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Inhibitoren und Aktivatoren

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Structure Chemical Name CAS MF
BTdCPU BTdCPU 1257423-87-2 C13H8Cl2N4OS
WH-4-023 (SRC inhibitor) WH-4-023 (SRC inhibitor)
TG101348 (JAK inhibitor) TG101348 (JAK inhibitor)
PFI-3 (EPIGENETIC READER DOMAIN inhibitor) PFI-3 (EPIGENETIC READER DOMAIN inhibitor)
PD184352 (MEK inhibitor) PD184352 (MEK inhibitor)
ML324 (HISTONE DEMETHYLASE inhibitor) ML324 (HISTONE DEMETHYLASE inhibitor)
KU0063794 (MTOR inhibitor) KU0063794 (MTOR inhibitor)
JNJ-7777120 (HISTAMINE RECEPTOR antagonist) JNJ-7777120 (HISTAMINE RECEPTOR antagonist)
GSK1292263 (GPR agonist) GSK1292263 (GPR agonist)
BYL719 (PI3K inhibitor) BYL719 (PI3K inhibitor)
BML-210 (HDAC inhibitor) BML-210 (HDAC inhibitor)
2H-Pyran-4-propanamide, α-[4-(cyclopropylsulfonyl)phenyl]-N-(5-fluoro-2-thiazolyl)tetrahydro-, (αR)- 2H-Pyran-4-propanamide, α-[4-(cyclopropylsulfonyl)phenyl]-N-(5-fluoro-2-thiazolyl)tetrahydro-, (αR)- 745051-61-0 C20H23FN2O4S2
VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor) VENETOCLAX (ABT-199, GDC-0199) (BCL-2 inhibitor)
U-104 (CARBONIC ANHYDRASE INHIBITOR) U-104 (CARBONIC ANHYDRASE INHIBITOR)
SALUBRINAL (PERK inhibitor) SALUBRINAL (PERK inhibitor)
FLAVOPIRIDOL HCL (CDK inhibitor) FLAVOPIRIDOL HCL (CDK inhibitor)
DEFACTINIB (FAK inhibitor) DEFACTINIB (FAK inhibitor)
CEDIRANIB (VEGFR inhibitor) CEDIRANIB (VEGFR inhibitor)
BAY11-7082 (IΚB/IKK inhibitor) BAY11-7082 (IΚB/IKK inhibitor)
(-)-BLEBBISTATIN (ATPASE inhibitor) (-)-BLEBBISTATIN (ATPASE inhibitor)
AG14361 (PARP1 inhibitor) AG14361 (PARP1 inhibitor)
ACP-196 (BTK inhibitor) ACP-196 (BTK inhibitor)
ABT-737 (BCL-2 inhibitor) ABT-737 (BCL-2 inhibitor)
CK-2127107 CK-2127107 1345410-31-2 C19H18F2N6O
VILAZODONE (SSRI inhibitor) VILAZODONE (SSRI inhibitor)
TBA-354 (anti-tuberculosis) TBA-354 (anti-tuberculosis)
SAG (HEDGEHOG/SMOOTHENED agonist) SAG (HEDGEHOG/SMOOTHENED agonist)
PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor) PACLITAXEL (MICROTUBULE ASSOSIATED inhibitor)
OSU-03012 (PDK-1 inhibitor) OSU-03012 (PDK-1 inhibitor)
MONOMETHYL AURISTATIN E (microtubule-associated inhibitor) MONOMETHYL AURISTATIN E (microtubule-associated inhibitor)
ML141 (RHO inhibitor) ML141 (RHO inhibitor)
KN-93 PHOSPHATE (CAMK Inhibitor) KN-93 PHOSPHATE (CAMK Inhibitor)
GSK126 (EZH2 inhibitor) GSK126 (EZH2 inhibitor)
GELDANAMYCIN (HSP90 inhibitor) GELDANAMYCIN (HSP90 inhibitor)
GANT61 (HEDGEHOG/SMOOTHENED Inhibitor) GANT61 (HEDGEHOG/SMOOTHENED Inhibitor)
EPZ-6438 (E7438) (EZH2 inhibitor) EPZ-6438 (E7438) (EZH2 inhibitor)
EMPAGLIFLOZIN (SGLT inhibitor) EMPAGLIFLOZIN (SGLT inhibitor)
DOXORUBICIN (TOPOISOMERASE inhibitor) DOXORUBICIN (TOPOISOMERASE inhibitor)
DAPT (Γ-SECRETASE inhibitor) DAPT (Γ-SECRETASE inhibitor)
DACLATASVIR (HCV NS5A inhibitor) DACLATASVIR (HCV NS5A inhibitor)
COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor) COMBRETASTATIN A4 (MICROTUBULE ASSOCIATED inhibitor)
CABOZANTINIB (VEGFR inhibitor) CABOZANTINIB (VEGFR inhibitor)
BREFELDIN A (protein transport inhibitor) BREFELDIN A (protein transport inhibitor)
BKM120 (PI3K inhibitor) BKM120 (PI3K inhibitor)
AKT INHIBITOR VIII (AKT inhibitor) AKT INHIBITOR VIII (AKT inhibitor)
ABT-199 (BCL-2 inhibitor) ABT-199 (BCL-2 inhibitor)
Porfiromycin Porfiromycin 801-52-5 C16H20N4O5
VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor) VINCRISTINE (MICROTUBULE ASSOSIATED inhibitor)
TETRABENAZINE (VMAT-2 Inhibitor) TETRABENAZINE (VMAT-2 Inhibitor)
SNX-2112 (PF-04928473) (HSP90 antimony inhibitor) SNX-2112 (PF-04928473) (HSP90 antimony inhibitor)
PLX4032 (RAF inhibitor) PLX4032 (RAF inhibitor)
PD123319 (RAAS inhibitor) PD123319 (RAAS inhibitor)
NS-2028 (SGC inhibitor) NS-2028 (SGC inhibitor)
NECROSTATIN-1 (TNF-ALPHA inhibitor) NECROSTATIN-1 (TNF-ALPHA inhibitor)
ML323 (DUB inhibitor) ML323 (DUB inhibitor)
KU-55933 (ATM inhibitor) KU-55933 (ATM inhibitor)
(+)-JQ1 (BRD4 inhibitor) (+)-JQ1 (BRD4 inhibitor)
GSK2141795 (AKT inhibitor) GSK2141795 (AKT inhibitor)
GANETESPIB (HSP inhibitor) GANETESPIB (HSP inhibitor)
ENZALUTAMIDE (MDV3100) (AR inhibitor) ENZALUTAMIDE (MDV3100) (AR inhibitor)
BRIVANIB (VEGFR inhibitor) BRIVANIB (VEGFR inhibitor)
BARDOXOLONE METHYL (IΚB/IKK inhibitor) BARDOXOLONE METHYL (IΚB/IKK inhibitor)
AZ20 (ATM/ATR inhibitor) AZ20 (ATM/ATR inhibitor)
ARN-509 (ANDROGEN RECEPTOR Inhibitor) ARN-509 (ANDROGEN RECEPTOR Inhibitor)
5-PREGNEN-3BETA-OL-20-ONE-16ALPHA-CARBONITRILE 5-PREGNEN-3BETA-OL-20-ONE-16ALPHA-CARBONITRILE 1434-54-4 C22H31NO2
TWS119 (GSK-3 inhibitor) TWS119 (GSK-3 inhibitor)
SC-514 (IΚB/IKK inhibitor) SC-514 (IΚB/IKK inhibitor)
ROMIDEPSIN (HDAC inhibitor) ROMIDEPSIN (HDAC inhibitor)
REGADENOSON (ADENOSINE RECEPTOR agonist) REGADENOSON (ADENOSINE RECEPTOR agonist)
PYRIDONE 6 (JAK inhibitor) PYRIDONE 6 (JAK inhibitor)
PRT062607 HCL (SYK inhibitor) PRT062607 HCL (SYK inhibitor)
PAZOPANIB (VEGFR inhibitor) PAZOPANIB (VEGFR inhibitor)
MLN9708 (20S PROTEASOME Inhibitor) MLN9708 (20S PROTEASOME Inhibitor)
INDIPLON (GABA RECEPTOR Conditioner) INDIPLON (GABA RECEPTOR Conditioner)
FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor) FIDAXOMICIN (DNA/RNA SYNTHESIS Inhibitor)
EVEROLIMUS (MTOR inhibitor) EVEROLIMUS (MTOR inhibitor)
ENTOSPLETINIB (SYK inhibitor) ENTOSPLETINIB (SYK inhibitor)
DABRAFENIB (RAF inhibitor) DABRAFENIB (RAF inhibitor)
CYT997 (LEXIBULIN) (MICROTUBULES inhibitor) CYT997 (LEXIBULIN) (MICROTUBULES inhibitor)
BMS-5 (LIMK inhibitor) BMS-5 (LIMK inhibitor)
AZD7762 (CHK inhibitor) AZD7762 (CHK inhibitor)
AG1024 (IGF-1R inhibitor) AG1024 (IGF-1R inhibitor)
VISMODEGIB (HEDGEHOG/SMOOTHENED INHIBITOR) VISMODEGIB (HEDGEHOG/SMOOTHENED INHIBITOR)
REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor) REMODELIN (HISTONE ACETYLTRANSFERASE inhibitor)
PAC-1 (CASPASE Activator) PAC-1 (CASPASE Activator)
OSELTAMIVIR PHOSPHATE (NEURAMINIDASE Inhibitor) OSELTAMIVIR PHOSPHATE (NEURAMINIDASE Inhibitor)
MONENSIN (protein transport inhibitor) MONENSIN (protein transport inhibitor)
LINIFANIB (VEGFR inhibitor) LINIFANIB (VEGFR inhibitor)
LCZ696 (RAAS inhibitor) LCZ696 (RAAS inhibitor)
IONOMYCIN (calcium ionophore) IONOMYCIN (calcium ionophore)
HYDROXYUREA (DNA SYNTHESIS inhibitor) HYDROXYUREA (DNA SYNTHESIS inhibitor)
GZD824 DIMESYLATE (BCR-ABL inhibitor) GZD824 DIMESYLATE (BCR-ABL inhibitor)
FORETINIB (C-MET inhibitor) FORETINIB (C-MET inhibitor)
DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor) DAPIVIRINE (REVERSE TRANSCRIPTASE Inhibitor)
CNX-774 (BTK inhibitor) CNX-774 (BTK inhibitor)
BIRB 796 (P38 MAPK Inhibitor) BIRB 796 (P38 MAPK Inhibitor)
BAY87-2243 (HIF inhibitor) BAY87-2243 (HIF inhibitor)
B-AP15 (DUB inhibitor) B-AP15 (DUB inhibitor)
APIXABAN (FACTOR XA Inhibitor) APIXABAN (FACTOR XA Inhibitor)
TPA Deficient Plasma TPA Deficient Plasma
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