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Pharmaceutical intermediates

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Structure Chemical Name CAS MF
4-Amino-2-chloro-3-bromo-5-(3-furyl)pyridine 4-Amino-2-chloro-3-bromo-5-(3-furyl)pyridine 1563532-06-8 C9H6BrClN2O
4-Amino-2-chloro-3-bromo-5-(4-chlorophenyl)pyridine 4-Amino-2-chloro-3-bromo-5-(4-chlorophenyl)pyridine 1563533-44-7 C11H7BrCl2N2
4-Amino-2-methyl-1-(oxan-4-yl)-1H-imidazole 4-Amino-2-methyl-1-(oxan-4-yl)-1H-imidazole 1563532-42-2 C9H15N3O
4-Amino-2-phenyl-6-(5-thiazolyl)pyrimidine 4-Amino-2-phenyl-6-(5-thiazolyl)pyrimidine 1159818-61-7 C13H10N4S
4-Amino-3,5-dibromo-2-(2-methylpiperidin-1-yl)pyridine 4-Amino-3,5-dibromo-2-(2-methylpiperidin-1-yl)pyridine 1563530-08-4 C11H15Br2N3
4-bromo-1-(2-(trifluoromethyl)phenyl-3,4,5,6-d4)-1H-imidazole-2,5-d2 4-bromo-1-(2-(trifluoromethyl)phenyl-3,4,5,6-d4)-1H-imidazole-2,5-d2 2256710-38-8 C10H6BrF3N2
4-Bromo-1-(2-fluorophenyl)-1H-imidazole 4-Bromo-1-(2-fluorophenyl)-1H-imidazole 1353855-24-9 C9H6BrFN2
4-bromo-1-(2-fluorophenyl-3,4,5,6-d4)-2-(methyl-d3)-1H-imidazole-5-d 4-bromo-1-(2-fluorophenyl-3,4,5,6-d4)-2-(methyl-d3)-1H-imidazole-5-d 2256710-26-4 C10H8BrFN2
4-Bromo-1-(2-trifluoromethylphenyl)pyrazole 4-Bromo-1-(2-trifluoromethylphenyl)pyrazole 1353856-37-7 C10H6BrF3N2
4-bromo-1-(3-(methyl-d3)phenyl-2,4,5,6-d4)-1H-imidazole-2,5-d2 4-bromo-1-(3-(methyl-d3)phenyl-2,4,5,6-d4)-1H-imidazole-2,5-d2 2256710-52-6 C10BrD9N2
4-Bromo-1-(3-bromophenyl)imidazole 4-Bromo-1-(3-bromophenyl)imidazole 1363253-98-8 C9H6Br2N2
4-Bromo-1-(3-fluorophenyl)-1H-imidazole 4-Bromo-1-(3-fluorophenyl)-1H-imidazole 1353855-68-1 C9H6BrFN2
4-bromo-1-(4-bromophenyl)-1,3-dihydro-2H-imidazol-2-one 4-bromo-1-(4-bromophenyl)-1,3-dihydro-2H-imidazol-2-one 2294950-67-5 C9H6Br2N2O
4-Bromo-1-(4-trifluoromethylphenyl)-1H-imidazole 4-Bromo-1-(4-trifluoromethylphenyl)-1H-imidazole 1353856-15-1 C10H6BrF3N2
4-Bromo-1-(cyclopropyl)-1H-imidazole 4-Bromo-1-(cyclopropyl)-1H-imidazole 1353856-38-8 C6H7BrN2
4-Bromo-1-(oxan-4-yl)-2-ethylimidazole 4-Bromo-1-(oxan-4-yl)-2-ethylimidazole 1622843-87-1 C10H15BrN2O
4-Bromo-1-(oxolan-3-yl)-2-(iso-propyl)imidazole 4-Bromo-1-(oxolan-3-yl)-2-(iso-propyl)imidazole 1622834-81-4 C10H15BrN2O
4-bromo-1,2-bis(methyl-d3)-1H-imidazole-5-d 4-bromo-1,2-bis(methyl-d3)-1H-imidazole-5-d 2294945-67-6 C5BrD7N2
4-bromo-1-ethyl-2-fluoro-1H-imidazole 4-bromo-1-ethyl-2-fluoro-1H-imidazole 2294957-47-2 C5H6BrFN2
4-bromo-1-isopropyl-N,N-dimethyl-1H-imidazol-2-amine 4-bromo-1-isopropyl-N,N-dimethyl-1H-imidazol-2-amine 1894327-17-3 C8H14BrN3
4-bromo-2-(methoxy-d3)-1H-imidazole-5-d 4-bromo-2-(methoxy-d3)-1H-imidazole-5-d 2256713-25-2 C4H5BrN2O
4-bromo-2-(methyl-d3)-1-(3-(trifluoromethyl)phenyl-2,4,5,6-d4)-1H-imidazole-5-d 4-bromo-2-(methyl-d3)-1-(3-(trifluoromethyl)phenyl-2,4,5,6-d4)-1H-imidazole-5-d 2256710-32-2 C11H8BrF3N2
4-Bromo-2-(piperidin-3-yl)thiazole 4-Bromo-2-(piperidin-3-yl)thiazole 1622834-96-1 C8H11BrN2S
4-bromo-2-fluoro-1H-imidazole 4-bromo-2-fluoro-1H-imidazole 2294946-54-4 C3H2BrFN2
4-bromo-2-methyl-1-(m-tolyl)-1H-imidazole 4-bromo-2-methyl-1-(m-tolyl)-1H-imidazole 2294947-18-3 C11H11BrN2
4-Bromo-2-morpholino-1H-imidazole 4-Bromo-2-morpholino-1H-imidazole 1622840-62-3 C7H10BrN3O
4-BROMO-3-(2-METHYLPIPERIDIN-1-YL)PYRIDINE 4-BROMO-3-(2-METHYLPIPERIDIN-1-YL)PYRIDINE 1563529-91-8 C11H15BrN2
4-Bromo-3-(3,4-difluorophenyl)pyridine 4-Bromo-3-(3,4-difluorophenyl)pyridine 1374665-72-1 C11H6BrF2N
4-Bromo-3-(sec-butyl)pyridine 4-Bromo-3-(sec-butyl)pyridine 1374664-89-7 C9H12BrN
4-Bromo-3-amino-6-(3-chlorophenyl)pyridine 4-Bromo-3-amino-6-(3-chlorophenyl)pyridine 1381933-47-6 C11H8BrClN2
4-Bromo-5-(iso-propyl)pyrimidine 4-Bromo-5-(iso-propyl)pyrimidine 1563534-28-0 C7H9BrN2
4-Bromo-5-methyl-2-(ethyl)pyridine 4-Bromo-5-methyl-2-(ethyl)pyridine 1374665-55-0 C8H10BrN
4-Bromo-6-(n-propyl)pyrimidine 4-Bromo-6-(n-propyl)pyrimidine 1086382-11-7 C7H9BrN2
4-Bromo-6-cyclobutylpyrimidine 4-Bromo-6-cyclobutylpyrimidine 1086382-15-1 C8H9BrN2
4-Chloro-2-(3-fluorophenyl)pyridine 4-Chloro-2-(3-fluorophenyl)pyridine 1159814-60-4 C11H7ClFN
4-Chloro-3-(4-tetrahydropyranyl)benzonitrile 4-Chloro-3-(4-tetrahydropyranyl)benzonitrile 1434128-06-9 C12H12ClNO
4-Chloro-5-bromo-2-(tert-butoxy)pyrimidine 4-Chloro-5-bromo-2-(tert-butoxy)pyrimidine 57054-95-2 C8H10BrClN2O
4-Cyclopropyl-3-(1H-imidazol-1-yl)aniline 4-Cyclopropyl-3-(1H-imidazol-1-yl)aniline 1622838-94-1 C12H13N3
5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine-2-carbonitrile-3,6-d2 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine-2-carbonitrile-3,6-d2 2241876-52-6 C11H14BN3O2
5-(tetrahydro-2H-pyran-2-yl)pyrazin-2-amine 5-(tetrahydro-2H-pyran-2-yl)pyrazin-2-amine 1622835-69-1 C9H13N3O
5-(tetrahydrofuran-3-yl)pyrazin-2-ol 5-(tetrahydrofuran-3-yl)pyrazin-2-ol 2222934-75-8 C8H10N2O2
5-(Thiazol-4-yl)-1,3-dibromobenzene 5-(Thiazol-4-yl)-1,3-dibromobenzene 1563534-14-4 C9H5Br2NS
5-bromo-1-(2-methoxyphenyl)-1,3-dihydro-2H-imidazol-2-one 5-bromo-1-(2-methoxyphenyl)-1,3-dihydro-2H-imidazol-2-one 2294947-22-9 C10H9BrN2O2
5-bromo-1-(3-methoxyphenyl)-1,3-dihydro-2H-imidazol-2-one 5-bromo-1-(3-methoxyphenyl)-1,3-dihydro-2H-imidazol-2-one 2294948-47-1 C10H9BrN2O2
5-bromo-1-(p-tolyl)-1,3-dihydro-2H-imidazol-2-one 5-bromo-1-(p-tolyl)-1,3-dihydro-2H-imidazol-2-one 2294945-93-8 C10H9BrN2O
5-bromo-1-cyclohexyl-1,3-dihydro-2H-imidazol-2-one 5-bromo-1-cyclohexyl-1,3-dihydro-2H-imidazol-2-one 2294957-89-2 C9H13BrN2O
5-bromo-2-(ethoxy-d5)-1-(methyl-d3)-1H-imidazole-4-d 5-bromo-2-(ethoxy-d5)-1-(methyl-d3)-1H-imidazole-4-d 2294950-32-4 C6H9BrN2O
5-Bromo-2-(piperidin-3-yl)thiazole 5-Bromo-2-(piperidin-3-yl)thiazole 1521684-25-2 C8H11BrN2S
5-Bromo-4-methyl-2-(piperidino)thiazole 5-Bromo-4-methyl-2-(piperidino)thiazole 857549-60-1 C9H13BrN2S
6-(1-METHYL-1H-PYRAZOL-4-YL)PYRIDIN-3-AMINE 6-(1-METHYL-1H-PYRAZOL-4-YL)PYRIDIN-3-AMINE 1190380-28-9 C9H10N4
6-(2-FLUOROPHENYL)PYRIDIN-2-AMINE 6-(2-FLUOROPHENYL)PYRIDIN-2-AMINE 882014-37-1 C11H9FN2
6-(tetrahydrofuran-2-yl)pyrazin-2-amine 6-(tetrahydrofuran-2-yl)pyrazin-2-amine 2166863-29-0 C8H11N3O
6-Amino-8-(cyclopropyl)imidazo[1,2-a]pyrazine 6-Amino-8-(cyclopropyl)imidazo[1,2-a]pyrazine 1159821-57-4 C9H10N4
6-bromopyrazin-3,5-d2-2-ol 6-bromopyrazin-3,5-d2-2-ol 2259316-01-1 C4HBrD2N2O
1-(5-Bromopyrimidin-2-yl)azetidin-3-ol 1-(5-Bromopyrimidin-2-yl)azetidin-3-ol 1209222-50-3 C7H8BrN3O
Indazole-3-carboxylic acid Indazole-3-carboxylic acid 4498-67-3 C8H6N2O2
1-(2-Chloropyrimidin-4-yl)-4-piperidinol 1-(2-Chloropyrimidin-4-yl)-4-piperidinol 94222-07-8 C9H12ClN3O
2-(Piperazin-1-yl)-4,6-dichloropyrimidine 2-(Piperazin-1-yl)-4,6-dichloropyrimidine 1017781-91-7 C8H10Cl2N4
1-(5-Bromo-2-pyridinyl)-3-pyrrolidinol 1-(5-Bromo-2-pyridinyl)-3-pyrrolidinol 1159816-64-4 C9H11BrN2O
2-Bromo-6-cyclohexylaminopyridine 2-Bromo-6-cyclohexylaminopyridine 959237-36-6 C11H15BrN2
2-Methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6-(trifluoromethyl)pyridine 2-Methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-6-(trifluoromethyl)pyridine 1150561-66-2 C13H17BF3NO3
6-Bromo-2-cyclopropylaminopyridine 6-Bromo-2-cyclopropylaminopyridine 959237-20-8 C8H9BrN2
(R)-5,9-Bis(3,5-bis(trifluoromethyl)phenyl)-7-hydroxy-14,15,16,17-tetrahydrodiphenaleno[1,9-de:1',9'-fg][1,3,2]dioxaphosphocine 7-oxide (R)-5,9-Bis(3,5-bis(trifluoromethyl)phenyl)-7-hydroxy-14,15,16,17-tetrahydrodiphenaleno[1,9-de:1',9'-fg][1,3,2]dioxaphosphocine 7-oxide 2695533-33-4 C41H23F12O4P
N,N-dimethyl-2-((2-(4-(trifluoromethyl)phenyl)oxazolo[5,4-d]pyrimidin-7-yl)oxy)ethan-1-amine N,N-dimethyl-2-((2-(4-(trifluoromethyl)phenyl)oxazolo[5,4-d]pyrimidin-7-yl)oxy)ethan-1-amine C16H15F3N4O2
4-chloro-2-(4-(trifluoromethyl)phenyl)oxazolo[4,5-c]quinoline 4-chloro-2-(4-(trifluoromethyl)phenyl)oxazolo[4,5-c]quinoline 2406213-93-0 C17H8ClF3N2O
6-isopropylpyridine-3-boronic acid pinacol ester 6-isopropylpyridine-3-boronic acid pinacol ester 1105665-37-9 C14H22BNO2
4-Bromo-6-tert-butylpyrimidine 4-Bromo-6-tert-butylpyrimidine 19136-36-8 C8H11BrN2
1-Methyl-4-[[4-nitro-2-(trifluoromethyl)phenyl]methyl]-piperazine 1-Methyl-4-[[4-nitro-2-(trifluoromethyl)phenyl]methyl]-piperazine 694499-24-6 C13H16F3N3O2
3-Hydroxy-6-ethylpyridine 3-Hydroxy-6-ethylpyridine 51834-96-9 C7H9NO
(1S,4R)-4-(2-Amino-6-chloro-9H-purin-9-yl)-2-cyclopentene-1-carboxylate (1S,4R)-4-(2-Amino-6-chloro-9H-purin-9-yl)-2-cyclopentene-1-carboxylate 1246819-78-2 C11H10ClN5O2
6-Fluoro-4-nitro-3H-isobenzofuran-1-one 6-Fluoro-4-nitro-3H-isobenzofuran-1-one 1207453-90-4 C8H4FNO4
benzyl 3,3-difluorocyclobutanecarboxylate benzyl 3,3-difluorocyclobutanecarboxylate 935273-86-2 C12H12F2O2
3-bromo-1-(4-(trifluoromethyl)phenyl)-1H-pyrazole 3-bromo-1-(4-(trifluoromethyl)phenyl)-1H-pyrazole 1622839-69-3 C10H6BrF3N2
4-(Hydroxymethyl)-5-methyl-1,3-dioxol-2-one 4-(Hydroxymethyl)-5-methyl-1,3-dioxol-2-one 91526-18-0 C5H6O4
6-Hydroxy-8-methylimidazo[1,2-a]pyrazine 6-Hydroxy-8-methylimidazo[1,2-a]pyrazine 1159815-77-6 C7H7N3O
8-Bromo-6-(iso-propyl)imidazo[1,2-a]pyrazine 8-Bromo-6-(iso-propyl)imidazo[1,2-a]pyrazine 1159816-07-5 C9H10BrN3
8-Hydroxy-6-(3-thienyl)imidazo[1,2-a]pyrazine 8-Hydroxy-6-(3-thienyl)imidazo[1,2-a]pyrazine 1159816-50-8 C10H7N3OS
methyl 2-(1H-imidazol-2-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoate methyl 2-(1H-imidazol-2-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoate 2256755-70-9 C17H21BN2O4
methyl 2-(4-bromo-2-methoxy-1H-imidazol-1-yl)benzoate methyl 2-(4-bromo-2-methoxy-1H-imidazol-1-yl)benzoate 2294944-04-8 C12H11BrN2O3
methyl 2-(4-methylpiperazin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoate methyl 2-(4-methylpiperazin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoate 2256756-12-2 C19H29BN2O4
methyl 3-(2-amino-5-bromo-1H-imidazol-1-yl)benzoate methyl 3-(2-amino-5-bromo-1H-imidazol-1-yl)benzoate 2294957-16-5 C11H10BrN3O2
methyl 3-(4-bromo-2-methoxy-1H-imidazol-1-yl)benzoate methyl 3-(4-bromo-2-methoxy-1H-imidazol-1-yl)benzoate 2294946-13-5 C12H11BrN2O3
methyl 4-(4-bromo-2-oxo-2,3-dihydro-1H-imidazol-1-yl)benzoate methyl 4-(4-bromo-2-oxo-2,3-dihydro-1H-imidazol-1-yl)benzoate 2294957-35-8 C11H9BrN2O3
N,N-dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-sulfonamide-2,5-d2 N,N-dimethyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-sulfonamide-2,5-d2 2256703-92-9 C11H20BN3O4S
tert-butyl 2-(ethoxy-d5)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-carboxylate-5-d tert-butyl 2-(ethoxy-d5)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-carboxylate-5-d 2256711-53-0 C16H27BN2O5
TERT-BUTYL 3-(3-BROMO-4-METHOXYPHENYL)PIPERIDINE-1-CARBOXYLATE TERT-BUTYL 3-(3-BROMO-4-METHOXYPHENYL)PIPERIDINE-1-CARBOXYLATE 1563528-73-3 C17H24BrNO3
tert-butyl 3-(6-hydroxypyrazin-2-yl)pyrrolidine-1-carboxylate tert-butyl 3-(6-hydroxypyrazin-2-yl)pyrrolidine-1-carboxylate 2222934-81-6 C13H19N3O3
tert-butyl 4-(2-amino-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(2-amino-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2256704-94-4 C21H34BN3O4
tert-butyl 4-(2-bromophenyl)-1H-imidazole-1-carboxylate-2,5-d2 tert-butyl 4-(2-bromophenyl)-1H-imidazole-1-carboxylate-2,5-d2 2256711-77-8 C14H15BrN2O2
tert-butyl 4-(3-((methoxy-d3)carbonyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(3-((methoxy-d3)carbonyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2256705-12-9 C23H35BN2O6
tert-butyl 4-(3-(methoxycarbonyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(3-(methoxycarbonyl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2256705-11-8 C23H35BN2O6
tert-butyl 4-(3-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(3-chloro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2256704-87-5 C21H32BClN2O4
tert-butyl 4-(3-cyclopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(3-cyclopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2256705-13-0 C24H37BN2O4
tert-butyl 4-(4-(methyl-d3)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(4-(methyl-d3)-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2256704-06-8 C22H24BD11N2O4
tert-butyl 4-(4-amino-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(4-amino-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2256704-17-1 C21H34BN3O4
tert-butyl 4-(4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(4-methyl-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2256704-05-7 C22H35BN2O4
tert-butyl 4-(5-bromopyrazin-2-yl-3,6-d2)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 tert-butyl 4-(5-bromopyrazin-2-yl-3,6-d2)piperazine-1-carboxylate-2,2,3,3,5,5,6,6-d8 2259316-03-3 C13H9BrD10N4O2
tert-butyl 4-hydroxypiperidine-1-carboxylate-2,2,3,3,4,5,5,6,6-d9 tert-butyl 4-hydroxypiperidine-1-carboxylate-2,2,3,3,4,5,5,6,6-d9 1246342-61-9 C10H19NO3
tetrahydro-4H-pyran-4-one-2,2,3,3,5,5,6,6-d8 tetrahydro-4H-pyran-4-one-2,2,3,3,5,5,6,6-d8 2294956-89-9 C5D8O2
Cefotiam (6R,7S) isomer reference Cefotiam (6R,7S) isomer reference
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