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Agonist Inhibitors

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Structure Chemical Name CAS MF
3-[N-(2-Hydroxyacetyl)-4-piperidyl]-4-(4-pyrimidinyl)-5-(4-chlorophenyl)pyrazole 3-[N-(2-Hydroxyacetyl)-4-piperidyl]-4-(4-pyrimidinyl)-5-(4-chlorophenyl)pyrazole 271576-80-8 C20H20ClN5O2
7-(Chlorodifluoromethyl)-5-(2-furanyl)-N-(2-thienylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide 7-(Chlorodifluoromethyl)-5-(2-furanyl)-N-(2-thienylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide 442666-98-0 C17H11ClF2N4O2S
CAY10650 CAY10650 1233706-88-1 C28H25NO6
Cl-Amidine Cl-Amidine 913723-61-2 C14H19ClN4O2
Genz-123346 Genz-123346 491833-30-8 C24H38N2O4
6-[(3-aMinophenyl)Methyl]-4,6-dihydro-4-Methyl-2-(Methylsulfinyl)-5H-Thieno[2',3':4,5]pyrrolo[2,3-d]pyridazin-5-one 6-[(3-aMinophenyl)Methyl]-4,6-dihydro-4-Methyl-2-(Methylsulfinyl)-5H-Thieno[2',3':4,5]pyrrolo[2,3-d]pyridazin-5-one 1221186-53-3 C17H16N4O2S2
N-Ethyl-7,10-dihydro-8-nitro-7-oxo-N-propyl-1,10-phenanthroline-3-carboxamide N-Ethyl-7,10-dihydro-8-nitro-7-oxo-N-propyl-1,10-phenanthroline-3-carboxamide 223666-07-7 C18H18N4O4
9-(6-Amino-3-pyridinyl)-1-[4-fluoro-3-(trifluoromethyl)phenyl]benzo[h]-1,6-naphthyridin-2(1H)-one 9-(6-Amino-3-pyridinyl)-1-[4-fluoro-3-(trifluoromethyl)phenyl]benzo[h]-1,6-naphthyridin-2(1H)-one 1223002-54-7 C24H14F4N4O
GNE 477 GNE 477 1032754-81-6 C21H28N8O3S2
JNJ-28312141 JNJ-28312141 885692-52-4 C26H32N6O2
CTS-1027 CTS-1027 193022-04-7 C19H20ClNO6S
CYT387 2H2SO4 salt CYT387 2H2SO4 salt 1056636-06-6 C23H26N6O10S2
sodiuM 4-pentynoate sodiuM 4-pentynoate 101917-30-0 C5H5O2.Na
CHF 5074 CHF 5074 749269-83-8 C16H11Cl2FO2
Rigosertib sodium Rigosertib sodium 592542-60-4 C21H24NNaO8S
SB-681323 SB-681323 444606-18-2 C23H19F3N4O3
INCB8761(PF-4136309) INCB8761(PF-4136309) 1341224-83-6 C29H31F3N6O3
LCQ-908 LCQ-908 956136-95-1 C25H24F3N3O2
MB-05032 MB-05032 261365-11-1 C11H15N2O4PS
MK-6892 MK-6892 917910-45-3 C19H22N4O5
NKP-1339 NKP-1339 197723-00-5 C14H12Cl4N4NaRu
RO 9187 RO 9187 876708-03-1 C9H12N6O5
SB-649868 SB-649868 380899-24-1 C26H24FN3O3S
TAK-960 TAK-960 1137868-52-0 C27H34F3N7O3
ST101 ST101 887603-94-3 C15H12N2O
ML 161 ML 161 423735-93-7 C17H17BrN2O2
N-(1-phenylethyl)-2-(pyrrolidin-1-yl)quinazolin-4-aMine N-(1-phenylethyl)-2-(pyrrolidin-1-yl)quinazolin-4-aMine 662163-81-7 C20H22N4
CHIR-090 CHIR-090 728865-23-4 C24H27N3O5
NSC 42834 NSC 42834 195371-52-9 C23H24N2O
L778123 L778123 253863-00-2 C22H21Cl2N5O
GDC-0032 GDC-0032 1282512-48-4 C24H28N8O2
360 A 360 A 794458-56-3 C27H23N5O2+2
Exjade Fe3+ chelate Exjade Fe3+ chelate 554435-83-5 C21H12FeN3O4
ZP 1609 Hydrochloride ZP 1609 Hydrochloride 943133-81-1 C14H18ClN3O4
IDO inhibitor 1 IDO inhibitor 1 1204669-37-3 C11H13BrFN7O4S
Kalydeco benzenesulfonate Kalydeco benzenesulfonate 1134822-09-5 C30H34N2O6S
R-1530 R-1530 882531-87-5 C18H14ClFN4O
RGFP-966 RGFP-966 1357389-11-7 C21H19FN4O
ZD 6474 trifluoroacetate ZD 6474 trifluoroacetate 338992-53-3 C24H25BrF4N4O4
XMD17 109 XMD17 109 1435488-37-1 C36H46N8O3
FG 2216 FG 2216 223387-75-5 C12H9ClN2O4
SKLB 610 SKLB 610 1125780-41-7 C21H16F3N3O3
APD668 APD668 832714-46-2 C21H24FN5O5S
BRD-9539 BRD-9539 1374601-41-8 C24H21N3O3
2-ThiophenecarboxaMide, 4-cyano-5-[(3,5-dichloro-4-pyridinyl)thio]-N-[4-(Methylsulfonyl)phenyl]- 2-ThiophenecarboxaMide, 4-cyano-5-[(3,5-dichloro-4-pyridinyl)thio]-N-[4-(Methylsulfonyl)phenyl]- 1247825-37-1 C18H11Cl2N3O3S3
MonoMethylauristatin F MonoMethylauristatin F 745017-94-1 C39H65N5O8
TAS-103 dihydrochloride TAS-103 dihydrochloride 174634-09-4 C20H21Cl2N3O2
Necrosulfonamide Necrosulfonamide 1360614-48-7 C18H15N5O6S2
2-(2-Chlorophenyl)-4-(3-(diMethylaMino)phenyl)-5-Methyl-1H-pyrazolo[4,3-c]pyridine-3,6(2H,5H)-dione 2-(2-Chlorophenyl)-4-(3-(diMethylaMino)phenyl)-5-Methyl-1H-pyrazolo[4,3-c]pyridine-3,6(2H,5H)-dione 1218942-37-0 C21H19ClN4O2
AVE 0991 (sodiuM salt) AVE 0991 (sodiuM salt) 306288-04-0 C29H33N4NaO5S2
Inauhzin Inauhzin 309271-94-1 C25H19N5OS2
ABT-333 ABT-333 1132935-63-7 C26H27N3O5S
Y320 Y320 288250-47-5 C27H29ClN6O2
CEP-37440 CEP-37440 1391712-60-9 C30H38ClN7O3
3-[(3-Methoxybenzoyl)aMino]-4-(4-Methyl-1-piperazinyl)benzoic Acid Methyl Ester 3-[(3-Methoxybenzoyl)aMino]-4-(4-Methyl-1-piperazinyl)benzoic Acid Methyl Ester 890190-22-4 C21H25N3O4
Dapagliflozin propanediol monohydrate Dapagliflozin propanediol monohydrate 960404-48-2 C24H33ClO8
Saroglitazar Saroglitazar 495399-09-2 C25H29NO4S
N-DesMethyl Netupitant N-DesMethyl Netupitant 290296-72-9 C29H30F6N4O
GSK2194069 GSK2194069 1332331-08-4 C25H24N4O3
ML355 ML355 1532593-30-8 C21H19N3O4S2
SAR245409 SAR245409 934493-76-2 C13H14N6O
6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- 202592-23-2 C19H17ClN4O2S
Elbasvir Elbasvir 1370468-36-2 C49H55N9O7
GDC-0994 GDC-0994 1453848-26-4 C21H18ClFN6O2
Umbralisib Umbralisib 1532533-67-7 C31H24F3N5O3
CVT-10216 CVT-10216 1005334-57-5 C24H19NO7S
URMC-099 URMC-099 1229582-33-5 C27H27N5
LSN2814617 LSN2814617 1313498-08-6 C18H20FN5O
K-Ras G12C-IN-3 K-Ras G12C-IN-3 1629268-19-4 C21H19Cl3N2O3
TRV-130 TRV-130 1401031-39-7 C22H31ClN2O2S
DM1-SMCC DM1-SMCC 1228105-51-8 C51H66ClN5O16S
BAL27862 BAL27862 798577-91-0 C20H17N7O2
EX-527 (R-enantioMer) EX-527 (R-enantioMer) 848193-69-1 C13H13ClN2O
TAK-063 TAK-063 1238697-26-1 C23H17FN6O2
AI-10-49 AI-10-49 1256094-72-0 C30H22F6N6O5
ethyl 4-(((2R,3R,4S,5R,6S)-4,5-bis(benzo[d][1,3]dioxol-5-ylcarbamoyloxy)-2-(hydroxymethyl)-6-methoxy-tetrahydro-2H-pyran-3-yloxy)carbonyl)benzoate ethyl 4-(((2R,3R,4S,5R,6S)-4,5-bis(benzo[d][1,3]dioxol-5-ylcarbamoyloxy)-2-(hydroxymethyl)-6-methoxy-tetrahydro-2H-pyran-3-yloxy)carbonyl)benzoate 1137359-47-7 C33H33N3O15
TP0903 TP0903 1341200-45-0 C24H30ClN7O2S
3-([1,4′-Bipiperidin]-1′-ylmethyl)-7-bromo-N-(1-phenylcyclopropyl)-2-[3-(trifluoromethyl)phenyl]-4-quinolinecarboxamide 3-([1,4′-Bipiperidin]-1′-ylmethyl)-7-bromo-N-(1-phenylcyclopropyl)-2-[3-(trifluoromethyl)phenyl]-4-quinolinecarboxamide 1336960-13-4 C37H38BrF3N4O
H-ASP-PHE-OH H-ASP-PHE-OH 13433-09-5 C13H16N2O5
Lumateperone Lumateperone 313368-91-1 C24H28FN3O
2-butylsulfinyl-4-phenyl-6-thiophen-2-ylthieno[5,4-b]pyridin-3-amine 2-butylsulfinyl-4-phenyl-6-thiophen-2-ylthieno[5,4-b]pyridin-3-amine 459147-39-8 C21H20N2OS3
cyclopentyl 2-cyclohexyl-2-((6-(3-(hydroxyamino)-3-oxopropyl)pyridin-3-yl)methylamino)acetate cyclopentyl 2-cyclohexyl-2-((6-(3-(hydroxyamino)-3-oxopropyl)pyridin-3-yl)methylamino)acetate 1018673-42-1 C22H33N3O4
sbc-115076 sbc-115076 489415-96-5 C31H33N3O5
4-(2-(3-amino-1H-pyrazol-4-yl)-4-chlorophenoxy)-5-chloro-2-fluoro-N-(thiazol-4-yl)benzenesulfonamide
Molecular Weight: 500.35 4-(2-(3-amino-1H-pyrazol-4-yl)-4-chlorophenoxy)-5-chloro-2-fluoro-N-(thiazol-4-yl)benzenesulfonamide Molecular Weight: 500.35 1235403-62-9 C18H12Cl2FN5O3S2
Endoxifen HCl Endoxifen HCl 1032008-74-4 C25H28ClNO2
Centrinone Centrinone 1798871-30-3 C26H25F2N7O6S2
K-Ras-IN-1 K-Ras-IN-1 84783-01-7 C11H13NOS
Verinurad Verinurad 1352792-74-5 C20H16N2O2S
1-(4-(5-(5-amino-6-(5-(tert-butyl)-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one 1-(4-(5-(5-amino-6-(5-(tert-butyl)-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one 1620576-64-8 C22H31N9O3
CPI-268456 CPI-268456 1380087-86-4 C20H15Cl2N3O2
AZ-33 AZ-33 1370290-34-8 C25H27N3O6S
AMG-337 AMG-337 1173699-31-4 C23H22FN7O3
JAK3-IN-1 JAK3-IN-1 1805787-93-2 C26H30ClN7O2
4-[4-(1-methyl-1H-pyrazol-4-yl)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl]-benzonitrile 4-[4-(1-methyl-1H-pyrazol-4-yl)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl]-benzonitrile 1665195-94-7 C20H19N7
TD-4208 TD-4208 864750-70-9 C35H43N5O4
CP-456773 sodium CP-456773 sodium 256373-96-3 C20H23N2NaO5S
MS023 MS023 1831110-54-3 C17H25N3O
XMU-MP-1 XMU-MP-1 2061980-01-4 C17H16N6O3S2
AKT inhibitor 2 AKT inhibitor 2 1313881-70-7 C27H24N6
MK-4101 MK-4101 935273-79-3 C24H24F5N5O
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