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Agonist Inhibitors

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Structure Chemical Name CAS MF
7ACC-2 7ACC-2 1472624-85-3 C18H15NO4
RDEA-594 sodiuM RDEA-594 sodiuM 1151516-14-1 C17H13BrN3O2S.Na
LY-2584702 (hydrochloride) LY-2584702 (hydrochloride) 1082948-81-9 C21H20ClF4N7
ABBV-075 ABBV-075 1445993-26-9 C22H19F2N3O4S
CZC-54252 CZC-54252 1191911-27-9 C22H25ClN6O4S
PU-WS13 PU-WS13 1454619-14-7 C17H20Cl2N6S
2-(1-Phenyl-cyclopropylamino)-pyrimidine-5-carboxylic acid hydroxyamide 2-(1-Phenyl-cyclopropylamino)-pyrimidine-5-carboxylic acid hydroxyamide 1375465-91-0 C14H14N4O2
N-methyl-3-(1-(4-(piperazin-1-yl)phenyl)-5-(4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl)-1H-pyrazol-3-yl)propanamide N-methyl-3-(1-(4-(piperazin-1-yl)phenyl)-5-(4'-(trifluoromethyl)-[1,1'-biphenyl]-4-yl)-1H-pyrazol-3-yl)propanamide 1333146-24-9 C30H30F3N5O
MI-503 MI-503 1857417-13-0 C28H27F3N8S
ABT450 ABT450 1216941-48-8 C40H43N7O7S
Acalabrutinib Acalabrutinib 1420477-60-6 C26H23N7O2
MK-8931 MK-8931 1286770-55-5 C17H17F2N5O3S
SR-9243 SR-9243 1613028-81-1 C31H32BrNO4S2
GSK5959 GSK5959 901245-65-6 C22H26N4O3
AFN-1252 AFN-1252 620175-39-5 C22H21N3O3
CNV1014802 (hydrochloride) CNV1014802 (hydrochloride) 934240-31-0 C18H20ClFN2O2
IDO-IN-7 IDO-IN-7 1402837-78-8 C18H21FN2O2
Mutant IDH1-IN-2 Mutant IDH1-IN-2 1429176-69-1 C24H31F2N5O2
LY3023414 LY3023414 1386874-06-1 C23H26N4O3
2-Piperidinecarboxylic acid, 1-[[2,6-dimethoxy-4-[(2-methyl[1,1'-biphenyl]-3-yl)methoxy]phenyl]methyl]-, (2S)- 2-Piperidinecarboxylic acid, 1-[[2,6-dimethoxy-4-[(2-methyl[1,1'-biphenyl]-3-yl)methoxy]phenyl]methyl]-, (2S)- 1675201-83-8 C29H33NO5
Mirogabalin Mirogabalin 1138245-13-2 C12H19NO2
N-(3-{2-[3-Fluoro-4-(4-methyl-piperazin-1-yl)-phenylamino]-7H-pyrrolo[2,3-d]pyrimidin-4-yloxy}-phenyl)-acrylamide N-(3-{2-[3-Fluoro-4-(4-methyl-piperazin-1-yl)-phenylamino]-7H-pyrrolo[2,3-d]pyrimidin-4-yloxy}-phenyl)-acrylamide 1557267-42-1 C26H26FN7O2
SAR-20347 SAR-20347 1450881-55-6 C21H18ClFN4O4
XY1 XY1 1624117-53-8 C17H19N3O2
TRX-0237 mesylate TRX-0237 mesylate 1236208-20-0 C16H19N3S.2(CH4O3S)
genz-682452 genz-682452 1401090-53-6 C20H24FN3O2S
LBP-1 LBP-1 1050478-18-6 C23H29ClN6O3
FRAX1036 FRAX1036 1432908-05-8 C28H32ClN7O
Acelarin Acelarin 840506-29-8 C25H27F2N4O8P
BMS-582949 (hydrochloride) BMS-582949 (hydrochloride) 912806-16-7 C22H27ClN6O2
M2I-1 M2I-1 312271-03-7 C19H24N4O4S
Val-Cit-PAB-MMAE Val-Cit-PAB-MMAE 644981-35-1 C58H94N10O12
4-nitro-1-trityl-1H-imidazole 4-nitro-1-trityl-1H-imidazole 173865-33-3 C22H17N3O2
WNK463 WNK463 2012607-27-9 C21H24F3N7O2
PF-06281355 PF-06281355 1435467-38-1 C14H15N3O4S
DprE1-IN-2 DprE1-IN-2 1615713-87-5 C19H24N6O2
H3B-6527 H3B-6527 1702259-66-2 C29H34Cl2N8O4
KPT-8602 KPT-8602 1642300-52-4 C17H10F6N6O
Sulfatinib Sulfatinib 1816307-67-1 C24H28N6O3S
ML364 ML364 1991986-30-1 C24H18F3N3O3S2
BIA10-2474 BIA10-2474 1233855-46-3 C16H20N4O2
4-(4-fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide 4-(4-fluorophenyl)-N-(1H-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide 817194-38-0 C19H16FN5O2
JD-5037 JD-5037 1392116-14-1 C27H27Cl2N5O3S
E-7046 E-7046 1369489-71-3 C22H18F5N3O4
ML329 ML329 19992-50-8 C16H12N2O4S
RGX-104 HCl RGX-104 HCl 610318-03-1 C34H34Cl2F3NO3
1-(2-DIPHENYLMETHOXYETHYL)-4-(3-PHENYLPROPYL)PIPERAZINE DIHYDROCHLORIDE 1-(2-DIPHENYLMETHOXYETHYL)-4-(3-PHENYLPROPYL)PIPERAZINE DIHYDROCHLORIDE 67469-81-2 C28H35ClN2O
YC-1 YC-1 170632-47-0 C19H16N2O2
(3S,3AS,6AR)-3-ISOPROPYL-1-(METHANESULFONYL)-4-[4-(1-PIPERIDINYL)-2(E)-BUTENOYL]PERHYDROPYRROLO[3,2B]PYRROL-2(1H)-ONE HYDROCHLORIDE (3S,3AS,6AR)-3-ISOPROPYL-1-(METHANESULFONYL)-4-[4-(1-PIPERIDINYL)-2(E)-BUTENOYL]PERHYDROPYRROLO[3,2B]PYRROL-2(1H)-ONE HYDROCHLORIDE 198062-54-3 C19H31N3O4S
(S)-2,3-DIHYDRO-N-METHYL-N-2-PROPYNYL-1H-INDEN-1-AMINE (S)-2,3-DIHYDRO-N-METHYL-N-2-PROPYNYL-1H-INDEN-1-AMINE 185517-74-2 C12H13N
4'-CHLORO-3-METHOXYCINNAMANILIDE 4'-CHLORO-3-METHOXYCINNAMANILIDE 472981-92-3 C16H14ClNO2
DAGO DAGO 78123-71-4 C26H35N5O6
TRANS-3-BROMO-N-ETHYLCINNAMAMIDE TRANS-3-BROMO-N-ETHYLCINNAMAMIDE 58473-74-8 C11H12BrNO
DL-PENICILLAMINE DL-PENICILLAMINE 52-66-4 C5H11NO2S
24(R), 25-DIHYDROXYVITAMIN D3 24(R), 25-DIHYDROXYVITAMIN D3 40013-87-4 C27H44O3
BMS-345541 BMS-345541 547757-23-3 C14Cl1H18N5
Denatonium Benzoate Denatonium Benzoate 3734-33-6 C28H34N2O3
4-HYDROXYPHENYLRETINAMIDE 4-HYDROXYPHENYLRETINAMIDE 65646-68-6 C26H33NO2
4,6-Dichloro-1H-indole-2-carboxylic acid 4,6-Dichloro-1H-indole-2-carboxylic acid 101861-63-6 C9H5Cl2NO2
Escitalopram Escitalopram 128196-01-0 C20H21FN2O
ZM 449829 ZM 449829 4452-06-6 C13H10O
N-ACETYL-5-HYDROXYTRYPTAMINE N-ACETYL-5-HYDROXYTRYPTAMINE 1210-83-9 C12H14N2O2
KN-93 KN-93 139298-40-1 C26H29ClN2O4S
(R)-NAPROXEN (R)-NAPROXEN 23979-41-1 C14H14O3
Metamizole magnesium Metamizole magnesium 63372-86-1 C26H32MgN6O8S2
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