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Agonist Inhibitors

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Structure Chemical Name CAS MF
ALK inhibitor 1 ALK inhibitor 1 761436-81-1 C23H28BrN7O3S
CDK9 inhibitor CDK9 inhibitor 1415559-43-1 C26H21N5O4S
SMND-309 SMND-309 1065559-56-9 C18H14O8
Phenol, 2-Methoxy-5-[[[(1E)-2-(2,4,6-triMethoxyphenyl)ethenyl]sulfonyl]Methyl]-, 1-(dihydrogen phosphate) Phenol, 2-Methoxy-5-[[[(1E)-2-(2,4,6-triMethoxyphenyl)ethenyl]sulfonyl]Methyl]-, 1-(dihydrogen phosphate) 865783-99-9 C19H23O10PS
AMG 487 AMG 487 473719-41-4 C32H28F3N5O4
BMS 303141 BMS 303141 943962-47-8 C19H15Cl2NO4S
CNS 7056 CNS 7056 308242-62-8 C21H19BrN4O2
EBE-A 22 EBE-A 22 229476-53-3 C17H16BrN3O2
EL-102 EL-102 1233948-61-2 C19H16N2O3S2
Topiroxostat Topiroxostat 577778-58-6 C13H8N6
JDTic JDTic 361444-66-8 C28H39N3O3
JNJ 31020028 JNJ 31020028 1094873-14-9 C34H36FN5O2
LCI699 LCI699 928134-65-0 C13H10FN3
MAY-262611 MAY-262611 1123231-07-1 C20H22N4
MK 0557 MK 0557 328232-95-7 C22H19FN4O3
PNU 100480 PNU 100480 168828-58-8 C16H20FN3O3S
RI-1 RI-1 415713-60-9 C14H11Cl3N2O3
Vorapaxar Vorapaxar 618385-01-6 C29H33FN2O4
TMEM16AInhibitorsRevealTMEM16A(T16Ainh-A01) TMEM16AInhibitorsRevealTMEM16A(T16Ainh-A01) 552309-42-9 C19H20N4O3S2
N-(2-(2-(4-chlorophenyl)thiazol-4-yl)ethyl)butyraMide N-(2-(2-(4-chlorophenyl)thiazol-4-yl)ethyl)butyraMide 932986-18-0 C15H17ClN2OS
SAR131675 SAR131675 1092539-44-0 C18H22N4O4
S0859 S0859 1019331-10-2 C29H24ClN3O3S
1,2,3-Benzenetriol, 4-[[[2-(cyclohexyliMino)-4- 1,2,3-Benzenetriol, 4-[[[2-(cyclohexyliMino)-4- 509102-00-5 C17H21N3O3S
UNBS-5162 UNBS-5162 956590-23-1 C17H18N4O3
PD0166285 PD0166285 185039-89-8 C26H27Cl2N5O2
Enocitabine Enocitabine 55726-47-1 C31H55N3O6
360 A iodide 360 A iodide 737763-37-0 C27H23IN5O2+
Fostemsavir Fostemsavir 864953-29-7 C25H26N7O8P
DB-07268 DB-07268 929007-72-7 C17H15N5O2
PST2744 (hydrochloride) PST2744 (hydrochloride) 374559-48-5 C21H33ClN2O3
ZD 6474 hydrochloride ZD 6474 hydrochloride 524722-52-9 C22H25BrClFN4O2
MK 6096 MK 6096 1088991-73-4 C24H25FN4O2
CNX-419 hydrobroMide CNX-419 hydrobroMide 1446700-26-0 C27H29BrF3N7O3
Auristatin E Auristatin E 160800-57-7 C40H69N5O7
TMC-647055 TMC-647055 1204416-97-6 C32H38N4O6S
S1RA S1RA 878141-96-9 C20H23N3O2
Debio 0932 ,CUDC-305 Debio 0932 ,CUDC-305 1061318-81-7 C22H30N6O2S
BPR1J-097 BPR1J-097 1327167-19-0 C27H28N6O3S
Radotinib Radotinib 926037-48-1 C27H21F3N8O
Kobe-0065 Kobe-0065 436133-68-5 C15H11ClF3N5O4S
Methyl [4,6-diaMino-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]pyriMidin-5-yl]carbaMate Methyl [4,6-diaMino-2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]pyriMidin-5-yl]carbaMate 625115-52-8 C19H17FN8O2
N-(4-chloropyridin-3-yl)-4-((2,2-difluorobenzo[d][1,3]dioxol-5-yl)Methyl)piperazine-1-carboxaMide N-(4-chloropyridin-3-yl)-4-((2,2-difluorobenzo[d][1,3]dioxol-5-yl)Methyl)piperazine-1-carboxaMide 1346528-50-4 C18H17ClF2N4O3
NSI-189 NSI-189 1270138-40-3 C22H30N4O
GNF179 Metabolite GNF179 Metabolite 1310455-86-7 C14H16FN3
HG-9-91-01 HG-9-91-01 1456858-58-4 C32H37N7O3
HBX 19818 HBX 19818 1426944-49-1 C25H28ClN3O
SiraMesine, Lu-28-179 SiraMesine, Lu-28-179 224177-60-0 C30H32ClFN2O
AMG 925 AMG 925 1401033-86-0 C26H29N7O2
Btk inhibitor 1 (R enantioMer hydrochloride) Btk inhibitor 1 (R enantioMer hydrochloride) 1553977-42-6 C22H23ClN6O
(S)-3-(4-((4'-(Trifluoromethyl)-[1,1'-biphenyl]-3-yl)methoxy)phenyl)hex-4-ynoic acid (S)-3-(4-((4'-(Trifluoromethyl)-[1,1'-biphenyl]-3-yl)methoxy)phenyl)hex-4-ynoic acid 865231-46-5 C26H21F3O3
N2-(7-Chloro-4-quinolinyl)-N1-[2-[(7-chloro-4-quinolinyl)aMino]ethyl]-N1-Methyl-1,2-ethanediaMine N2-(7-Chloro-4-quinolinyl)-N1-[2-[(7-chloro-4-quinolinyl)aMino]ethyl]-N1-Methyl-1,2-ethanediaMine 1391426-22-4 C23H23Cl2N5
2{[(5Z)2(1,2diazinan1yl)4oxo4,5dihydro1,3thiazol5ylidene]Methyl}5fluorophenyl pyrrolidine1carboxylate 2{[(5Z)2(1,2diazinan1yl)4oxo4,5dihydro1,3thiazol5ylidene]Methyl}5fluorophenyl pyrrolidine1carboxylate 1181083-81-7 C19H21FN4O3S
G007-LK G007-LK 1380672-07-0 C25H16ClN7O3S
Dispiro[cyclohexane-1,2'-[2H]indene-1'(3'H),2''-[2H]iMidazol]-4''-aMine, 4-Methoxy-5''-Methyl-6'-[5-(1-propyn-1-yl)-3-pyridinyl]-, (1α,1'R,4β)- Dispiro[cyclohexane-1,2'-[2H]indene-1'(3'H),2''-[2H]iMidazol]-4''-aMine, 4-Methoxy-5''-Methyl-6'-[5-(1-propyn-1-yl)-3-pyridinyl]-, (1α,1'R,4β)- 1383982-64-6 C26H28N4O
[4-(2,4-Dimethoxy-phenyl)-5-oxo-4,5-dihydro-[1,2]dithiolo[4,3]pyrro-6-yl]-carbamic acid ethyl ester [4-(2,4-Dimethoxy-phenyl)-5-oxo-4,5-dihydro-[1,2]dithiolo[4,3]pyrro-6-yl]-carbamic acid ethyl ester 1015064-87-5 C16H16N2O5S2
PF-04979064 PF-04979064 1220699-06-8 C24H26N6O3
BAMB-4 BAMB-4 891025-25-5 C15H12N2O2
GSK2110183 GSK2110183 1047634-63-8 C18H16Cl2F2N4OS
ML277 ML277 1401242-74-7 C23H25N3O4S2
1-(2,4-Dichlorophenyl)-N-1-piperidinyl-4-[[(1-pyrrolidinylsulfonyl)amino]methyl]-5-[5-[2-[4-(trifluoromethyl)phenyl]ethynyl]-2-thienyl]-1H-pyrazole-3-carboxamide 1-(2,4-Dichlorophenyl)-N-1-piperidinyl-4-[[(1-pyrrolidinylsulfonyl)amino]methyl]-5-[5-[2-[4-(trifluoromethyl)phenyl]ethynyl]-2-thienyl]-1H-pyrazole-3-carboxamide 1429239-98-4 C33H31Cl2F3N6O3S2
Peficitinib Peficitinib 944118-01-8 C18H22N4O2
FMoc-Val-Cit-PAB-MMAE FMoc-Val-Cit-PAB-MMAE 1350456-56-2 C73H104N10O14
K-7174 K-7174 191089-59-5 C33H48N2O6
Voruciclib Voruciclib 1000023-04-0 C22H19ClF3NO5
AZD8186 AZD8186 1627494-13-6 C24H25F2N3O4
VRT-1353385 VRT-1353385 1616113-45-1 C35H39NO11
AMG319 AMG319 1608125-21-8 C21H16FN7
IQ-1 sodium IQ-1 sodium 23146-22-7 C15H9N3O
NSC 600157 NSC 600157 31083-55-3 C15H9NO2
BD 1047 dihydrobromide BD 1047 dihydrobromide 138356-21-5 C13H22Br2Cl2N2
2-(4-(2-amino-2-oxoethoxy)-1-benzyl-2-ethyl-1H-indol-3-yl)-2-oxoacetamide 2-(4-(2-amino-2-oxoethoxy)-1-benzyl-2-ethyl-1H-indol-3-yl)-2-oxoacetamide 185298-58-2 C21H21N3O4
EGF816 EGF816 1508250-71-2 C26H31ClN6O2
mavatrep mavatrep 956274-94-5 C25H21F3N2O
BHPI BHPI 56632-39-4 C21H17NO3
Onatasertib (CC-223) Onatasertib (CC-223) 1228013-30-6 C21H27N5O3
Mps1-IN-5 Mps1-IN-5 1443763-60-7 C29H26FN5O4S
TG6-10-1 TG6-10-1 1415716-58-3 C23H23F3N2O4
SPDB SPDB 115088-06-7 C13H14N2O4S2
DEL-22379 DEL-22379 181223-80-3 C26H28N4O3
BDA-366 BDA-366 1821496-27-8 C25H29N3O4
SCR-1481B1 SCR-1481B1 1174161-86-4 C28H29ClF2N5O10P
Aldose reductase-IN-1 Aldose reductase-IN-1 1355612-71-3 C17H10F3N5O3S
ORM-15341 ORM-15341 1297537-33-7 C19H17ClN6O2
HM-61713 (BI-1482694) HM-61713 (BI-1482694) 1802181-20-9
LJI308 LJI308 1627709-94-7 C21H18F2N2O2
CCT251545 CCT251545 1661839-45-7 C23H24ClN5O
ML-098 ML-098 878978-76-8 C19H19NO3
GNF-6231 GNF-6231 1243245-18-2 C24H25FN6O2
GSK591 GSK591 1616391-87-7 C22H28N4O2
Madrasin Madrasin 374913-63-0 C16H17N5O2
GDC-0853 GDC-0853 1434048-34-6 C37H44N8O4
CPI-1205 CPI-1205 1621862-70-1 C27H33F3N4O3
KRIBB11 KRIBB11 342639-96-7 C13H12N6O2
GNE-140 (racemate) GNE-140 (racemate) 1802977-61-2 C25H23ClN2O3S2
GPR120 Compound A GPR120 Compound A 1599477-75-4 C19H23ClF3NO3
BAR 501 BAR 501 1632118-69-4 C26H46O3
CLR1501 CLR1501 1250963-36-0 C38H59BF2N3O3P
T5601640 T5601640 924473-59-6 C19H14F3N3O3
KR-33494 KR-33494 1021497-97-1 C20H18BrN3O3S
CFI-402257 CFI-402257 1610759-22-2 C28H30N6O3
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