1-AZAKENPAULLONE
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- $68 - $7363.82
- Product name: 1-AZAKENPAULLONE
- CAS: 676596-65-9
- MF: C15H10BrN3O
- MW: 328.16
- EINECS:200-258-5
- MDL Number:MFCD09037522
- Synonyms:1-AZAKENPAULLONE;9-Bromo-7,12-dihydropyrido[3',2':2,3]azepino[4,5-b]indol-6(5H)-one;Pyrido[3',2':2,3]azepino[4,5-b]indol-6(5H)-one, 9-broMo-7,12-dihydro-;InSolution? 1-Azakenpaullone ;1-Azakenpaullone 9-Bromo-7,12-dihydropyrido[3',2':2,3]azepino[4,5-b]indol-6(5H)-one;InSolution 1-Azakenpaullone - CAS 676596-65-9 - Calbiochem;1-Azakenpaullone - CAS 676596-65-9 - Calbiochem;azakenpaullone
76 prices
Selected condition:
Brand
- aablocks
- ACHEMBLOCK
- Adipogen Life Sciences
- American Custom Chemicals Corporation
- ApexBio Technology
- Biosynth
- Cayman Chemical
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Medical Isotopes, Inc.
- Sigma-Aldrich
- TRC
- Usbiological
Package
- 10mM(in1mLDMSO)
- 2mg
- 2.5mg
- 500μg
- 1mg
- 10mM(in 1mL DMSO)
- 5mg
- 10mg
- 25mg
- 50mg
- 100mg
- 200mg
- 250MG
- 500MG
- 1g
- 2.5G
- 5G
- 10G
- 25G
- 50G
- 100G
- 1KG
- Manufactureraablocks
- Product numberAA005QU9
- Product description1-Azakenpaullone 98%
- Packaging2mg
- Price$68
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA005QU9
- Product description1-Azakenpaullone 98%
- Packaging5mg
- Price$133
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA005QU9
- Product description1-Azakenpaullone 98%
- Packaging10mg
- Price$227
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA005QU9
- Product description1-Azakenpaullone 98
- Packaging50mg
- Price$572
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA005QU9
- Product description1-Azakenpaullone 98
- Packaging100mg
- Price$810
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA005QU9
- Product description1-Azakenpaullone 98
- Packaging25mg
- Price$411
- Updated2026-05-28
- Buy
- Manufactureraablocks
- Product numberAA005QU9
- Product description1-Azakenpaullone 98
- Packaging200mg
- Price$1084
- Updated2026-05-28
- Buy
- ManufacturerACHEMBLOCK
- Product numberY228766
- Product description1-Azakenpaullone 97.00%
- Packaging100MG
- Price$1360
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberY228766
- Product description1-Azakenpaullone 97.00%
- Packaging5MG
- Price$155
- Updated2026-05-27
- Buy
- ManufacturerACHEMBLOCK
- Product numberY228766
- Product description1-Azakenpaullone 97.00%
- Packaging25MG
- Price$525
- Updated2026-05-27
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CR1-0035-M005
- Product description1-Azakenpaullone ≥98%(HPLC,NMR)
- Packaging5mg
- Price$225
- Updated2026-05-06
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CR1-0035-M001
- Product description1-Azakenpaullone ≥98%(HPLC,NMR)
- Packaging1mg
- Price$75
- Updated2021-12-16
- Buy
- ManufacturerAdipogen Life Sciences
- Product numberAG-CR1-0035-M001
- Product description1-Azakenpaullone ≥98%(HPLC,NMR)
- Packaging1mg
- Price$75
- Updated2026-05-06
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0002418
- Product description1-Azakenpaullone 95.00%
- Packaging1MG
- Price$202.65
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0002418
- Product description1-Azakenpaullone 95.00%
- Packaging500MG
- Price$632.81
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberKIN0002418
- Product description1-Azakenpaullone 95.00%
- Packaging5MG
- Price$756.25
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| aablocks | AA005QU9 | 1-Azakenpaullone 98% | 2mg | $68 | 2026-05-28 | Buy |
| aablocks | AA005QU9 | 1-Azakenpaullone 98% | 5mg | $133 | 2026-05-28 | Buy |
| aablocks | AA005QU9 | 1-Azakenpaullone 98% | 10mg | $227 | 2026-05-28 | Buy |
| aablocks | AA005QU9 | 1-Azakenpaullone 98 | 50mg | $572 | 2026-05-28 | Buy |
| aablocks | AA005QU9 | 1-Azakenpaullone 98 | 100mg | $810 | 2026-05-28 | Buy |
| aablocks | AA005QU9 | 1-Azakenpaullone 98 | 25mg | $411 | 2026-05-28 | Buy |
| aablocks | AA005QU9 | 1-Azakenpaullone 98 | 200mg | $1084 | 2026-05-28 | Buy |
| ACHEMBLOCK | Y228766 | 1-Azakenpaullone 97.00% | 100MG | $1360 | 2026-05-27 | Buy |
| ACHEMBLOCK | Y228766 | 1-Azakenpaullone 97.00% | 5MG | $155 | 2026-05-27 | Buy |
| ACHEMBLOCK | Y228766 | 1-Azakenpaullone 97.00% | 25MG | $525 | 2026-05-27 | Buy |
| Adipogen Life Sciences | AG-CR1-0035-M005 | 1-Azakenpaullone ≥98%(HPLC,NMR) | 5mg | $225 | 2026-05-06 | Buy |
| Adipogen Life Sciences | AG-CR1-0035-M001 | 1-Azakenpaullone ≥98%(HPLC,NMR) | 1mg | $75 | 2021-12-16 | Buy |
| Adipogen Life Sciences | AG-CR1-0035-M001 | 1-Azakenpaullone ≥98%(HPLC,NMR) | 1mg | $75 | 2026-05-06 | Buy |
| American Custom Chemicals Corporation | KIN0002418 | 1-Azakenpaullone 95.00% | 1MG | $202.65 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0002418 | 1-Azakenpaullone 95.00% | 500MG | $632.81 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | KIN0002418 | 1-Azakenpaullone 95.00% | 5MG | $756.25 | 2021-12-16 | Buy |
Properties
Melting point :>290°C (dec.)
Boiling point :648.8±50.0 °C(Predicted)
Density :1.655±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: >10mg/mL
pka :13.36±0.20(Predicted)
form :Tan solid
color :gray-brown
InChI :InChI=1S/C15H10BrN3O/c16-8-3-4-11-9(6-8)10-7-13(20)18-12-2-1-5-17-15(12)14(10)19-11/h1-6,19H,7H2,(H,18,20)
InChIKey :NTSBZVCEIVPKBJ-UHFFFAOYSA-N
SMILES :N1C2=C(C=C(Br)C=C2)C2CC(=O)NC3=CC=CN=C3C1=2
Boiling point :648.8±50.0 °C(Predicted)
Density :1.655±0.06 g/cm3(Predicted)
storage temp. :2-8°C
solubility :DMSO: >10mg/mL
pka :13.36±0.20(Predicted)
form :Tan solid
color :gray-brown
InChI :InChI=1S/C15H10BrN3O/c16-8-3-4-11-9(6-8)10-7-13(20)18-12-2-1-5-17-15(12)14(10)19-11/h1-6,19H,7H2,(H,18,20)
InChIKey :NTSBZVCEIVPKBJ-UHFFFAOYSA-N
SMILES :N1C2=C(C=C(Br)C=C2)C2CC(=O)NC3=CC=CN=C3C1=2
Safety Information
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Description
1-Azakenpaullone is an analog of kenpaullone that inhibits glycogen synthase kinase 3β (GSK3β) more potently (IC50 = 18 nM) than CDK1/cyclin B or CDK5/p25 (IC50s = 2.0 and 4.2 μM, respectively). Through its effects on GSK3β, 1-azakenpaullone stimulates the proliferation of human pancreatic islets and drives the differentiation of mouse embryonic stem cells and Nematostella larvae.Related product price
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