-5-15(20)17(26-9-12)13-4-11(18)2-3-14(13)19/h2-4,7,12,15,17H,5-6,8-9,20H2,1H3/t12-,15+,17-/m1/s1
InChIKey :MKMPWKUAHLTIBJ-ISTRZQFTSA-N
SMILES :[C@H]1(C2=CC(F)=CC=C2F)OC[C@H](N2CC3=CN(S(C)(=O)=O)N=C3C2)C[C@@H]1N
CAS DataBase Reference :1226781-44-7
Density :1.61±0.1 g/cm3(Predicted)
storage temp. :2-8°C(protect from light)
solubility :insoluble in EtOH; insoluble in H2O; ≥17.15 mg/mL in DMSO
form :solid
pka :9.11±0.60(Predicted)
color :White to off-white
InChI :InChI=1S/C17H20F2N4O3S/c1-27(24,25)23-7-10-6-22(8-16(10)21-23)12-5-15(20)17(26-9-12)13-4-11(18)2-3-14(13)19/h2-4,7,12,15,17H,5-6,8-9,20H2,1H3/t12-,15+,17-/m1/s1
InChIKey :MKMPWKUAHLTIBJ-ISTRZQFTSA-N
SMILES :[C@H]1(C2=CC(F)=CC=C2F)OC[C@H](N2CC3=CN(S(C)(=O)=O)N=C3C2)C[C@@H]1N
CAS DataBase Reference :1226781-44-7
Safety Information
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Description
Merck earned its first global approval for omarigliptin in Japan in 2015, and phase III development is ongoing in other countries around the globe for this interesting small molecule DPP-4 inhibitor. Interestingly, while most DPP-4 inhibitors used to treat type 2 DM require daily administration, omarigliptin is a weekly treatment. The process-scale synthesis of omarigliptin has been nicely described in an October 2015 paper from the Merck process group.Related product price
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tert-butyl [(2R,3S)-2-(2,5-difluorophenyl)-5-hydroxytetrahydro-2H-pyran-3-yl]carbaMate
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Suppliers and manufacturers
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