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Pharmaceutical intermediates

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Structure Chemical Name CAS MF
2-Bromo-5-(4-tolyl)pyrazine 2-Bromo-5-(4-tolyl)pyrazine 1142195-89-8 C11H9BrN2
2-Bromo-6-(1H-pyrrol-1-yl)pyrazine 2-Bromo-6-(1H-pyrrol-1-yl)pyrazine 1027512-40-8 C8H6BrN3
2-Bromo-6-(4-methylimidazol-1-yl)pyridine 2-Bromo-6-(4-methylimidazol-1-yl)pyridine 1027512-12-4 C9H8BrN3
2-Bromo-6-(pyrrolidinon-1-yl)pyrazine 2-Bromo-6-(pyrrolidinon-1-yl)pyrazine 1027512-34-0 C8H8BrN3O
2-Chloro-3-(3-fluorophenyl)pyridine 2-Chloro-3-(3-fluorophenyl)pyridine 1214381-69-7 C11H7ClFN
2-Chloro-3-(sec-butyl)pyridine 2-Chloro-3-(sec-butyl)pyridine 1417519-68-6 C9H12ClN
2-chloro-4-(1H-4-methylpyrozol-1-yl)-6-(tert-butyl)pyrimidine 2-chloro-4-(1H-4-methylpyrozol-1-yl)-6-(tert-butyl)pyrimidine 1412957-56-2 C12H15ClN4
2-Chloro-4-(3-methylpiperidin-1-yl)-1,3,5-triazine 2-Chloro-4-(3-methylpiperidin-1-yl)-1,3,5-triazine 1417518-62-7 C9H13ClN4
2-Chloro-4-(4-tetrahydropyranyl)-1,3,5-triazine 2-Chloro-4-(4-tetrahydropyranyl)-1,3,5-triazine 1417519-72-2 C8H10ClN3O
2-chloro-4-(cyclopentyl)-6-(tert-butyl)pyrimidine 2-chloro-4-(cyclopentyl)-6-(tert-butyl)pyrimidine 1412960-79-2 C13H19ClN2
2-chloro-4,6-di(tert-butyl)pyrimidine 2-chloro-4,6-di(tert-butyl)pyrimidine 71162-19-1 C12H19ClN2
2-cyclopentyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2-cyclopentyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyrazine 2223048-41-5 C15H23BN2O2
2-Cyclopentyl-6-(oxan-4-yl)pyridine-4-boronic acid pinacol ester 2-Cyclopentyl-6-(oxan-4-yl)pyridine-4-boronic acid pinacol ester 2223045-80-3 C21H32BNO3
2-cyclopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3-(trifluoromethyl)pyridine 2-cyclopropyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-3-(trifluoromethyl)pyridine 1355071-84-9 C15H19BF3NO2
2-cyclopropyl-5-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2-cyclopropyl-5-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridine 2223041-03-8 C14H19BFNO2
2-ethyl-1-(tetrahydrofuran-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2-ethyl-1-(tetrahydrofuran-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223006-87-7 C15H25BN2O3
2-Fluoro-4-(3-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2-Fluoro-4-(3-methylpiperidin-1-yl)phenylboronic acid pinacol ester 2223004-34-8 C18H27BFNO2
2-Fluoro-6-bromopyridine-4-boronic acid pinacol ester 2-Fluoro-6-bromopyridine-4-boronic acid pinacol ester 2223035-36-5 C11H14BBrFNO2
2-Hydroxy-3-(2-trifluoromethylphenyl)pyridine 2-Hydroxy-3-(2-trifluoromethylphenyl)pyridine 426823-49-6 C12H8F3NO
2-Hydroxy-3-(iso-propyl)pyridine 2-Hydroxy-3-(iso-propyl)pyridine 1417519-11-9 C8H11NO
2-Hydroxy-4-(2-tolyl)-6-cyclopropylpyrimidine 2-Hydroxy-4-(2-tolyl)-6-cyclopropylpyrimidine 1412955-05-5 C14H14N2O
2-Hydroxy-5-(cyclobutyl)pyrazine 2-Hydroxy-5-(cyclobutyl)pyrazine 1159816-45-1 C8H10N2O
2-isopropyl-1-(tetrahydrofuran-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2-isopropyl-1-(tetrahydrofuran-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole 2223006-18-4 C16H27BN2O3
2-Trifluoromethyl-4-(N-methylpiperazin-1-yl)phenylboronic acid pinacol ester 2-Trifluoromethyl-4-(N-methylpiperazin-1-yl)phenylboronic acid pinacol ester 2223041-59-4 C18H26BF3N2O2
3-(3-FLUOROPHENYL)PYRIDIN-2-AMINE 3-(3-FLUOROPHENYL)PYRIDIN-2-AMINE 1214379-93-7 C11H9FN2
3-(3-methylpiperidin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 3-(3-methylpiperidin-1-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzonitrile 2223004-61-1 C19H27BN2O2
3-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-2-AMINE 3-(4-FLUORO-2-METHYLPHENYL)PYRIDIN-2-AMINE 1258608-61-5 C12H11FN2
3-(4-METHOXYPHENYL)PYRIDIN-2-AMINE 3-(4-METHOXYPHENYL)PYRIDIN-2-AMINE 1258618-76-6 C12H12N2O
3-(N-Boc-Piperidin-4-yl)-4-chlorophenylboronic acid pinacol ester 3-(N-Boc-Piperidin-4-yl)-4-chlorophenylboronic acid pinacol ester 2223055-36-3 C22H33BClNO4
3,6-Diiodo-4-bromopyridine 3,6-Diiodo-4-bromopyridine 1643543-81-0 C5H2BrI2N
3-Bromo-4-(1,4-dioxan-2-yl)pyridine 3-Bromo-4-(1,4-dioxan-2-yl)pyridine 1622834-36-9 C9H10BrNO2
3-Bromo-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 3-Bromo-5-(N-Boc-piperidin-4-yl)phenylboronic acid pinacol ester 2223033-78-9 C22H33BBrNO4
3-Chloro-4-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 3-Chloro-4-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2223049-03-2 C15H18BClN2O2
3-Cyano-5-(imidazol-1-yl)phenylboronic acid pinacol ester 3-Cyano-5-(imidazol-1-yl)phenylboronic acid pinacol ester 2223039-71-0 C16H18BN3O2
3-Fluoro-4-(piperidin-1-yl)phenylboronic acid pinacol ester 3-Fluoro-4-(piperidin-1-yl)phenylboronic acid pinacol ester 2223042-46-2 C17H25BFNO2
3-Fluoro-5-(piperazin-1-yl)phenylboronic acid pinacol ester 3-Fluoro-5-(piperazin-1-yl)phenylboronic acid pinacol ester 2223031-26-1 C16H24BFN2O2
3-Methyl-2-(n-propyl)pyridine-4-boronic acid pinacol ester 3-Methyl-2-(n-propyl)pyridine-4-boronic acid pinacol ester 2223036-16-4 C15H24BNO2
3-Trifluoromethyl-4-(N-Boc-piperidin-3-yl)phenylboronic acid pinacol ester 3-Trifluoromethyl-4-(N-Boc-piperidin-3-yl)phenylboronic acid pinacol ester 2222996-61-2 C23H33BF3NO4
4-(2-chloro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(2-chloro-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223042-08-6 C17H25BClNO2
4-(3-bromo-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(3-bromo-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223031-89-6 C17H25BBrNO2
4-(3-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(3-methoxy-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223053-57-2 C18H28BNO3
4-(4-chloro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(4-chloro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223052-82-0 C17H25BClNO2
4-(4-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 4-(4-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 2223031-88-5 C16H26BNO2S
4-(5-chloro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(5-chloro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223045-67-6 C17H25BClNO2
4-(5-methyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 4-(5-methyl-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl)piperidine 2223030-55-3 C18H28BNO2
4,4,5,5-tetramethyl-2-(2-(tetrahydro-2H-pyran-4-yl)-5-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(2-(tetrahydro-2H-pyran-4-yl)-5-(trifluoromethyl)phenyl)-1,3,2-dioxaborolane 2223031-61-4 C18H24BF3O3
4,4,5,5-tetramethyl-2-(4-(tetrahydro-2H-pyran-2-yl)thiophen-2-yl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(4-(tetrahydro-2H-pyran-2-yl)thiophen-2-yl)-1,3,2-dioxaborolane 2223005-72-7 C15H23BO3S
4,4,5,5-tetramethyl-2-(4-(tetrahydro-2H-pyran-4-yl)thiophen-2-yl)-1,3,2-dioxaborolane 4,4,5,5-tetramethyl-2-(4-(tetrahydro-2H-pyran-4-yl)thiophen-2-yl)-1,3,2-dioxaborolane 2223054-39-3 C15H23BO3S
4-Amino-2-(3-aminophenyl)pyrimidine 4-Amino-2-(3-aminophenyl)pyrimidine 1215072-62-0 C10H10N4
4-Amino-2-(3-methyl-1H-pyrazol-1-yl)thiazole 4-Amino-2-(3-methyl-1H-pyrazol-1-yl)thiazole 1314355-47-9 C7H8N4S
4-Amino-2-(cyclopentyl)pyrimidine 4-Amino-2-(cyclopentyl)pyrimidine 871823-79-9 C9H13N3
4-Amino-2-(iso-propenyl)pyridine 4-Amino-2-(iso-propenyl)pyridine 1314355-59-3 C8H10N2
4-Amino-2-cyclopropyl-6-(1H-pyrazol-1-yl)pyrimidine 4-Amino-2-cyclopropyl-6-(1H-pyrazol-1-yl)pyrimidine 1412957-58-4 C10H11N5
4-Bromo-1-(iso-butyl)-2-methylimidazole 4-Bromo-1-(iso-butyl)-2-methylimidazole 1622843-45-1 C8H13BrN2
4-Bromo-1-(oxan-3-yl)-2-methylimidazole 4-Bromo-1-(oxan-3-yl)-2-methylimidazole 1622836-16-1 C9H13BrN2O
4-Bromo-1-methyl-2-ethylimidazole 4-Bromo-1-methyl-2-ethylimidazole 1622843-93-9 C6H9BrN2
4-Bromo-2-(3-furan)pyrimidine 4-Bromo-2-(3-furan)pyrimidine 1086381-95-4 C8H5BrN2O
4-Bromo-2-(iso-propyl)-6-(1H-imidazol-1-yl)pyrimidine 4-Bromo-2-(iso-propyl)-6-(1H-imidazol-1-yl)pyrimidine 1412958-46-3 C10H11BrN4
4-Bromo-2-(iso-propyl)-6-(piperidin-1-yl)-pyrimidine 4-Bromo-2-(iso-propyl)-6-(piperidin-1-yl)-pyrimidine 1412960-60-1 C12H18BrN3
4-Bromo-2-(pyrrolidin-3-yl)-5-fluoropyridine 4-Bromo-2-(pyrrolidin-3-yl)-5-fluoropyridine 1643537-26-1 C9H10BrFN2
4-bromo-2,6-di(cyclopropyl)pyrimidine 4-bromo-2,6-di(cyclopropyl)pyrimidine 1412958-76-9 C10H11BrN2
4-Bromo-2-cyclopropyl-6-(4-chlorophenyl)pyrimidine 4-Bromo-2-cyclopropyl-6-(4-chlorophenyl)pyrimidine 1412957-88-0 C13H10BrClN2
4-bromo-2-cyclopropyl-6-methylpyrimidine 4-bromo-2-cyclopropyl-6-methylpyrimidine 1412953-04-8 C8H9BrN2
4-Bromo-2-methyl-6-(1H-pyridin-2-one)pyrimidine 4-Bromo-2-methyl-6-(1H-pyridin-2-one)pyrimidine 1412958-59-8 C10H8BrN3O
4-Bromo-3-fluoro-2-(pyrrolidin-3-yl)pyridine 4-Bromo-3-fluoro-2-(pyrrolidin-3-yl)pyridine 1643543-76-3 C9H10BrFN2
4-Cyclopropyl-2-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 4-Cyclopropyl-2-(1H-pyrazol-1-yl)phenylboronic acid pinacol ester 2223042-60-0 C18H23BN2O2
4-Cyclopropyl-3-(1H-imidazol-1-yl)phenylboronic acid pinacol ester 4-Cyclopropyl-3-(1H-imidazol-1-yl)phenylboronic acid pinacol ester 2223036-18-6 C18H23BN2O2
4-ethyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 4-ethyl-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)thiazole 2223035-41-2 C11H18BNO2S
4-Fluoro-2-(thiazol-5-yl)pyridine 4-Fluoro-2-(thiazol-5-yl)pyridine 1563530-69-7 C8H5FN2S
4-Fluoro-2-ethylpyridine 4-Fluoro-2-ethylpyridine 1563532-10-4 C7H8FN
4-Hydroxy-2-(3-methoxyphenyl)pyrimidine 4-Hydroxy-2-(3-methoxyphenyl)pyrimidine 1155597-76-4 C11H10N2O2
4-Hydroxy-2-cyclopropyl-6-(2-methylpiperidin-1-yl)pyrimidine 4-Hydroxy-2-cyclopropyl-6-(2-methylpiperidin-1-yl)pyrimidine 1412957-99-3 C13H19N3O
5-(1-Methyl-1-acetoxyethyl)thiophene-2-boronic acid pinacol ester 5-(1-Methyl-1-acetoxyethyl)thiophene-2-boronic acid pinacol ester 1402174-74-6 C15H23BO4S
5-(3,5-Difluorophenyl)pyrazine-2-boronic acid pinacol ester 5-(3,5-Difluorophenyl)pyrazine-2-boronic acid pinacol ester 1402227-69-3 C16H17BF2N2O2
5-(3-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 5-(3-Methylpiperidin-1-yl)thiophene-2-boronic acid pinacol ester 2223002-76-2 C16H26BNO2S
5-(3-Thienyl)-2-hydroxypyrazine 5-(3-Thienyl)-2-hydroxypyrazine 1159817-99-8 C8H6N2OS
5-(4-Methyl-1H-pyrazol-1-yl)pyridine-3-boronic acid pinacol ester 5-(4-Methyl-1H-pyrazol-1-yl)pyridine-3-boronic acid pinacol ester 1402240-21-4 C15H20BN3O2
5-(4-Pyridyl)-2-hydroxypyrazine 5-(4-Pyridyl)-2-hydroxypyrazine 1159819-68-7 C9H7N3O
5-(methyl-d3)pyrazin-3,6-d2-2-amine 5-(methyl-d3)pyrazin-3,6-d2-2-amine 1643542-47-5 C5H7N3
5-(N-Boc-Piperidin-4-yl)-2-fluorophenylboronic acid pinacol ester 5-(N-Boc-Piperidin-4-yl)-2-fluorophenylboronic acid pinacol ester 2223032-00-4 C22H33BFNO4
5-(tert-Butyl)-2-hydroxypyrazine 5-(tert-Butyl)-2-hydroxypyrazine 1159820-93-5 C8H12N2O
5-(Thiazol-4-yl)pyridine-3-boronic acid pinacol ester 5-(Thiazol-4-yl)pyridine-3-boronic acid pinacol ester 2223039-14-1 C14H17BN2O2S
5-Amino-2-(2-methylimidazol-1-yl)thiazole 5-Amino-2-(2-methylimidazol-1-yl)thiazole 1314355-60-6 C7H8N4S
5-Amino-2-(3-thienyl)pyrimidine 5-Amino-2-(3-thienyl)pyrimidine 1094373-81-5 C8H7N3S
5-Amino-2-(diethylamino)thiazole 5-Amino-2-(diethylamino)thiazole 791060-68-9 C7H13N3S
5-Bromo-6-(5-pyrimidyl)pyridine-3-boronic acid pinacol ester 5-Bromo-6-(5-pyrimidyl)pyridine-3-boronic acid pinacol ester 2223029-47-6 C15H17BBrN3O2
5-Cyclopropyl-2-trifluoromethylpyridine-4-boronic acid pinacol ester 5-Cyclopropyl-2-trifluoromethylpyridine-4-boronic acid pinacol ester 2223047-92-3 C15H19BF3NO2
5-Hydroxy-2-(1H-pyrrol-1-yl)pyrimidine 5-Hydroxy-2-(1H-pyrrol-1-yl)pyrimidine 1260812-32-5 C8H7N3O
5-Methyl-6-(tert-butyl)pyridine-3-boronic acid pinacol ester 5-Methyl-6-(tert-butyl)pyridine-3-boronic acid pinacol ester 2223048-02-8 C16H26BNO2
5-TERT-BUTYLPYRIDIN-3-OL 5-TERT-BUTYLPYRIDIN-3-OL 1243371-93-8 C9H13NO
6-(3,5-Difluorophenyl)pyrazine-2-boronic acid pinacol ester 6-(3,5-Difluorophenyl)pyrazine-2-boronic acid pinacol ester 1402227-71-7 C16H17BF2N2O2
6-(3-Tolyl)pyrazine-2-boronic acid pinacol ester 6-(3-Tolyl)pyrazine-2-boronic acid pinacol ester 1402172-33-1 C17H21BN2O2
6-Chloro-5-(cyclopentoxy)pyridine-3-boronic acid pinacol ester 6-Chloro-5-(cyclopentoxy)pyridine-3-boronic acid pinacol ester 2223030-22-4 C16H23BClNO3
6-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 6-cyclopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 2223046-66-8 C15H19BN2O2
6-Fluoro-5-bromopyridine-3-boronic acid pinacol ester 6-Fluoro-5-bromopyridine-3-boronic acid pinacol ester 2223038-87-5 C11H14BBrFNO2
6-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 6-isopropyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinonitrile 2223044-21-9 C15H21BN2O2
methyl 3-(tetrahydro-2H-pyran-3-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoate methyl 3-(tetrahydro-2H-pyran-3-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)benzoate 2223009-80-9 C19H27BO5
methyl 6-(tetrahydro-2H-pyran-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate methyl 6-(tetrahydro-2H-pyran-3-yl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 2223009-02-5 C18H26BNO5
methyl 6-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate methyl 6-fluoro-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)picolinate 2223042-14-4 C13H17BFNO4
tert-butyl 2-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-carboxylate tert-butyl 2-methyl-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-imidazole-1-carboxylate 1402174-60-0 C15H25BN2O4
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