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Pharmaceutical intermediates

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Structure Chemical Name CAS MF
1-(5-bromofuran-2-yl)-4-methylpiperazine 1-(5-bromofuran-2-yl)-4-methylpiperazine 2241865-32-5 C9H13BrN2O
1-(Pyrrolidin-3-yl)-2-methylimidazol-4-amine 1-(Pyrrolidin-3-yl)-2-methylimidazol-4-amine 1622834-54-1 C8H14N4
1-(tert-butyl)-2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 1-(tert-butyl)-2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223040-48-8 C16H29BN2O2
1-[4-(TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-3-TRIFLUOROMETHYLPHENYL]PIPERIDIN-2-ONE 1-[4-(TETRAMETHYL-1,3,2-DIOXABOROLAN-2-YL)-3-TRIFLUOROMETHYLPHENYL]PIPERIDIN-2-ONE 2223045-95-0 C18H23BF3NO3
1-Cyclobutyl-2-ethylimidazol-4-amine 1-Cyclobutyl-2-ethylimidazol-4-amine 1622843-81-5 C9H15N3
1-Cyclohexyl-2-methylimidazol-4-amine 1-Cyclohexyl-2-methylimidazol-4-amine 1622840-24-7 C10H17N3
1-ethyl-2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 1-ethyl-2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223040-15-9 C14H25BN2O2
2-(1H-imidazol-1-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 2-(1H-imidazol-1-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 1310404-67-1 C12H16BN3O2S
2-(1H-pyrazol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(1H-pyrazol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1312942-18-9 C13H17BN4O2
2-(2-(methoxy-d3)phenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(2-(methoxy-d3)phenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2241867-40-1 C17H21BN2O3
2-(2-fluorophenyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 2-(2-fluorophenyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 1402174-42-8 C15H17BFNO2S
2-(2-Fluorophenyl)pyridine-3-boronic acid pinacol ester 2-(2-Fluorophenyl)pyridine-3-boronic acid pinacol ester 2223038-68-2 C17H19BFNO2
2-(2-methoxyphenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(2-methoxyphenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1402227-09-1 C17H21BN2O3
2-(2-methylpiperidin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(2-methylpiperidin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1309982-42-0 C16H26BN3O2
2-(3-bromo-4-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(3-bromo-4-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2222997-39-7 C17H24BBrO3
2-(3-bromo-5-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(3-bromo-5-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2223009-37-6 C17H24BBrO3
2-(3-cyclopropyl-4-(tetrahydro-2H-pyran-4-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(3-cyclopropyl-4-(tetrahydro-2H-pyran-4-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2223040-94-4 C20H29BO3
2-(3-fluoro-4-(tetrahydro-2H-pyran-4-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(3-fluoro-4-(tetrahydro-2H-pyran-4-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2223030-32-6 C17H24BFO3
2-(3-methoxyphenyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2-(3-methoxyphenyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2223027-53-8 C18H22BNO3
2-(3-Methoxyphenyl)pyridine-3-boronic acid 2-(3-Methoxyphenyl)pyridine-3-boronic acid 2225180-73-2 C12H12BNO3
2-(3-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)pyrazine 2-(3-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)pyrazine 2223052-61-5 C17H21BN2O2
2-(4-chloro-2-(tetrahydro-2H-pyran-4-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(4-chloro-2-(tetrahydro-2H-pyran-4-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2223038-73-9 C17H24BClO3
2-(4-methoxy-3-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(4-methoxy-3-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2222996-28-1 C18H27BO4
2-(4-Methylimidazol-1-yl)pyridine-5-boronic acid 2-(4-Methylimidazol-1-yl)pyridine-5-boronic acid 2225180-12-9 C9H10BN3O2
2-(ethoxy-d5)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(ethoxy-d5)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2241876-92-4 C12H19BN2O3
2-(piperazin-1-yl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(piperazin-1-yl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1310405-13-0 C14H23BN4O2
2-(piperidin-1-yl-d10)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(piperidin-1-yl-d10)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2241876-73-1 C15H24BN3O2
2-(Piperidino)thiophene-4-boronic acid pinacol ester 2-(Piperidino)thiophene-4-boronic acid pinacol ester 2223033-58-5 C15H24BNO2S
2-(PYRAZIN-2-YL)PROPAN-2-AMINE 2-(PYRAZIN-2-YL)PROPAN-2-AMINE 1082271-79-1 C7H11N3
2-(sec-butyl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(sec-butyl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2223004-09-7 C14H23BN2O2
2,4-Dibromo-5-(3-furyl)pyridine 2,4-Dibromo-5-(3-furyl)pyridine 1381936-73-7 C9H5Br2NO
2,4-Dibromo-5-iodopyridine 2,4-Dibromo-5-iodopyridine 1563530-52-8 C5H2Br2IN
2,4-Dibromo-6-(tert-butyl)pyridine 2,4-Dibromo-6-(tert-butyl)pyridine 1353856-97-9 C9H11Br2N
2,5-Dibromo-4-(3-pyridyl)pyridine 2,5-Dibromo-4-(3-pyridyl)pyridine 1381933-55-6 C10H6Br2N2
2,5-Dibromo-4-(4-fluorophenyl)pyridine 2,5-Dibromo-4-(4-fluorophenyl)pyridine 1381933-56-7 C11H6Br2FN
2,5-Dibromo-4-(iso-propyl)pyridine 2,5-Dibromo-4-(iso-propyl)pyridine 1256833-52-9 C8H9Br2N
2-AMINO-3-(4-TOLYL)PYRIDINE 2-AMINO-3-(4-TOLYL)PYRIDINE 1340103-90-3 C12H12N2
2-Amino-3-bromo-5-(cyclobutyl)pyridine 2-Amino-3-bromo-5-(cyclobutyl)pyridine 1381938-52-8 C9H11BrN2
2-Amino-5-(2-fluorophenyl)pyrazine 2-Amino-5-(2-fluorophenyl)pyrazine 1044574-46-0 C10H8FN3
2-Amino-5-(3-methoxyphenyl)pyrazine 2-Amino-5-(3-methoxyphenyl)pyrazine 328233-25-6 C11H11N3O
2-Amino-5-(4-ethylphenyl)pyrazine 2-Amino-5-(4-ethylphenyl)pyrazine 71544-66-6 C12H13N3
2-Amino-5-(cyclohexyl)pyrazine 2-Amino-5-(cyclohexyl)pyrazine 1159817-85-2 C10H15N3
2-Amino-5-(iso-propyl)pyrazine 2-Amino-5-(iso-propyl)pyrazine 114176-64-6 C7H11N3
2-Amino-5-bromo-4-(3-methyl-1H-pyrazol-1-yl)pyridine 2-Amino-5-bromo-4-(3-methyl-1H-pyrazol-1-yl)pyridine 1381937-07-0 C9H9BrN4
2-Amino-5-chloropyridine-4-boronic acid pinacol ester 2-Amino-5-chloropyridine-4-boronic acid pinacol ester 1222522-38-4 C11H16BClN2O2
2-Amino-6-(4-methyl-1H-pyrazol-1-yl)pyrazine 2-Amino-6-(4-methyl-1H-pyrazol-1-yl)pyrazine 1314353-56-4 C8H9N5
2-Amino-6-(pyrrolidino)pyrazine 2-Amino-6-(pyrrolidino)pyrazine 54015-46-2 C8H12N4
2-AMINO-6-TRIFLUOROMETHYLPYRIDINE-4-BORONIC ACID PINACOL ESTER 2-AMINO-6-TRIFLUOROMETHYLPYRIDINE-4-BORONIC ACID PINACOL ESTER 1558927-41-5 C12H16BF3N2O2
2-Bromo-3-(pyridin-4-yl)pyridine 2-Bromo-3-(pyridin-4-yl)pyridine 1417518-53-6 C10H7BrN2
2-Bromo-3-methoxycarbonyl-4-cyclopentylpyridine 2-Bromo-3-methoxycarbonyl-4-cyclopentylpyridine 1622844-18-1 C12H14BrNO2
2-Bromo-4-(1H-pyrazol-1-yl)furan 2-Bromo-4-(1H-pyrazol-1-yl)furan 1622839-59-1 C7H5BrN2O
2-Bromo-4-(2-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2-Bromo-4-(2-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2222997-61-5 C18H27BBrNO2
2-Bromo-4-(3-methyl-1H-pyrazol-1-yl)phenylboronic acid 2-Bromo-4-(3-methyl-1H-pyrazol-1-yl)phenylboronic acid 2225169-93-5 C10H10BBrN2O2
2-Bromo-4-(4-methylpiperidin-1-yl)thiophene 2-Bromo-4-(4-methylpiperidin-1-yl)thiophene 1622842-94-7 C10H14BrNS
2-Bromo-4-(piperidino)furan 2-Bromo-4-(piperidino)furan 1622840-84-9 C9H12BrNO
2-Bromo-4-(tert-butyl)pyrimidine 2-Bromo-4-(tert-butyl)pyrimidine 1353856-94-6 C8H11BrN2
2-Bromo-4,6-diisopropylpyrimidine 2-Bromo-4,6-diisopropylpyrimidine 1412961-55-7 C10H15BrN2
2-Bromo-4-chloro-5-(2-trifluoromethylphenyl)pyridine 2-Bromo-4-chloro-5-(2-trifluoromethylphenyl)pyridine 1381943-31-2 C12H6BrClF3N
2-bromo-4-phenyl-6-cyclopropylpyrimidine 2-bromo-4-phenyl-6-cyclopropylpyrimidine 1412955-75-9 C13H11BrN2
2-Bromo-5-(2-furyl)pyrazine 2-Bromo-5-(2-furyl)pyrazine 1142195-85-4 C8H5BrN2O
2-Bromo-5-(2-methylpiperidin-1-yl)furan 2-Bromo-5-(2-methylpiperidin-1-yl)furan 1622834-78-9 C10H14BrNO
2-Bromo-5-(3-methyl-1H-pyrazol-1-yl)furan 2-Bromo-5-(3-methyl-1H-pyrazol-1-yl)furan 1368301-60-3 C8H7BrN2O
2-Bromo-5-(4-methylimidazol-1-yl)furan 2-Bromo-5-(4-methylimidazol-1-yl)furan 1622843-38-2 C8H7BrN2O
2-Bromo-5-(piperidin-4-ol)pyrazine 2-Bromo-5-(piperidin-4-ol)pyrazine 959239-22-6 C9H12BrN3O
2-Chloro-4-(2-chlorophenyl)-6-(iso-propyl)pyrimidine 2-Chloro-4-(2-chlorophenyl)-6-(iso-propyl)pyrimidine 1412958-02-1 C13H12Cl2N2
2-Chloro-4-(3-chlorophenyl)-6-(iso-propyl)pyrimidine 2-Chloro-4-(3-chlorophenyl)-6-(iso-propyl)pyrimidine 1412960-95-2 C13H12Cl2N2
2-Chloro-4-(4-hydroxypiperidin-1-yl)-1,3,5-triazine 2-Chloro-4-(4-hydroxypiperidin-1-yl)-1,3,5-triazine 1417518-26-3 C8H11ClN4O
2-chloro-4-(cyclopropyl)-6-(tert-butyl)pyrimidine 2-chloro-4-(cyclopropyl)-6-(tert-butyl)pyrimidine 1412957-49-3 C11H15ClN2
2-Chloro-4-(pyrrolidin-1-yl)-6-(iso-propyl)pyrimidine 2-Chloro-4-(pyrrolidin-1-yl)-6-(iso-propyl)pyrimidine 1412959-82-0 C11H16ClN3
2-Chloro-4-(pyrrolidino)phenylboronic acid pinacol ester 2-Chloro-4-(pyrrolidino)phenylboronic acid pinacol ester 2223054-06-4 C16H23BClNO2
2-Chloro-4-bromo-6-methylpyrimidine 2-Chloro-4-bromo-6-methylpyrimidine 1137576-45-4 C5H4BrClN2
2-cyclobutoxy-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-cyclobutoxy-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2223030-06-4 C14H21BN2O3
2-Cyclopropyl-5-(imidazol-1-yl)phenylboronic acid pinacol ester 2-Cyclopropyl-5-(imidazol-1-yl)phenylboronic acid pinacol ester 2223036-05-1 C18H23BN2O2
2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-fluoro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1309981-66-5 C10H14BFN2O2
2-Fluoro-6-(iso-propyl)pyridine 2-Fluoro-6-(iso-propyl)pyridine 1563530-41-5 C8H10FN
2-Fluoro-6-(thiazol-2-yl)pyridine 2-Fluoro-6-(thiazol-2-yl)pyridine 1563530-00-6 C8H5FN2S
2-hydroxy-4-(3-chlorophenyl)-6-(tert-butyl)pyrimidine 2-hydroxy-4-(3-chlorophenyl)-6-(tert-butyl)pyrimidine 1412959-42-2 C14H15ClN2O
2-hydroxy-4-(3-furyl)-6-(tert-butyl)pyrimidine 2-hydroxy-4-(3-furyl)-6-(tert-butyl)pyrimidine 1412956-07-0 C12H14N2O2
2-Hydroxy-4-(iso-propoxy)-6-(tert-butyl)pyrimidine 2-Hydroxy-4-(iso-propoxy)-6-(tert-butyl)pyrimidine 1412959-99-9 C11H18N2O2
2-Hydroxy-5-(4-ethylphenyl)pyrazine 2-Hydroxy-5-(4-ethylphenyl)pyrazine 1159818-76-4 C12H12N2O
2-isopropyl-1-(tetrahydro-2H-pyran-4-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2-isopropyl-1-(tetrahydro-2H-pyran-4-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223034-82-8 C17H29BN2O3
2-Methoxy-6-(oxan-4-yl)pyridine-4-boronic acid pinacol ester 2-Methoxy-6-(oxan-4-yl)pyridine-4-boronic acid pinacol ester 2223033-94-9 C17H26BNO4
2-methyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-methyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1260152-72-4 C11H17BN2O2
2-Methyl-6-trifluoromethylpyridine-3-boronic acid pinacol ester 2-Methyl-6-trifluoromethylpyridine-3-boronic acid pinacol ester 2223041-89-0 C13H17BF3NO2
2-phenyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-phenyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2223032-39-9 C16H19BN2O2
3-(4-Tetrahydropyranyl)-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 3-(4-Tetrahydropyranyl)-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 2223051-46-3 C27H42BNO5
3-Amino-6-(3-methyl-1H-pyrazol-1-yl)pyrazine 3-Amino-6-(3-methyl-1H-pyrazol-1-yl)pyrazine 1314354-66-9 C8H9N5
3-Amino-6-(4-methylpiperidin-1-yl)pyridazine 3-Amino-6-(4-methylpiperidin-1-yl)pyridazine 69184-67-4 C10H16N4
3-Amino-6-(iso-propyl)pyridine-4-boronic acid pinacol ester 3-Amino-6-(iso-propyl)pyridine-4-boronic acid pinacol ester 2223052-51-3 C14H23BN2O2
3-Bromo-4-(iso-propyl)-2-chloropyridine 3-Bromo-4-(iso-propyl)-2-chloropyridine 1622842-64-1 C8H9BrClN
3-Bromo-5-(2-methylpiperidin-1-yl)phenylboronic acid pinacol ester 3-Bromo-5-(2-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2223005-18-1 C18H27BBrNO2
3-Bromo-5-(pyrazin-2-yl)phenylboronic acid pinacol ester 3-Bromo-5-(pyrazin-2-yl)phenylboronic acid pinacol ester 2223037-10-1 C16H18BBrN2O2
3-methyl-1-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethyl)phenyl)piperidine 3-methyl-1-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethyl)phenyl)piperidine 2223008-89-5 C19H27BF3NO2
4-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4-(trifluoromethyl)phenyl)piperidine 4-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-4-(trifluoromethyl)phenyl)piperidine 2223036-90-4 C18H25BF3NO2
4-(3-chloro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(3-chloro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223034-04-4 C17H25BClNO2
4-(3-cyclopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(3-cyclopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223048-68-6 C20H30BNO2
4-(3-Methyl-1H-pyrazol-1-yl)thiophene-2-boronic acid pinacol ester 4-(3-Methyl-1H-pyrazol-1-yl)thiophene-2-boronic acid pinacol ester 2223043-28-3 C14H19BN2O2S
4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3-(trifluoromethyl)phenyl)piperidine 4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3-(trifluoromethyl)phenyl)piperidine 2223032-88-8 C18H25BF3NO2
4-(4-Methylimidazol-1-yl)furan-2-boronic acid pinacol ester 4-(4-Methylimidazol-1-yl)furan-2-boronic acid pinacol ester 2223033-68-7 C14H19BN2O3
4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl)morpholine-2,2,3,3,5,5,6,6-d8 4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-yl)morpholine-2,2,3,3,5,5,6,6-d8 2241876-72-0 C14H22BN3O3
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