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Pharmaceutical intermediates

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Structure Chemical Name CAS MF
1-benzyl-2-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 1-benzyl-2-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223045-05-2 C17H23BN2O2
1-cyclopentyl-2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 1-cyclopentyl-2-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223043-78-3 C17H29BN2O2
1-methyl-4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiophen-3-yl)piperazine 1-methyl-4-(5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiophen-3-yl)piperazine 2241864-99-1 C15H25BN2O2S
2-((2-(methyl-d3)propan-2-yl-1,1,1,3,3,3-d6)oxy)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-((2-(methyl-d3)propan-2-yl-1,1,1,3,3,3-d6)oxy)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2241876-71-9 C14H23BN2O3
2-(1H-pyrazol-1-yl)pyridine-5-boronic acid 2-(1H-pyrazol-1-yl)pyridine-5-boronic acid 1613187-72-6 C8H8BN3O2
2-(2-methoxy-4-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(2-methoxy-4-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2222997-42-2 C18H27BO4
2-(2-methyl-1H-imidazol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(2-methyl-1H-imidazol-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1309981-47-2 C14H19BN4O2
2-(3-(methyl-d3)phenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(3-(methyl-d3)phenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2241867-42-3 C17H21BN2O2
2-(3,4-difluorophenyl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(3,4-difluorophenyl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1402227-72-8 C16H17BF2N2O2
2-(3-cyclopropyl-4-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(3-cyclopropyl-4-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2223003-72-1 C20H29BO3
2-(3-fluorophenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(3-fluorophenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1402172-91-1 C16H18BFN2O2
2-(3-Methylpiperidin-1-yl)pyridine-4-boronic acid 2-(3-Methylpiperidin-1-yl)pyridine-4-boronic acid 2225152-63-4 C11H17BN2O2
2-(3-Pyridyl)pyridine-3-boronic acid pinacol ester 2-(3-Pyridyl)pyridine-3-boronic acid pinacol ester 2223045-78-9 C16H19BN2O2
2-(4-(methyl-d3)phenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(4-(methyl-d3)phenyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2241867-41-2 C17H18BD3N2O2
2-(4-cyclopropyl-3-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(4-cyclopropyl-3-(tetrahydro-2H-pyran-3-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2222997-54-6 C20H29BO3
2-(4-fluoro-3-(tetrahydro-2H-pyran-4-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2-(4-fluoro-3-(tetrahydro-2H-pyran-4-yl)phenyl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane 2223041-80-1 C17H24BFO3
2-(4-methyl-1H-pyrazol-1-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 2-(4-methyl-1H-pyrazol-1-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 1260152-83-7 C13H18BN3O2S
2-(4-methylpiperidin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(4-methylpiperidin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 1263152-91-5 C16H26BN3O2
2-(4-Tetrahydropyranyl)-4-cyanophenylboronic acid pinacol ester 2-(4-Tetrahydropyranyl)-4-cyanophenylboronic acid pinacol ester 2223040-01-3 C18H24BNO3
2-(Cyclohexyl)-6-(N-Boc-piperidin-3-yl)pyridine-4-boronic acid pinacol ester 2-(Cyclohexyl)-6-(N-Boc-piperidin-3-yl)pyridine-4-boronic acid pinacol ester 2222997-46-6 C27H43BN2O4
2-(Cyclopropyl)-6-(trifluoromethyl)pyridine-4-boronic acid 2-(Cyclopropyl)-6-(trifluoromethyl)pyridine-4-boronic acid 1446486-08-3 C9H9BF3NO2
2-(furan-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(furan-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2223048-58-4 C14H17BN2O3
2-(propoxy-d7)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(propoxy-d7)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2241876-69-5 C13H21BN2O3
2-(pyrrolidin-1-yl-d8)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(pyrrolidin-1-yl-d8)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2241876-98-0 C14H22BN3O2
2-(sec-Butyl)pyridine-3-boronic acid 2-(sec-Butyl)pyridine-3-boronic acid 2225153-53-5 C9H14BNO2
2-(tert-Butyl)-6-(piperidin-4-yl)pyridine-4-boronic acid 2-(tert-Butyl)-6-(piperidin-4-yl)pyridine-4-boronic acid 2225175-09-5 C14H23BN2O2
2-(tetrahydro-2H-pyran-3-yl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-(tetrahydro-2H-pyran-3-yl)-6-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2223005-28-3 C15H23BN2O3
2-(tetrahydro-2H-pyran-4-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2-(tetrahydro-2H-pyran-4-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2223030-23-5 C17H26BNO3
2,4-Dichloro-6-(5-pyrimidyl)pyrimidine 2,4-Dichloro-6-(5-pyrimidyl)pyrimidine 1353854-64-4 C8H4Cl2N4
2,5-Dibromo-4-(2-methylpiperidin-1-yl)pyridine 2,5-Dibromo-4-(2-methylpiperidin-1-yl)pyridine 1381933-51-2 C11H14Br2N2
2,5-Dibromo-4-(4-methylimidazol-1-yl)pyridine 2,5-Dibromo-4-(4-methylimidazol-1-yl)pyridine 1381935-68-7 C9H7Br2N3
2,5-Dibromo-4-(5-pyrimidyl)pyridine 2,5-Dibromo-4-(5-pyrimidyl)pyridine 1381943-28-7 C9H5Br2N3
2,6-Dibromo-3-(iso-propyl)pyridine 2,6-Dibromo-3-(iso-propyl)pyridine 1563529-72-5 C8H9Br2N
2-AMINO-3-(2-METHOXYPHENYL)PYRIDINE 2-AMINO-3-(2-METHOXYPHENYL)PYRIDINE 1344287-81-5 C12H12N2O
2-AMINO-3-(3,5-DIFLUOROPHENYL)PYRIDINE 2-AMINO-3-(3,5-DIFLUOROPHENYL)PYRIDINE 1343449-21-7 C11H8F2N2
2-Amino-4-(iso-propenyl)pyridine 2-Amino-4-(iso-propenyl)pyridine 1314354-79-4 C8H10N2
2-Amino-4-(tert-butyl)-6-methylpyridine 2-Amino-4-(tert-butyl)-6-methylpyridine 1247703-09-8 C9H15N3
2-Amino-5-(2-methylimidazol-1-yl)pyrazine 2-Amino-5-(2-methylimidazol-1-yl)pyrazine 1314353-53-1 C8H9N5
2-Amino-5-(2-trifluoromethylphenyl)pyrazine 2-Amino-5-(2-trifluoromethylphenyl)pyrazine 1125435-65-5 C11H8F3N3
2-Amino-5-(4-methylimidazol-1-yl)pyrazine 2-Amino-5-(4-methylimidazol-1-yl)pyrazine 1314356-48-3 C8H9N5
2-Amino-5-(4-tolyl)pyrazine 2-Amino-5-(4-tolyl)pyrazine 59489-73-5 C11H11N3
2-Amino-5-(N-Boc-piperidin-3-yl)phenylboronic acid pinacol ester 2-Amino-5-(N-Boc-piperidin-3-yl)phenylboronic acid pinacol ester 2223005-45-4 C22H35BN2O4
2-AMINO-6-(ETHOXYCARBONYL)PYRIDINE-4-BORONIC ACID PINACOL ESTER 2-AMINO-6-(ETHOXYCARBONYL)PYRIDINE-4-BORONIC ACID PINACOL ESTER 2223028-97-3 C14H21BN2O4
2-Bromo-4-(1H-pyrazol-1-yl)-6-methylpyrimidine 2-Bromo-4-(1H-pyrazol-1-yl)-6-methylpyrimidine 1412959-32-0 C8H7BrN4
2-Bromo-4-(1H-pyrazol-1-yl)thiophene 2-Bromo-4-(1H-pyrazol-1-yl)thiophene 1622839-52-4 C7H5BrN2S
2-Bromo-4-(2-methylimidazol-1-yl)furan 2-Bromo-4-(2-methylimidazol-1-yl)furan 1622840-61-2 C8H7BrN2O
2-Bromo-4-(3-methylpiperidin-1-yl)phenylboronic acid 2-Bromo-4-(3-methylpiperidin-1-yl)phenylboronic acid 2225151-94-8 C12H17BBrNO2
2-bromo-4-(4-chlorophenyl)-6-(tert-butyl)pyrimidine 2-bromo-4-(4-chlorophenyl)-6-(tert-butyl)pyrimidine 1412957-03-9 C14H14BrClN2
2-Bromo-4-(imidazol-1-yl)furan 2-Bromo-4-(imidazol-1-yl)furan 1622840-58-7 C7H5BrN2O
2-Bromo-4-(N-methylpiperazin-1-yl)furan 2-Bromo-4-(N-methylpiperazin-1-yl)furan 1622843-02-0 C9H13BrN2O
2-Bromo-4-(n-propyl)-6-(iso-propyl)pyrimidine 2-Bromo-4-(n-propyl)-6-(iso-propyl)pyrimidine 1412956-96-7 C10H15BrN2
2-bromo-4-(pyridin-3-yl)-6-cyclopropylpyrimidine 2-bromo-4-(pyridin-3-yl)-6-cyclopropylpyrimidine 1412961-42-2 C12H10BrN3
2-Bromo-4-chloro-5-(cyclobutyl)pyridine 2-Bromo-4-chloro-5-(cyclobutyl)pyridine 1381937-73-0 C9H9BrClN
2-Bromo-5-(1H-pyrazol-1-yl)furan 2-Bromo-5-(1H-pyrazol-1-yl)furan 1368328-75-9 C7H5BrN2O
2-Bromo-5-(2-methylimidazol-1-yl)thiophene 2-Bromo-5-(2-methylimidazol-1-yl)thiophene 1312099-62-9 C8H7BrN2S
2-Bromo-5-(2-thiazolylamino)pyrazine 2-Bromo-5-(2-thiazolylamino)pyrazine 1159820-26-4 C7H5BrN4S
2-Bromo-5-(3-methoxyphenyl)pyrazine 2-Bromo-5-(3-methoxyphenyl)pyrazine 1142196-01-7 C11H9BrN2O
2-Bromo-5-(3-pyridyl)pyrazine 2-Bromo-5-(3-pyridyl)pyrazine 1159819-77-8 C9H6BrN3
2-Bromo-5-(3-trifluoromethylphenyl)pyrazine 2-Bromo-5-(3-trifluoromethylphenyl)pyrazine 1142195-98-9 C11H6BrF3N2
2-Bromo-5-(4-methylpiperidin-1-yl)thiophene 2-Bromo-5-(4-methylpiperidin-1-yl)thiophene 1622842-88-9 C10H14BrNS
2-Bromo-5-(4-thiazolyl)pyrazine 2-Bromo-5-(4-thiazolyl)pyrazine 1142196-17-5 C7H4BrN3S
2-Bromo-5-(imidazol-1-yl)thiophene 2-Bromo-5-(imidazol-1-yl)thiophene 201656-11-3 C7H5BrN2S
2-Bromo-6-(4-methyl-1H-pyrazol-1-yl)pyrazine 2-Bromo-6-(4-methyl-1H-pyrazol-1-yl)pyrazine 1159816-83-7 C8H7BrN4
2-Bromo-6-(imidazol-1-yl)pyrazine 2-Bromo-6-(imidazol-1-yl)pyrazine 1086383-24-5 C7H5BrN4
2-Bromo-6-iodopyridine-4-boronic acid pinacol ester 2-Bromo-6-iodopyridine-4-boronic acid pinacol ester 2223011-60-5 C11H14BBrINO2
2-Chloro-3-(cyclohexyl)pyridine 2-Chloro-3-(cyclohexyl)pyridine 1417517-75-9 C11H14ClN
2-Chloro-4-(2-hydroxypiperidin-1-yl)-1,3,5-triazine 2-Chloro-4-(2-hydroxypiperidin-1-yl)-1,3,5-triazine 1417517-87-3 C8H11ClN4O
2-Chloro-4-(2-pyridyl)pyrimidine 2-Chloro-4-(2-pyridyl)pyrimidine 630423-85-7 C9H6ClN3
2-Chloro-4-(3-furyl)pyrimidine 2-Chloro-4-(3-furyl)pyrimidine 124959-29-1 C8H5ClN2O
2-Chloro-4-(3-tolyl)pyrimidine 2-Chloro-4-(3-tolyl)pyrimidine 954217-16-4 C11H9ClN2
2-Cyano-4-(4-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2-Cyano-4-(4-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2223037-11-2 C19H27BN2O2
2-Cyano-6-(oxan-3-yl)pyridine-4-boronic acid pinacol ester 2-Cyano-6-(oxan-3-yl)pyridine-4-boronic acid pinacol ester 2223009-64-9 C17H23BN2O3
2-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 1321518-37-9 C14H20BNO2
2-ethyl-1-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2-ethyl-1-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223048-04-0 C12H21BN2O2
2-Fluoro-4-(3-methyl-1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2-Fluoro-4-(3-methyl-1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2223047-57-0 C16H20BFN2O2
2-Fluoro-6-(2-tolyl)pyridine 2-Fluoro-6-(2-tolyl)pyridine 1356336-18-9 C12H10FN
2-Fluoro-6-(oxan-2-yl)pyridine-3-boronic acid pinacol ester 2-Fluoro-6-(oxan-2-yl)pyridine-3-boronic acid pinacol ester 2223009-63-8 C16H23BFNO3
2-hydroxy-4-(2-chlorophenyl)-6-methylpyrimidine 2-hydroxy-4-(2-chlorophenyl)-6-methylpyrimidine 1412954-76-7 C11H9ClN2O
2-Hydroxy-4-(2-fluorophenyl)pyrimidine 2-Hydroxy-4-(2-fluorophenyl)pyrimidine 952399-97-2 C10H7FN2O
2-isobutyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 2-isobutyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 905300-74-5 C13H22BNO2S
2-Methoxy-4-(4-methyl-1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2-Methoxy-4-(4-methyl-1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2223035-33-2 C17H23BN2O3
2-methyl-1-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethyl)phenyl)piperidine 2-methyl-1-(3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-5-(trifluoromethyl)phenyl)piperidine 2223004-50-8 C19H27BF3NO2
2-Methyl-5-trifluoromethylpyridine-3-boronic acid pinacol ester 2-Methyl-5-trifluoromethylpyridine-3-boronic acid pinacol ester 1356579-72-0 C13H17BF3NO2
3-(3-Methoxyphenyl)pyridine-2-boronic acid pinacol ester 3-(3-Methoxyphenyl)pyridine-2-boronic acid pinacol ester 2223050-68-6 C18H22BNO3
3-(5-Chloropyridin-2-yl)phenylboronic acid pinacol ester 3-(5-Chloropyridin-2-yl)phenylboronic acid pinacol ester 2223035-70-7 C17H19BClNO2
3-(N-Boc-Piperidin-3-yl)-5-aminophenylboronic acid pinacol ester 3-(N-Boc-Piperidin-3-yl)-5-aminophenylboronic acid pinacol ester 2222996-65-6 C22H35BN2O4
3-(pyrazin-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 3-(pyrazin-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 2223049-28-1 C17H18BN3O2
3-(tetrahydro-2H-pyran-3-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 3-(tetrahydro-2H-pyran-3-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)aniline 2223004-60-0 C17H26BNO3
3-Amino-6-methylpyridine-4-boronic acid pinacol ester 3-Amino-6-methylpyridine-4-boronic acid pinacol ester 1558927-35-7 C12H19BN2O2
3-Bromo-2-fluoro-6-ethylpyridine 3-Bromo-2-fluoro-6-ethylpyridine 1622839-40-0 C7H7BrFN
3-Bromo-5-(imidazol-1-yl)phenylboronic acid pinacol ester 3-Bromo-5-(imidazol-1-yl)phenylboronic acid pinacol ester 2223030-96-2 C15H18BBrN2O2
3-Bromo-6-(1-hydroxy-1-methylethyl)pyridazine 3-Bromo-6-(1-hydroxy-1-methylethyl)pyridazine 1303968-01-5 C7H9BrN2O
3-Cyano-5-(4-methyl-1H-pyrazol-1-yl)phenylboronic acid pinacol ester 3-Cyano-5-(4-methyl-1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2223053-19-6 C17H20BN3O2
3-Trifluoromethyl-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 3-Trifluoromethyl-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 2223042-01-9 C23H33BF3NO4
4-(2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(2-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223053-51-6 C17H25BFNO2
4-(4-Methylpiperidin-1-yl)furan-2-boronic acid pinacol ester 4-(4-Methylpiperidin-1-yl)furan-2-boronic acid pinacol ester 2223040-00-2 C16H26BNO3
4-(iso-Propyl)thiophene-2-boronic acid pinacol ester 4-(iso-Propyl)thiophene-2-boronic acid pinacol ester 2223033-13-2 C13H21BO2S
4-(N-Boc-Piperidin-4-yl)-3-chlorophenylboronic acid pinacol ester 4-(N-Boc-Piperidin-4-yl)-3-chlorophenylboronic acid pinacol ester 2223048-88-0 C22H33BClNO4
4-(Piperidino)thiophene-2-boronic acid pinacol ester 4-(Piperidino)thiophene-2-boronic acid pinacol ester 2223045-94-9 C15H24BNO2S
4,4,5,5-tetramethyl-2-(3-(tetrahydro-2H-pyran-4-yl)-4-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(3-(tetrahydro-2H-pyran-4-yl)-4-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 2223030-41-7 C18H24BF3O3
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