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Pharmaceutical intermediates

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Structure Chemical Name CAS MF
2-Amino-5-(1H-pyrazol-1-yl)pyrazine 2-Amino-5-(1H-pyrazol-1-yl)pyrazine 1211584-88-1 C7H7N5
2-Amino-5-(3-trifluoromethylphenyl)pyrazine 2-Amino-5-(3-trifluoromethylphenyl)pyrazine 59489-74-6 C11H8F3N3
2-Amino-5-(cyclobutoxy)pyrazine 2-Amino-5-(cyclobutoxy)pyrazine 1159818-56-0 C8H11N3O
2-Amino-5-(imidazol-1-yl)pyrazine 2-Amino-5-(imidazol-1-yl)pyrazine 1211536-30-9 C7H7N5
2-Amino-6-(piperazin-1-yl)pyrazine 2-Amino-6-(piperazin-1-yl)pyrazine 1314355-16-2 C8H13N5
2-Bromo-3-(3-thienyl)pyridine 2-Bromo-3-(3-thienyl)pyridine 1417518-57-0 C9H6BrNS
2-Bromo-3-fluoro-4-(2-furyl)pyridine 2-Bromo-3-fluoro-4-(2-furyl)pyridine 1622842-61-8 C9H5BrFNO
2-bromo-4-(1H-3-methylpyrozol-1-yl)-6-cyclopropylpyrimidine 2-bromo-4-(1H-3-methylpyrozol-1-yl)-6-cyclopropylpyrimidine 1412956-28-5 C11H11BrN4
2-Bromo-4-(2-chlorophenyl)-6-methylpyrimidine 2-Bromo-4-(2-chlorophenyl)-6-methylpyrimidine 1412952-89-6 C11H8BrClN2
2-Bromo-4-(2-methylimidazol-1-yl)thiophene 2-Bromo-4-(2-methylimidazol-1-yl)thiophene 1622839-62-6 C8H7BrN2S
2-Bromo-4-(2-methylpiperidin-1-yl)furan 2-Bromo-4-(2-methylpiperidin-1-yl)furan 1622835-31-7 C10H14BrNO
2-Bromo-4-(4-methyl-1H-pyrazol-1-yl)phenylboronic acid 2-Bromo-4-(4-methyl-1H-pyrazol-1-yl)phenylboronic acid 2225176-04-3 C10H10BBrN2O2
2-Bromo-4-(4-tetrahydropyranyl)-1,3,5-triazine 2-Bromo-4-(4-tetrahydropyranyl)-1,3,5-triazine 1417518-75-2 C8H10BrN3O
2-Bromo-4-(iso-propoxy)-6-cyclopropylpyrimidine 2-Bromo-4-(iso-propoxy)-6-cyclopropylpyrimidine 1412955-61-3 C10H13BrN2O
2-bromo-4-(pyrimindin-5-yl)-6-(tert-butyl)pyrimidine 2-bromo-4-(pyrimindin-5-yl)-6-(tert-butyl)pyrimidine 1412956-72-9 C12H13BrN4
2-Bromo-4,6-di(tert-butyl)pyrimidine 2-Bromo-4,6-di(tert-butyl)pyrimidine 1412956-29-6 C12H19BrN2
2-Bromo-4-chloro-5-(3-methoxyphenyl)pyridine 2-Bromo-4-chloro-5-(3-methoxyphenyl)pyridine 1381937-79-6 C12H9BrClNO
2-Bromo-5-(1-hydroxy-1-methylethyl)pyrazine 2-Bromo-5-(1-hydroxy-1-methylethyl)pyrazine 1303967-23-8 C7H9BrN2O
2-Bromo-5-(2-fluorophenyl)pyrazine 2-Bromo-5-(2-fluorophenyl)pyrazine 1142196-20-0 C10H6BrFN2
2-Bromo-5-(2-trifluoromethylphenyl)pyrazine 2-Bromo-5-(2-trifluoromethylphenyl)pyrazine 1159819-41-6 C11H6BrF3N2
2-Bromo-5-(3-tolyl)pyrazine 2-Bromo-5-(3-tolyl)pyrazine 1142195-92-3 C11H9BrN2
2-Bromo-5-(4-ethylphenyl)pyrazine 2-Bromo-5-(4-ethylphenyl)pyrazine 1142195-95-6 C12H11BrN2
2-Bromo-5-(4-tetrahydropyranyl)furan 2-Bromo-5-(4-tetrahydropyranyl)furan 1369138-95-3 C9H11BrO2
2-Bromo-5-(4-trifluoromethylphenyl)pyrazine 2-Bromo-5-(4-trifluoromethylphenyl)pyrazine 1142196-08-4 C11H6BrF3N2
2-Bromo-5-(imidazol-1-yl)furan 2-Bromo-5-(imidazol-1-yl)furan 1369079-10-6 C7H5BrN2O
2-Bromo-6-(2-Aminopropan-2-yl)pyrazine 2-Bromo-6-(2-Aminopropan-2-yl)pyrazine 1563528-69-7 C7H10BrN3
2-Bromo-6-(2-methylimidazol-1-yl)pyrazine 2-Bromo-6-(2-methylimidazol-1-yl)pyrazine 1159816-87-1 C8H7BrN4
2-Chloro-4-(1H-imidazol-1-yl)-6-(iso-propyl)pyrimidine 2-Chloro-4-(1H-imidazol-1-yl)-6-(iso-propyl)pyrimidine 1412961-75-1 C10H11ClN4
2-Chloro-4-(cyclopropoxy)pyrimidine 2-Chloro-4-(cyclopropoxy)pyrimidine 1289157-22-7 C7H7ClN2O
2-Cyano-6-(trifluoromethyl)pyridine-4-boronic acid pinacol ester 2-Cyano-6-(trifluoromethyl)pyridine-4-boronic acid pinacol ester 2223035-07-0 C13H14BF3N2O2
2-Fluoro-6-(cyclopropyl)pyridine 2-Fluoro-6-(cyclopropyl)pyridine 1563529-53-2 C8H8FN
2-fluoro-6-(tetrahydro-2H-pyran-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2-fluoro-6-(tetrahydro-2H-pyran-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2223008-74-8 C16H23BFNO3
2-fluoro-6-(tetrahydrofuran-3-yl)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2-fluoro-6-(tetrahydrofuran-3-yl)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2223009-11-6 C15H21BFNO3
2-Fluoro-6-cyanopyridine-3-boronic acid pinacol ester 2-Fluoro-6-cyanopyridine-3-boronic acid pinacol ester 2223049-37-2 C12H14BFN2O2
2-Hydroxy-4-(1H-2-methylimidazol-1-yl)-6-(iso-propyl)pyrimidine 2-Hydroxy-4-(1H-2-methylimidazol-1-yl)-6-(iso-propyl)pyrimidine 1412953-39-9 C11H14N4O
2-hydroxy-4-(cyclohexyl)-6-(tert-butyl)pyrimidine 2-hydroxy-4-(cyclohexyl)-6-(tert-butyl)pyrimidine 1412954-14-3 C14H22N2O
2-Hydroxy-5-(3,4-difluorophenyl)pyrazine 2-Hydroxy-5-(3,4-difluorophenyl)pyrazine 1159819-04-1 C10H6F2N2O
2-isopropoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-isopropoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1309981-65-4 C13H21BN2O3
2-isopropyl-1-propyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2-isopropyl-1-propyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223047-83-2 C15H27BN2O2
2-Methoxy-4-(piperidin-1-yl)phenylboronic acid pinacol ester 2-Methoxy-4-(piperidin-1-yl)phenylboronic acid pinacol ester 1366131-52-3 C18H28BNO3
2-Methyl-5-ethylpyridine-3-boronic acid pinacol ester 2-Methyl-5-ethylpyridine-3-boronic acid pinacol ester 2223046-89-5 C14H22BNO2
2-propyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-propyl-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2223027-33-4 C13H21BN2O2
3-(1H-pyrazol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 3-(1H-pyrazol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 2223030-92-8 C16H18BN3O2
3-(2-FLUOROPHENYL)PYRIDIN-2-AMINE 3-(2-FLUOROPHENYL)PYRIDIN-2-AMINE 1214367-39-1 C11H9FN2
3-(4-methylpiperidin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 3-(4-methylpiperidin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 2223045-79-0 C19H27BN2O2
3-(4-Trifluoromethylphenyl)pyridine-2-boronic acid pinacol ester 3-(4-Trifluoromethylphenyl)pyridine-2-boronic acid pinacol ester 2223012-90-4 C18H19BF3NO2
3-(N-Boc-Piperidin-4-yl)-4-methylphenylboronic acid pinacol ester 3-(N-Boc-Piperidin-4-yl)-4-methylphenylboronic acid pinacol ester 2223051-66-7 C23H36BNO4
3-(piperidin-4-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 3-(piperidin-4-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2223042-22-4 C17H27BN2O2
3,4-Dibromo-6-cyclopropylpyridine 3,4-Dibromo-6-cyclopropylpyridine 1353856-17-3 C8H7Br2N
3-Amino-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 3-Amino-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 2223041-13-0 C22H35BN2O4
3-Bromo-4-(3-thienyl)-2-pyridinecarbonitrile 3-Bromo-4-(3-thienyl)-2-pyridinecarbonitrile 1622844-19-2 C10H5BrN2S
3-Bromo-4-ethyl-2-chloropyridine 3-Bromo-4-ethyl-2-chloropyridine 1622843-50-8 C7H7BrClN
3-Bromo-5-(thiazol-4-yl)phenylboronic acid pinacol ester 3-Bromo-5-(thiazol-4-yl)phenylboronic acid pinacol ester 2223047-67-2 C15H17BBrNO2S
3-Chloro-5-(pyrazin-2-yl)phenylboronic acid pinacol ester 3-Chloro-5-(pyrazin-2-yl)phenylboronic acid pinacol ester 2223043-93-2 C16H18BClN2O2
3-Trifluoromethyl-4-(piperidin-4-yl)phenylboronic acid pinacol ester 3-Trifluoromethyl-4-(piperidin-4-yl)phenylboronic acid pinacol ester 2223036-92-6 C18H25BF3NO2
4-(1H-Pyrazol-1-yl)thiophene-2-boronic acid pinacol ester 4-(1H-Pyrazol-1-yl)thiophene-2-boronic acid pinacol ester 2223029-59-0 C13H17BN2O2S
4-(2-bromo-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(2-bromo-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223039-37-8 C17H25BBrNO2
4-(2-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(2-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223054-78-0 C18H28BNO3
4-(3-bromo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(3-bromo-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223042-16-6 C17H25BBrNO2
4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3'-bipyridine 4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2,3'-bipyridine 2223036-42-6 C16H19BN2O2
4-(4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223041-78-7 C18H28BNO2
4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)phenyl)piperidine 4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)phenyl)piperidine 2223042-15-5 C18H25BF3NO2
4-(tetrahydro-2H-pyran-3-yl)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 4-(tetrahydro-2H-pyran-3-yl)-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2223008-83-9 C17H26BNO3
4,4,5,5-tetramethyl-2-(2-(tetrahydro-2H-pyran-3-yl)-4-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(2-(tetrahydro-2H-pyran-3-yl)-4-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 2223005-62-5 C18H24BF3O3
4,4,5,5-tetramethyl-2-(4-(tetrahydro-2H-pyran-3-yl)furan-2-yl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(4-(tetrahydro-2H-pyran-3-yl)furan-2-yl)-1,3,2-dioxaborolane 2223003-63-0 C15H23BO4
4,4,5,5-tetramethyl-2-(5-methyl-2-(tetrahydro-2H-pyran-3-yl)phenyl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(5-methyl-2-(tetrahydro-2H-pyran-3-yl)phenyl)-1,3,2-dioxaborolane 2223003-87-8 C18H27BO3
4,6-Dichloro-2-(3-thienyl)pyrimidine 4,6-Dichloro-2-(3-thienyl)pyrimidine 57059-14-0 C8H4Cl2N2S
4-Amino-2-cyclopropyl-6-(2-thienyl)pyrimidine 4-Amino-2-cyclopropyl-6-(2-thienyl)pyrimidine 1247492-19-8 C11H11N3S
4-amino-2-cyclopropyl-6-(n-propyl)pyrimidine 4-amino-2-cyclopropyl-6-(n-propyl)pyrimidine 1412955-89-5 C10H15N3
4-Amino-6-(cyclopentyl)pyridine-3-boronic acid pinacol ester 4-Amino-6-(cyclopentyl)pyridine-3-boronic acid pinacol ester 2223037-52-1 C16H25BN2O2
4-Bromo-1-(n-propyl)-2-ethylimidazole 4-Bromo-1-(n-propyl)-2-ethylimidazole 1622840-74-7 C8H13BrN2
4-Bromo-1-(piperidin-4-yl)-2-methylimidazole 4-Bromo-1-(piperidin-4-yl)-2-methylimidazole 1622839-68-2 C9H14BrN3
4-Bromo-2-(4-methoxyphenyl)pyrimidine 4-Bromo-2-(4-methoxyphenyl)pyrimidine 164738-63-0 C11H9BrN2O
4-Bromo-2,6-dicyanopyridine 4-Bromo-2,6-dicyanopyridine 1643577-45-0 C7H2BrN3
4-bromo-2-methyl-6-(3-thienyl)pyrimidine 4-bromo-2-methyl-6-(3-thienyl)pyrimidine 1412957-78-8 C9H7BrN2S
4-BROMO-2-METHYL-N-ACETYL-IMIDAZOLE 4-BROMO-2-METHYL-N-ACETYL-IMIDAZOLE 1434127-05-5 C6H7BrN2O
4-Bromo-5-fluoropicolinonitrile 4-Bromo-5-fluoropicolinonitrile 1211582-95-4 C6H2BrFN2
4-Chloro-2-(3,4-difluorophenyl)pyrimidine 4-Chloro-2-(3,4-difluorophenyl)pyrimidine 1156585-24-8 C10H5ClF2N2
4-Chloro-2-(3-furan)pyrimidine 4-Chloro-2-(3-furan)pyrimidine 1260803-07-3 C8H5ClN2O
4-Chloro-6-(1H-pyridin-2-one)pyrimidine 4-Chloro-6-(1H-pyridin-2-one)pyrimidine 959240-43-8 C9H6ClN3O
4-Cyclopropyl-3-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 4-Cyclopropyl-3-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2223051-86-1 C18H23BN2O2
4-Fluoro-2-(3-trifluoromethylphenyl)pyridine 4-Fluoro-2-(3-trifluoromethylphenyl)pyridine 1261771-30-5 C12H7F4N
4-Hydroxy-2-(2-furyl)pyrimidine 4-Hydroxy-2-(2-furyl)pyrimidine 27110-98-1 C8H6N2O2
4-Hydroxy-2-methyl-6-(1H-pyridin-2-one)pyrimidine 4-Hydroxy-2-methyl-6-(1H-pyridin-2-one)pyrimidine 1412955-49-7 C10H9N3O2
4-Hydroxy-6-(3-chlorophenyl)-2-(iso-propyl)pyrimidine 4-Hydroxy-6-(3-chlorophenyl)-2-(iso-propyl)pyrimidine 1412956-01-4 C13H13ClN2O
4-methyl-2-(tetrahydro-2H-pyran-4-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 4-methyl-2-(tetrahydro-2H-pyran-4-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 2223029-24-9 C15H24BNO3S
4-Methyl-3-chloropyridine-5-boronic acid pinacol ester 4-Methyl-3-chloropyridine-5-boronic acid pinacol ester 2223051-94-1 C12H17BClNO2
5-(1H-Pyrazol-1-yl)thiophene-2-boronic acid pinacol ester 5-(1H-Pyrazol-1-yl)thiophene-2-boronic acid pinacol ester 2223032-96-8 C13H17BN2O2S
5-(2-Aminopropan-2-yl)pyrazine-2-boronic acid pinacol ester 5-(2-Aminopropan-2-yl)pyrazine-2-boronic acid pinacol ester 2223035-92-3 C13H22BN3O2
5-(3-Fluorophenyl)-2-hydroxypyrazine 5-(3-Fluorophenyl)-2-hydroxypyrazine 1159818-89-9 C10H7FN2O
5-(Imidazol-1-yl)thiophene-2-boronic acid pinacol ester 5-(Imidazol-1-yl)thiophene-2-boronic acid pinacol ester 2223051-07-6 C13H17BN2O2S
5-(iso-Propyl)-2-trifluoromethylpyridine-4-boronic acid pinacol ester 5-(iso-Propyl)-2-trifluoromethylpyridine-4-boronic acid pinacol ester 2223045-26-7 C15H21BF3NO2
5,5'-Dibromo-2,2'-bipyrazine 5,5'-Dibromo-2,2'-bipyrazine 1622840-94-1 C8H4Br2N4
5-Amino-2-(4-fluorophenyl)pyrimidine 5-Amino-2-(4-fluorophenyl)pyrimidine 1260777-61-4 C10H8FN3
5-Amino-2-(ethoxy)thiazole 5-Amino-2-(ethoxy)thiazole 1314355-67-3 C5H8N2OS
5-Bromo-2-(diethylamino)thiazole 5-Bromo-2-(diethylamino)thiazole 959240-16-5 C7H11BrN2S
6-(Tetrahydrofuran-3-yloxy)pyrazine-2-boronic acid pinacol ester 6-(Tetrahydrofuran-3-yloxy)pyrazine-2-boronic acid pinacol ester 1402166-47-5 C14H21BN2O4
6-Chloro-5-(3-hydroxypyrrolidin-1-yl)pyridine-3-boronic acid pinacol ester 6-Chloro-5-(3-hydroxypyrrolidin-1-yl)pyridine-3-boronic acid pinacol ester 2222996-42-9 C15H22BClN2O3
6-Chloro-5-(pyridin-4-yl)pyridine-3-boronic acid pinacol ester 6-Chloro-5-(pyridin-4-yl)pyridine-3-boronic acid pinacol ester 2223049-84-9 C16H18BClN2O2
6-Chloro-5-phenylpyridine-3-boronic acid pinacol ester 6-Chloro-5-phenylpyridine-3-boronic acid pinacol ester 2223049-76-9 C17H19BClNO2
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