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Pharmaceutical intermediates

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Structure Chemical Name CAS MF
6-Methyl-5-(tert-butyl)pyridine-3-boronic acid pinacol ester 6-Methyl-5-(tert-butyl)pyridine-3-boronic acid pinacol ester 2223031-95-4 C16H26BNO2
methyl 6-(tetrahydrofuran-2-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate methyl 6-(tetrahydrofuran-2-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 2223009-06-9 C17H24BNO5
N,N-bis(methyl-d3)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-amine N,N-bis(methyl-d3)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazin-2-amine 2241876-93-5 C12H20BN3O2
tert-butyl 4-(2-(methoxycarbonyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate tert-butyl 4-(2-(methoxycarbonyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate 2223045-55-2 C24H36BNO6
tert-butyl 4-(2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazol-1-yl)piperidine-1-carboxylate tert-butyl 4-(2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazol-1-yl)piperidine-1-carboxylate 2223034-00-0 C22H38BN3O4
tert-butyl 4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazol-2-yl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazol-2-yl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2241876-22-0 C18H30BN3O4S
tert-butyl 4-(4-cyclopropyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate tert-butyl 4-(4-cyclopropyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine-1-carboxylate 2256708-97-9 C25H38BNO4
(4-(1H-imidazol-1-yl-d3)phenyl)boronic acid (4-(1H-imidazol-1-yl-d3)phenyl)boronic acid 2256709-39-2 C9H9BN2O2
(5-(4-(methyl-d3)piperazin-1-yl)thiophen-2-yl)boronic acid (5-(4-(methyl-d3)piperazin-1-yl)thiophen-2-yl)boronic acid 2256709-46-1 C9H15BN2O2S
1-(2-(methoxy-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-4-(methyl-d3)piperazine-2,2,3,3,5,5,6,6-d8 1-(2-(methoxy-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-4-(methyl-d3)piperazine-2,2,3,3,5,5,6,6-d8 2256705-20-9 C18H29BN2O3
1-(2-bromo-5-cyclopropylphenyl)piperidine 1-(2-bromo-5-cyclopropylphenyl)piperidine 2222937-84-8 C14H18BrN
1-(2-bromophenyl)-1H-pyrazole-3,4,5-d3 1-(2-bromophenyl)-1H-pyrazole-3,4,5-d3 2256712-39-5 C9H7BrN2
1-(2-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-4-(methyl-d3)piperazine-2,2,3,3,5,5,6,6-d8 1-(2-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-4-(methyl-d3)piperazine-2,2,3,3,5,5,6,6-d8 2256705-27-6 C20H31BN2O2
1-(3-(methoxy-d3)phenyl-2,4,5,6-d4)-2-(methyl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 1-(3-(methoxy-d3)phenyl-2,4,5,6-d4)-2-(methyl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 2256710-57-1 C17H23BN2O3
1-(3-bromo-5-cyclopropylphenyl)-1H-imidazole 1-(3-bromo-5-cyclopropylphenyl)-1H-imidazole 1622843-97-3 C12H11BrN2
1-(3-chlorophenyl)-1H-imidazol-2-amine 1-(3-chlorophenyl)-1H-imidazol-2-amine 1698675-45-4 C9H8ClN3
1-(3-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-4-(methyl-d3)piperazine-2,2,3,3,5,5,6,6-d8 1-(3-methoxy-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-4-(methyl-d3)piperazine-2,2,3,3,5,5,6,6-d8 2256704-69-3 C18H18BD11N2O3
1-(4-(methoxy-d3)phenyl-2,3,5,6-d4)-2-(methyl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 1-(4-(methoxy-d3)phenyl-2,3,5,6-d4)-2-(methyl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 2256710-55-9 C17H23BN2O3
1-(4-bromo-3-cyclopropylphenyl)-1H-imidazole 1-(4-bromo-3-cyclopropylphenyl)-1H-imidazole 2222937-31-5 C12H11BrN2
1-(4-bromophenyl-2,3,5,6-d4)-2-(methyl-d3)-1H-imidazole-4,5-d2 1-(4-bromophenyl-2,3,5,6-d4)-2-(methyl-d3)-1H-imidazole-4,5-d2 2256712-97-5 C10BrD9N2
1-(4-Bromothiazol-2-yl)-4-bromoimidazole 1-(4-Bromothiazol-2-yl)-4-bromoimidazole 1353853-42-5 C6H3Br2N3S
1-(4-fluorophenyl-2,3,5,6-d4)-2-(methyl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 1-(4-fluorophenyl-2,3,5,6-d4)-2-(methyl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 2256710-67-3 C16H20BFN2O2
1-(4-methoxy-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-4-(methyl-d3)piperazine-2,2,3,3,5,5,6,6-d8 1-(4-methoxy-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-4-(methyl-d3)piperazine-2,2,3,3,5,5,6,6-d8 2256704-26-2 C18H29BN2O3
1-(5-Bromo-2-pyrazyl)-4-bromopyrazole 1-(5-Bromo-2-pyrazyl)-4-bromopyrazole 1353857-17-6 C7H4Br2N4
1-(6-Amino-2-pyrazyl)-4-bromoimidazole 1-(6-Amino-2-pyrazyl)-4-bromoimidazole 1353856-79-7 C7H6BrN5
1-(6-Bromo-2-pyrazyl)-4-bromoimidazole 1-(6-Bromo-2-pyrazyl)-4-bromoimidazole 1353855-84-1 C7H4Br2N4
1-(ethyl-d5)piperazine 1-(ethyl-d5)piperazine 1246817-21-9 C6H14N2
1-(methyl-d3)-1H-imidazol-2-amine 1-(methyl-d3)-1H-imidazol-2-amine 2294946-96-4 C4H7N3
1-(methyl-d3)-4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)phenyl)piperazine-2,2,3,3,5,5,6,6-d8 1-(methyl-d3)-4-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-2-(trifluoromethyl)phenyl)piperazine-2,2,3,3,5,5,6,6-d8 2256704-53-5 C18H15BD11F3N2O2
1-(methyl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 1-(methyl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 2256704-31-9 C10H12BD5N2O2
1-(methyl-d3)piperazine-2,5-dione-3,3,6,6-d4 1-(methyl-d3)piperazine-2,5-dione-3,3,6,6-d4 2259315-86-9 C5H8N2O2
1-(phenyl-d5)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 1-(phenyl-d5)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-2,5-d2 2256710-81-1 C15H19BN2O2
1-(Piperidin-4-yl)-2-(1-methylethyl)-1H-imidazol-4-amine 1-(Piperidin-4-yl)-2-(1-methylethyl)-1H-imidazol-4-amine 1622843-72-4 C11H20N4
1-(Thiazol-2-yl)-4-bromoimidazole 1-(Thiazol-2-yl)-4-bromoimidazole 1353855-33-0 C6H4BrN3S
1,3-Dibromo-5-(N-Boc-piperidin-4-yl)benzene 1,3-Dibromo-5-(N-Boc-piperidin-4-yl)benzene 1563533-29-8 C16H21Br2NO2
1-cyclopentyl-1,3-dihydro-2H-imidazol-2-one 1-cyclopentyl-1,3-dihydro-2H-imidazol-2-one 1505495-60-2 C8H12N2O
1-Methyl-2-(1-methylethyl)-1H-imidazol-4-amine 1-Methyl-2-(1-methylethyl)-1H-imidazol-4-amine 1314973-79-9 C7H13N3
2-(1H-imidazol-1-yl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 2-(1H-imidazol-1-yl-d3)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 2256707-01-2 C12H16BN3O2S
2-(1H-imidazol-1-yl-d3)benzen-3,4,5,6-d4-amine 2-(1H-imidazol-1-yl-d3)benzen-3,4,5,6-d4-amine 2256712-87-3 C9H9N3
2-(1H-imidazol-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(1H-imidazol-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2256755-57-2 C13H17BN4O2
2-(1H-pyrazol-1-yl-d3)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine-3,5-d2 2-(1H-pyrazol-1-yl-d3)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine-3,5-d2 2256709-59-6 C13H12BD5N4O2
2-(2-bromophenyl)pyrazine-3,5,6-d3 2-(2-bromophenyl)pyrazine-3,5,6-d3 2256711-16-5 C10H7BrN2
2-(2-bromophenyl)tetrahydro-2H-pyran 2-(2-bromophenyl)tetrahydro-2H-pyran 1784614-86-3 C11H13BrO
2-(2-FLUOROPHENYL)PYRIDIN-3-AMINE 2-(2-FLUOROPHENYL)PYRIDIN-3-AMINE 1214351-77-5 C11H9FN2
2-(3-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-1H-imidazole 2-(3-methyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-1H-imidazole 2256755-93-6 C16H21BN2O2
2-(4-bromo-1H-imidazol-1-yl-2,5-d2)pyrazine-3,5,6-d3 2-(4-bromo-1H-imidazol-1-yl-2,5-d2)pyrazine-3,5,6-d3 2256710-98-0 C7H5BrN4
2-(4-bromo-2-oxo-2,3-dihydro-1H-imidazol-1-yl)benzonitrile 2-(4-bromo-2-oxo-2,3-dihydro-1H-imidazol-1-yl)benzonitrile 2294956-90-2 C10H6BrN3O
2-(4-bromophenyl)pyrazine-3,5,6-d3 2-(4-bromophenyl)pyrazine-3,5,6-d3 2256712-16-8 C10H7BrN2
2-(4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-1H-imidazole 2-(4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)-1H-imidazole 2256755-99-2 C16H21BN2O2
2-(Cyclopropyl)-5-(4-tetrahydropyranyl)chlorobenzene 2-(Cyclopropyl)-5-(4-tetrahydropyranyl)chlorobenzene 1434127-20-4 C14H17ClO
2-(methyl-d3)-1-(2-(methyl-d3)phenyl-3,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 2-(methyl-d3)-1-(2-(methyl-d3)phenyl-3,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 2256710-61-7 C17H12BD11N2O2
2-(methyl-d3)-5-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazol-1-yl-2,5-d2)pyrazine 2-(methyl-d3)-5-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazol-1-yl-2,5-d2)pyrazine 2256705-88-9 C14H14BD5N4O2
2-(methyl-d3)-6-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl-4,5-d2)pyrazine-3,5-d2 2-(methyl-d3)-6-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl-4,5-d2)pyrazine-3,5-d2 2256705-93-6 C14H12BD7N4O2
2-(N-Boc-Piperidin-4-yl)-5-bromo-1-chlorobenzene 2-(N-Boc-Piperidin-4-yl)-5-bromo-1-chlorobenzene 1563532-59-1 C16H21BrClNO2
2-(propoxy-d7)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine-3,6-d2 2-(propoxy-d7)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine-3,6-d2 2241876-59-3 C13H21BN2O3
2,3-Dibromo-4-(4-fluorophenyl)pyridine 2,3-Dibromo-4-(4-fluorophenyl)pyridine 1381933-82-9 C11H6Br2FN
2,4-dibromo-1H-imidazole-5-d 2,4-dibromo-1H-imidazole-5-d 2256713-27-4 C3HBr2DN2
2,5-Diiodopyrimidine 2,5-Diiodopyrimidine 1261658-49-4 C4H2I2N2
2-Amino-4-(2-methyl-4-fluorophenyl)pyridine 2-Amino-4-(2-methyl-4-fluorophenyl)pyridine 1417518-94-5 C12H11FN2
2-AMINO-4-(2-PYRIDYL)PYRIDINE 2-AMINO-4-(2-PYRIDYL)PYRIDINE 1159816-51-9 C10H9N3
2-Amino-4-(3-methyl-1H-pyrazol-1-yl)thiazole 2-Amino-4-(3-methyl-1H-pyrazol-1-yl)thiazole 1314357-06-6 C7H8N4S
2-Amino-4-(N-Boc-piperidin-3-yl)pyridine 2-Amino-4-(N-Boc-piperidin-3-yl)pyridine 1563530-10-8 C15H23N3O2
2-Amino-4-(piperidin-3-yl)-1,3,5-triazine 2-Amino-4-(piperidin-3-yl)-1,3,5-triazine 1622835-63-5 C8H13N5
Tetrahydrofurfuryl bromide Tetrahydrofurfuryl bromide 1192-30-9 C5H9BrO
2-Amino-4-chloro-6-(4-pyridyl)pyrimidine 2-Amino-4-chloro-6-(4-pyridyl)pyrimidine 53421-90-2 C9H7ClN4
2-Amino-5-(2-chlorophenyl)pyrimidine 2-Amino-5-(2-chlorophenyl)pyrimidine 947592-41-8 C10H8ClN3
2-Amino-5-(2-methylpiperidino)thiazole 2-Amino-5-(2-methylpiperidino)thiazole 1314357-13-5 C9H15N3S
2-Amino-5-(3-methylpiperidino)thiazole 2-Amino-5-(3-methylpiperidino)thiazole 1314357-14-6 C9H15N3S
2-Amino-5-(4-tetrahydropyranyl)bromobenzene 2-Amino-5-(4-tetrahydropyranyl)bromobenzene 1434128-19-4 C11H14BrNO
2-AMINO-5-(CYCLOBUTOXY)PYRIDINE 2-AMINO-5-(CYCLOBUTOXY)PYRIDINE 1250024-59-9 C9H12N2O
2-Amino-5-(oxan-4-yl)pyrimidine 2-Amino-5-(oxan-4-yl)pyrimidine 1547045-67-9 C9H13N3O
2-Amino-6-(2-furyl)pyrazine 2-Amino-6-(2-furyl)pyrazine 925677-91-4 C8H7N3O
2-Amino-6-(2-methylpiperidin-1-yl)pyrazine 2-Amino-6-(2-methylpiperidin-1-yl)pyrazine 1314356-96-1 C10H16N4
2-Amino-6-(3-furyl)pyrazine 2-Amino-6-(3-furyl)pyrazine 1159818-58-2 C8H7N3O
2-Amino-6-(N-Boc-piperidin-3-yl)pyrazine 2-Amino-6-(N-Boc-piperidin-3-yl)pyrazine 1563530-04-0 C14H22N4O2
2-Amino-6-(oxan-4-yl)pyrazine 2-Amino-6-(oxan-4-yl)pyrazine 1563531-25-8 C9H13N3O
2-bromo-1-(2-bromophenyl-3,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 2-bromo-1-(2-bromophenyl-3,4,5,6-d4)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-5-d 2256703-99-6 C15H17BBr2N2O2
2-bromo-1-(methyl-d3)-1H-imidazole-4,5-d2 2-bromo-1-(methyl-d3)-1H-imidazole-4,5-d2 2294946-81-7 C4BrD5N2
2-Bromo-4-chloro-6-(2-thienyl)pyrimidine 2-Bromo-4-chloro-6-(2-thienyl)pyrimidine 1434128-12-7 C8H4BrClN2S
2-Bromo-5-(1-Boc-piperidin-4-yl)pyrazine 2-Bromo-5-(1-Boc-piperidin-4-yl)pyrazine 1159816-19-9 C14H20BrN3O2
2-Bromo-5-(2,4-difluorophenyl)pyridine 2-Bromo-5-(2,4-difluorophenyl)pyridine 1374664-71-7 C11H6BrF2N
2-Bromo-5-(3-chlorophenyl)pyridine 2-Bromo-5-(3-chlorophenyl)pyridine 1142193-80-3 C11H7BrClN
2-Bromo-5-(iso-propyl)thiophene 2-Bromo-5-(iso-propyl)thiophene 29488-23-1 C7H9BrS
2-Bromo-5-(N-Boc-piperidin-3-yl)pyrazine 2-Bromo-5-(N-Boc-piperidin-3-yl)pyrazine 1442101-44-1 C14H20BrN3O2
2-Bromo-5,6-dihydro-4H-pyran 2-Bromo-5,6-dihydro-4H-pyran 1622839-26-2 C5H7BrO
2-Bromo-5-amino-4-(iso-propyl)pyridine 2-Bromo-5-amino-4-(iso-propyl)pyridine 1381934-76-4 C8H11BrN2
2-bromo-6-(1H-imidazol-1-yl-d3)pyrazine 2-bromo-6-(1H-imidazol-1-yl-d3)pyrazine 2256707-17-0 C7H5BrN4
2-bromo-6-(1H-pyrazol-1-yl-d3)pyrazine-3,5-d2 2-bromo-6-(1H-pyrazol-1-yl-d3)pyrazine-3,5-d2 2256707-15-8 C7H5BrN4
2-Bromo-6-(2-methyl-4-thiazolyl)pyrazine 2-Bromo-6-(2-methyl-4-thiazolyl)pyrazine 1142196-90-4 C8H6BrN3S
2-Bromo-6-(2-thiazolylamino)pyridine 2-Bromo-6-(2-thiazolylamino)pyridine 439578-84-4 C8H6BrN3S
2-Bromo-6-(3-fluorophenyl)pyrazine 2-Bromo-6-(3-fluorophenyl)pyrazine 1142196-59-5 C10H6BrFN2
2-Bromo-6-(3-methylpiperidino)pyrazine 2-Bromo-6-(3-methylpiperidino)pyrazine 1027512-68-0 C10H14BrN3
2-Bromo-6-(4-methoxyphenyl)pyrazine 2-Bromo-6-(4-methoxyphenyl)pyrazine 1142196-73-3 C11H9BrN2O
2-Bromo-6-(cyclohexyl)pyrazine 2-Bromo-6-(cyclohexyl)pyrazine 1086383-04-1 C10H13BrN2
2-Bromo-6-(n-propoxy)pyrazine 2-Bromo-6-(n-propoxy)pyrazine 1027512-81-7 C7H9BrN2O
2-BROMO-6-ACETYLPYRAZINE 2-BROMO-6-ACETYLPYRAZINE 1197235-82-7 C6H5BrN2O
2-Chloro-4-(4-tetrahydropyranyl)bromobenzene 2-Chloro-4-(4-tetrahydropyranyl)bromobenzene 1434127-76-0 C11H12BrClO
2-Chloro-4-(piperidin-3-yl)-1,3,5-triazine 2-Chloro-4-(piperidin-3-yl)-1,3,5-triazine 1622835-51-1 C8H11ClN4
2-CHLORO-4-AMINO-3-(4-CYANOPHENYL)PYRIDINE 2-CHLORO-4-AMINO-3-(4-CYANOPHENYL)PYRIDINE 1563532-28-4 C12H8ClN3
2-CHLORO-5-(2-FLUOROPHENYL)PYRIMIDINE 2-CHLORO-5-(2-FLUOROPHENYL)PYRIMIDINE 1048338-45-9 C10H6ClFN2
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