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Pharmaceutical intermediates

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Structure Chemical Name CAS MF
3-(3-methyl-1H-pyrazol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 3-(3-methyl-1H-pyrazol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 2223053-78-7 C17H20BN3O2
3-(N-Boc-Piperidin-3-yl)-5-bromophenylboronic acid pinacol ester 3-(N-Boc-Piperidin-3-yl)-5-bromophenylboronic acid pinacol ester 2223009-35-4 C22H33BBrNO4
3-(tetrahydro-2H-pyran-4-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 3-(tetrahydro-2H-pyran-4-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2223030-34-8 C17H26BNO3
3,6-DIHYDRO-2H-4-BROMOPYRIDINE 3,6-DIHYDRO-2H-4-BROMOPYRIDINE 1622840-69-0 C5H8BrN
3-Bromo-4-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 3-Bromo-4-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2223047-75-2 C15H18BBrN2O2
3-Fluoro-4-(3-methylpiperidin-1-yl)phenylboronic acid pinacol ester 3-Fluoro-4-(3-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2223004-47-3 C18H27BFNO2
3-Fluoro-4-(N-Boc-piperidin-3-yl)phenylboronic acid pinacol ester 3-Fluoro-4-(N-Boc-piperidin-3-yl)phenylboronic acid pinacol ester 2223004-08-6 C22H33BFNO4
3-Methoxy-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 3-Methoxy-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 2223046-77-1 C23H36BNO5
3-Methyl-4-(piperazin-1-yl)phenylboronic acid pinacol ester 3-Methyl-4-(piperazin-1-yl)phenylboronic acid pinacol ester 1613285-94-1 C17H27BN2O2
4-(2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(2-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223032-43-5 C17H25BClNO2
4-(2-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 4-(2-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 2223009-25-2 C16H26BNO2S
4-(3-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 4-(3-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 2223003-62-9 C16H26BNO2S
4-(4-bromo-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(4-bromo-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223033-01-8 C17H25BBrNO2
4-(4-Tetrahydropyranyl)-1,3,5-triazin-2-amine 4-(4-Tetrahydropyranyl)-1,3,5-triazin-2-amine 1417519-51-7 C8H12N4O
4-(5-methoxy-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(5-methoxy-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223050-00-6 C18H28BNO3
4-(N-Boc-piperidin-4-yl)thiophene-2-boronic acid pinacol ester 4-(N-Boc-piperidin-4-yl)thiophene-2-boronic acid pinacol ester 2223045-62-1 C20H32BNO4S
4-(Thiazol-4-yl)-2-fluorophenylboronic acid pinacol ester 4-(Thiazol-4-yl)-2-fluorophenylboronic acid pinacol ester 2223046-64-6 C15H17BFNO2S
4,4,5,5-tetramethyl-2-(3-(tetrahydro-2H-pyran-4-yl)-5-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(3-(tetrahydro-2H-pyran-4-yl)-5-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 2223029-76-1 C18H24BF3O3
4,4,5,5-tetramethyl-2-(4-(tetrahydro-2H-pyran-4-yl)furan-2-yl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(4-(tetrahydro-2H-pyran-4-yl)furan-2-yl)-1,3,2-dioxaborolane 2223033-50-7 C15H23BO4
4-Amino-2-(imidazol-1-yl)thiazole 4-Amino-2-(imidazol-1-yl)thiazole 1314354-26-1 C6H6N4S
4-Amino-2-(iso-propyl)-6-(piperidin-1-yl)-pyrimidine 4-Amino-2-(iso-propyl)-6-(piperidin-1-yl)-pyrimidine 1412960-78-1 C12H20N4
4-AMINO-2-CHLORO-5-(1-METHYLETHENYL)PYRIDINE 4-AMINO-2-CHLORO-5-(1-METHYLETHENYL)PYRIDINE 1622839-17-1 C8H9ClN2
4-Amino-6-methylpyridine-3-boronic acid pinacol ester 4-Amino-6-methylpyridine-3-boronic acid pinacol ester 1668475-78-2 C12H19BN2O2
4-Bromo-1-methyl-2-acetyl-1H-pyrrole 4-Bromo-1-methyl-2-acetyl-1H-pyrrole 1337993-67-5 C7H8BrNO
4-Bromo-2-(iso-propyl)-6-(iso-propoxy)pyrimidine 4-Bromo-2-(iso-propyl)-6-(iso-propoxy)pyrimidine 1412957-00-6 C10H15BrN2O
4-Bromo-2-cyclopropyl-6-(3-chlorophenyl)pyrimidine 4-Bromo-2-cyclopropyl-6-(3-chlorophenyl)pyrimidine 1412961-99-9 C13H10BrClN2
4-Bromo-3-fluoro-2-cyclohexylpyridine 4-Bromo-3-fluoro-2-cyclohexylpyridine 1643576-34-4 C11H13BrFN
4-Chloro-2-(2-methoxyphenyl)pyrimidine 4-Chloro-2-(2-methoxyphenyl)pyrimidine 1155594-52-7 C11H9ClN2O
4-chloro-2-(iso-propyl)-6-(1H-3-methylpyrozol-1-yl)pyrimidine 4-chloro-2-(iso-propyl)-6-(1H-3-methylpyrozol-1-yl)pyrimidine 1412953-05-9 C11H13ClN4
4-Chloro-6-bromo-2-methylpyrimidine 4-Chloro-6-bromo-2-methylpyrimidine 1353854-88-2 C5H4BrClN2
4-Fluoro-2-(1-hydroxy-1-methylethyl)pyridine 4-Fluoro-2-(1-hydroxy-1-methylethyl)pyridine 1563530-09-5 C8H10FNO
4-Fluoro-2-ethoxypyridine 4-Fluoro-2-ethoxypyridine 858675-62-4 C7H8FNO
4-Hydroxy-2-(3-furyl)pyrimidine 4-Hydroxy-2-(3-furyl)pyrimidine 1159817-11-4 C8H6N2O2
4-Hydroxy-2-(iso-propyl)-6-(1H-pyrozol-1-yl)pyrimidine 4-Hydroxy-2-(iso-propyl)-6-(1H-pyrozol-1-yl)pyrimidine 1412954-06-3 C10H12N4O
4-Hydroxy-2-cyclopropyl-6-(1H-pyrazol-1-yl)pyrimidine 4-Hydroxy-2-cyclopropyl-6-(1H-pyrazol-1-yl)pyrimidine 1412958-47-4 C10H10N4O
5-(2-Fluorophenyl)-2-hydroxypyrazine 5-(2-Fluorophenyl)-2-hydroxypyrazine 1159819-38-1 C10H7FN2O
5-(2-Methylimidazol-1-yl)thiophene-2-boronic acid pinacol ester 5-(2-Methylimidazol-1-yl)thiophene-2-boronic acid pinacol ester 2223039-66-3 C14H19BN2O2S
5-(3-Furyl)-2-hydroxypyrazine 5-(3-Furyl)-2-hydroxypyrazine 1159818-07-1 C8H6N2O2
5-(4-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 5-(4-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 2223042-35-9 C16H26BNO2S
5-(Cyclopropylamino)pyrazine-2-boronic acid pinacol ester 5-(Cyclopropylamino)pyrazine-2-boronic acid pinacol ester 2223033-33-6 C13H20BN3O2
5-(iso-Propyl)-2-hydroxypyrazine 5-(iso-Propyl)-2-hydroxypyrazine 1159817-33-0 C7H10N2O
5-(methyl-d3)pyrazin-2-ol 5-(methyl-d3)pyrazin-2-ol 1185316-73-7 C5H3D3N2O
5-(N-Boc-Piperidin-4-yl)-2-cyanophenylboronic acid pinacol ester 5-(N-Boc-Piperidin-4-yl)-2-cyanophenylboronic acid pinacol ester 2223047-71-8 C23H33BN2O4
5-(Piperidino)furan-2-boronic acid pinacol ester 5-(Piperidino)furan-2-boronic acid pinacol ester 2223051-14-5 C15H24BNO3
5,5'-Di(tert-butyl)2,2'-bipyrazine 5,5'-Di(tert-butyl)2,2'-bipyrazine 1622840-53-2 C16H22N4
5-Amino-2-(2-methoxyphenyl)pyrimidine 5-Amino-2-(2-methoxyphenyl)pyrimidine 1152519-92-0 C11H11N3O
5-Amino-2-(2-tolyl)pyrimidine 5-Amino-2-(2-tolyl)pyrimidine 1094311-60-0 C11H11N3
5-Amino-2-(cyclobutoxy)thiazole 5-Amino-2-(cyclobutoxy)thiazole 1314356-04-1 C7H10N2OS
5-Amino-2-(cyclopentyl)pyrimidine 5-Amino-2-(cyclopentyl)pyrimidine 1178158-55-8 C9H13N3
5-Bromo-2-(2-aminopropan-2-yl)thiazole 5-Bromo-2-(2-aminopropan-2-yl)thiazole 1368049-77-7 C6H9BrN2S
5-Bromo-2-(cyclohexyloxy)pyrimidine 5-Bromo-2-(cyclohexyloxy)pyrimidine 1289041-20-8 C10H13BrN2O
5-Bromo-2-(piperidin-3-ol)thiazole 5-Bromo-2-(piperidin-3-ol)thiazole 959239-68-0 C8H11BrN2OS
5-Bromo-2-amino-4-(4-pyridyl)pyridine 5-Bromo-2-amino-4-(4-pyridyl)pyridine 1381938-04-0 C10H8BrN3
5-Bromo-6-(3-furyl)pyridine-3-boronic acid pinacol ester 5-Bromo-6-(3-furyl)pyridine-3-boronic acid pinacol ester 2223030-76-8 C15H17BBrNO3
5-Bromo-6-(3-methylpiperidin-1-yl)pyridine-3-boronic acid pinacol ester 5-Bromo-6-(3-methylpiperidin-1-yl)pyridine-3-boronic acid pinacol ester 1353877-34-5 C17H26BBrN2O2
5-Ethyl-6-methoxypyridine-3-boronic acid pinacol ester 5-Ethyl-6-methoxypyridine-3-boronic acid pinacol ester 2223032-94-6 C14H22BNO3
5-Hydroxy-2-(1H-pyrazol-1-yl)pyrimidine 5-Hydroxy-2-(1H-pyrazol-1-yl)pyrimidine 1260811-24-2 C7H6N4O
5-Methyl-2-(cyclopropyl)pyridine-4-boronic acid pinacol ester 5-Methyl-2-(cyclopropyl)pyridine-4-boronic acid pinacol ester 2223028-93-9 C15H22BNO2
5-Methyl-6-(sec-butyl)pyridine-3-boronic acid pinacol ester 5-Methyl-6-(sec-butyl)pyridine-3-boronic acid pinacol ester 2223008-80-6 C16H26BNO2
5-Methylpiperazine-2-boronic acid pinacol ester 5-Methylpiperazine-2-boronic acid pinacol ester 2223009-57-0 C11H23BN2O2
6-(2-Tolyl)pyrazine-2-boronic acid pinacol ester 6-(2-Tolyl)pyrazine-2-boronic acid pinacol ester 1402172-32-0 C17H21BN2O2
6-(3-Thienyl)pyrazine-2-boronic acid pinacol ester 6-(3-Thienyl)pyrazine-2-boronic acid pinacol ester 1402165-82-5 C14H17BN2O2S
6-(Cyclohexyl)pyrazine-2-boronic acid pinacol ester 6-(Cyclohexyl)pyrazine-2-boronic acid pinacol ester 1402166-02-2 C16H25BN2O2
6-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 6-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 2223032-34-4 C12H14BClN2O2
methyl 6-(tetrahydro-2H-pyran-2-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate methyl 6-(tetrahydro-2H-pyran-2-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 2222995-78-8 C18H26BNO5
N-(2-Acetoxyethyl)-2-methylimidazole-4-boronic acid pinacol ester N-(2-Acetoxyethyl)-2-methylimidazole-4-boronic acid pinacol ester 1402166-63-5 C14H23BN2O4
tert-butyl (4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazol-2-yl)carbamate tert-butyl (4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazol-2-yl)carbamate 2223044-39-9 C14H23BN2O4S
tert-butyl 2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-carboxylate tert-butyl 2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-carboxylate 2223046-19-1 C17H29BN2O4
tert-butyl 3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazol-2-yl)piperidine-1-carboxylate tert-butyl 3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazol-2-yl)piperidine-1-carboxylate 2223009-73-0 C19H31BN2O4S
tert-butyl 3-(5-bromopyridin-2-yl)pyrrolidine-1-carboxylate tert-butyl 3-(5-bromopyridin-2-yl)pyrrolidine-1-carboxylate 1245914-48-0 C14H19BrN2O2
tert-butyl 4-(2-amino-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate tert-butyl 4-(2-amino-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate 2223043-79-4 C22H35BN2O4
tert-butyl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-carboxylate-2,5-d2 tert-butyl 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-carboxylate-2,5-d2 2241864-95-7 C14H21BD2N2O4
(1-(methyl-d3)-1H-pyrazol-4-yl)boronic acid (1-(methyl-d3)-1H-pyrazol-4-yl)boronic acid 2256709-52-9 C4H7BN2O2
(3-(1H-pyrazol-1-yl-d3)phenyl)boronic acid (3-(1H-pyrazol-1-yl-d3)phenyl)boronic acid 2256709-37-0 C9H9BN2O2
(4-(piperidin-1-yl-d10)phenyl)boronic acid (4-(piperidin-1-yl-d10)phenyl)boronic acid 2241870-76-6 C11H16BNO2
1-(2-(methyl-d3)phenyl-3,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-3,5-d2 1-(2-(methyl-d3)phenyl-3,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-3,5-d2 2256711-19-8 C16H12BD9N2O2
1-(2-(trifluoromethyl)phenyl)-1H-imidazol-2-amine 1-(2-(trifluoromethyl)phenyl)-1H-imidazol-2-amine 1692857-34-3 C10H8F3N3
1-(2-bromo-4-cyclopropylphenyl)piperidine 1-(2-bromo-4-cyclopropylphenyl)piperidine 2222935-02-4 C14H18BrN
1-(2-bromo-5-cyclopropylphenyl)-1H-pyrazole 1-(2-bromo-5-cyclopropylphenyl)-1H-pyrazole 1622843-84-8 C12H11BrN2
1-(2-bromophenyl-3,4,5,6-d4)-2-(methyl-d3)-1H-imidazole-4,5-d2 1-(2-bromophenyl-3,4,5,6-d4)-2-(methyl-d3)-1H-imidazole-4,5-d2 2256713-05-8 C10H9BrN2
1-(2-fluorophenyl-3,4,5,6-d4)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-4,5-d2 1-(2-fluorophenyl-3,4,5,6-d4)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-4,5-d2 2256705-69-6 C15H18BFN2O2
1-(3-bromo-4-cyclopropylphenyl)piperidine 1-(3-bromo-4-cyclopropylphenyl)piperidine 2222934-99-6 C14H18BrN
1-(3-bromophenyl-2,4,5,6-d4)-1H-imidazole-2,4,5-d3 1-(3-bromophenyl-2,4,5,6-d4)-1H-imidazole-2,4,5-d3 2256712-89-5 C9H7BrN2
1-(3-fluorophenyl)-2-methyl-1H-imidazol-4-amine 1-(3-fluorophenyl)-2-methyl-1H-imidazol-4-amine 2294957-85-8 C10H10FN3
1-(3-fluorophenyl-2,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 1-(3-fluorophenyl-2,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 2256710-89-9 C15H12BD6FN2O2
1-(4-(methyl-d3)phenyl-2,3,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-3,5-d2 1-(4-(methyl-d3)phenyl-2,3,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-3,5-d2 2256711-23-4 C16H21BN2O2
1-(4,5-Dibromothiazol-2-yl)-4-bromopyrazole 1-(4,5-Dibromothiazol-2-yl)-4-bromopyrazole 1353856-59-3 C6H2Br3N3S
1-(4-bromo-2-cyclopropylphenyl)piperazine 1-(4-bromo-2-cyclopropylphenyl)piperazine 2126811-35-4 C13H17BrN2
1-(4-bromophenyl)-1H-imidazole-2,4,5-d3 1-(4-bromophenyl)-1H-imidazole-2,4,5-d3 2256712-63-5 C9H7BrN2
1-(4-bromophenyl)-4-(methyl-d3)-1H-pyrazole-3,5-d2 1-(4-bromophenyl)-4-(methyl-d3)-1H-pyrazole-3,5-d2 2256712-35-1 C10H9BrN2
1-(4-fluorophenyl)-1,3-dihydro-2H-imidazol-2-one 1-(4-fluorophenyl)-1,3-dihydro-2H-imidazol-2-one 155431-17-7 C9H7FN2O
1-(4-fluorophenyl-2,3,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 1-(4-fluorophenyl-2,3,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 2256710-91-3 C15H18BFN2O2
1-(5-bromo-2-cyclopropylphenyl)piperidine 1-(5-bromo-2-cyclopropylphenyl)piperidine 2222935-39-7 C14H18BrN
1-(6-(methyl-d3)pyrazin-2-yl-3,5-d2)-1H-pyrazol-3,5-d2-4-amine 1-(6-(methyl-d3)pyrazin-2-yl-3,5-d2)-1H-pyrazol-3,5-d2-4-amine 2256708-06-0 C8H2D7N5
1-(ethyl-d5)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-4,5-d2 1-(ethyl-d5)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazole-4,5-d2 2241877-35-8 C11H19BN2O2
1-(methyl-d3)-4-(3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-2,2,3,3,5,5,6,6-d8 1-(methyl-d3)-4-(3-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-2,2,3,3,5,5,6,6-d8 2256705-14-1 C18H18BD11N2O2
1-(methyl-d3)-4-(4-(methyl-d3)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-2,2,3,3,5,5,6,6-d8 1-(methyl-d3)-4-(4-(methyl-d3)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-2,2,3,3,5,5,6,6-d8 2256704-08-0 C18H29BN2O2
1-(Oxolan-3-yl)-2-(1-methylethyl)-1H-imidazol-4-amine 1-(Oxolan-3-yl)-2-(1-methylethyl)-1H-imidazol-4-amine 1622835-16-8 C10H17N3O
1-(phenylmethyl-d2)piperidin-4-one-2,2,3,3,5,5,6,6-d8 1-(phenylmethyl-d2)piperidin-4-one-2,2,3,3,5,5,6,6-d8 2259315-76-7 C12H15NO
1-(Pyrrolidin-3-yl)-2-ethylimidazol-4-amine 1-(Pyrrolidin-3-yl)-2-ethylimidazol-4-amine 1622835-79-3 C9H16N4
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