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Agonist Inhibitors

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Structure Chemical Name CAS MF
EVP 6124 EVP 6124 550999-75-2 C16H17ClN2OS
Sarecycline Hydrochloride Sarecycline Hydrochloride 1035979-44-2 C24H30ClN3O8
KML-29 KML-29 1380424-42-9 C24H21F6NO7
4H-1,2,4-Triazole-4-carboxaMide, 1-(2,4-dichlorophenyl) -N-(2,4-difluorophenyl)-1,5-dihydro-N-(1-Methylethyl)- 5-oxo- 4H-1,2,4-Triazole-4-carboxaMide, 1-(2,4-dichlorophenyl) -N-(2,4-difluorophenyl)-1,5-dihydro-N-(1-Methylethyl)- 5-oxo- 212201-70-2 C18H14Cl2F2N4O2
Relugolix Relugolix 737789-87-6 C29H27F2N7O5S
VTX-2337 VTX-2337 926927-61-9 C28H34N4O2
TUG-770 TUG-770 1402601-82-4 C19H14FNO2
AMD 070 hydrochloride AMD 070 hydrochloride 880549-30-4 C21H28ClN5
Azaphenonxazine dihydrochloride Monohydrate Azaphenonxazine dihydrochloride Monohydrate 63302-99-8 C16H23Cl2N5O2
CCT 241533 hydrochloride CCT 241533 hydrochloride 1431697-96-9 C23H28ClFN4O4
CX 6258 hydrochloride hydrate CX 6258 hydrochloride hydrate 1353858-99-7 C26H27Cl2N3O4
LDE-225 Diphosphate LDE-225 Diphosphate 1218778-77-8 C26H32F3N3O11P2
LY-2795050 LY-2795050 1346133-08-1 C23H22ClN3O2
SodiuM Channel inhibitor 1 SodiuM Channel inhibitor 1 1198117-23-5 C24H19F4N3O3
Tipiracil hydrochloride Tipiracil hydrochloride 183204-72-0 C9H12Cl2N4O2
CEP-28122 CEP-28122 1022958-60-6 C28H35ClN6O3
HMN 176 HMN 176 173529-10-7 C20H18N2O4S
HM 30181A HM 30181A 849675-66-7 C38H36N6O7
CTEP Derivative CTEP Derivative 802906-73-6 C18H13ClFN3
1H-Isoindole-1,3(2H)-dione, 5-[5-[[3-(4-broMophenyl)-2-iMino-4-oxo-5-thiazolidinylidene]Methyl]-2-furanyl]- 1H-Isoindole-1,3(2H)-dione, 5-[5-[[3-(4-broMophenyl)-2-iMino-4-oxo-5-thiazolidinylidene]Methyl]-2-furanyl]- 1420071-30-2 C22H12BrN3O4S
PF-04995274 PF-04995274 1331782-27-4 C23H32N2O6
AC710 AC710 1351522-04-7 C31H42N6O4
AgoMelatine (hydrochloride) AgoMelatine (hydrochloride) 1176316-99-6 C15H18ClNO2
Ledipasvir (acetone) Ledipasvir (acetone) 1441674-54-9 C52H60F2N8O7
SP-420 SP-420 911714-45-9 C16H21NO6S
Mps1-IN-2 Mps1-IN-2 1228817-38-6 C26H36N6O3
QL47 QL47 1469988-75-7 C27H21N5O2
PF-01247324 PF-01247324 875051-72-2 C13H10Cl3N3O
AP-III-a4 AP-III-a4 1177827-73-4 C31H43FN8O3
PSI-7976 PSI-7976 1190308-01-0 C22H29FN3O9P
GSK2141795 GSK2141795 1047634-65-0 C18H16Cl2F2N4O2
NVP-TNKS656 NVP-TNKS656 1419949-20-4 C27H34N4O5
N1-(2,2,6,6-tetraMethylpiperidin-4-yl)-N2-p-tolyloxalaMide N1-(2,2,6,6-tetraMethylpiperidin-4-yl)-N2-p-tolyloxalaMide 144217-65-2 C18H27N3O2
Optovin Optovin 348575-88-2 C15H13N3OS2
Resmetirom Resmetirom 920509-32-6 C17H12Cl2N6O4
Dafadine-A Dafadine-A 1065506-69-5 C23H25N3O3
GK921 GK921 1025015-40-0 C21H20N4O
LDN-27219 LDN-27219 312946-37-5 C20H16N4O2S2
Skp2 Inhibitor C1 Skp2 Inhibitor C1 432001-69-9 C18H13BrN2O4S2
Decernotinib Decernotinib 944842-54-0 C18H19F3N6O
JIB-04 (NSC 693627) -Z JIB-04 (NSC 693627) -Z 199596-24-2 C17H13ClN4
Eluxadoline Dihydrochloride Eluxadoline Dihydrochloride 864825-13-8 C32H39Cl2N5O5
ERDAFITINIB ERDAFITINIB 1346242-81-6 C25H30N6O2
N,N'-(2,2'-(1,4-phenylene)bis(ethane-2,1-diyl))dipropane-2-sulfonaMide N,N'-(2,2'-(1,4-phenylene)bis(ethane-2,1-diyl))dipropane-2-sulfonaMide 380607-77-2 C16H28N2O4S2
(S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride (S)-2-phenyl-1-(thiazol-2-yl)ethanaMine hydrochloride 135383-60-7 C11H13ClN2S
CPI 360 CPI 360 1802175-06-9 C25H31N3O4
IKK epsilon-IN-1 IKK epsilon-IN-1 1292310-49-6 C26H27N5O3
GV-58 GV-58 1402821-41-3 C18H26N6OS
Z-360 Z-360 209219-38-5 C29H36N4O5
CX-4945 (sodiuM salt) CX-4945 (sodiuM salt) 1309357-15-0 C19H13ClN3NaO2
Exherin (trifluoroacetate) Exherin (trifluoroacetate) 1135237-88-5 C24H35F3N8O8S2
Pyridoclax Pyridoclax 1651890-44-6 C29H22N4
GSK2879552 GSK2879552 1401966-69-5 C23H28N2O2
CAS:932749-62-7 CAS:932749-62-7 932749-62-7 C20H16Br2O3
(S)-1-((5-chloropyridin-3-yl)methyl)-8-((R)-3-methylmorpholino)-2-(trifluoromethyl)-3,4-dihydro-1H-pyrimido[1,2-a]pyrimidin-6(2H)-one (S)-1-((5-chloropyridin-3-yl)methyl)-8-((R)-3-methylmorpholino)-2-(trifluoromethyl)-3,4-dihydro-1H-pyrimido[1,2-a]pyrimidin-6(2H)-one 1523406-39-4 C19H21ClF3N5O2
ML-228 ML-228 1357171-62-0 C27H21N5
4-((3,5-Dichloro-2-hydroxybenzyl)amino)-2-hydroxybenzoic acid 4-((3,5-Dichloro-2-hydroxybenzyl)amino)-2-hydroxybenzoic acid 1181226-02-7 C14H11Cl2NO4
Wnt Agonist Wnt Agonist 853220-52-7 C19H18N4O3
N-(2-Aminophenyl)pyrazine-2-carboxamide N-(2-Aminophenyl)pyrazine-2-carboxamide 926259-99-6 C11H10N4O
Theophylline-7-acetic acid Theophylline-7-acetic acid 652-37-9 C9H10N4O4
PFK-158 PFK-158 1462249-75-7 C18H11F3N2O
CYM 50260 CYM 50260 1355026-60-6 C14H11Cl3FNO2
N-(4-ethylphenyl)-3-(hydroxymethyl)-N-isobutyl-4-((tetrahydro-2H-pyran-4-yl)methoxy)benzenesulfonamide N-(4-ethylphenyl)-3-(hydroxymethyl)-N-isobutyl-4-((tetrahydro-2H-pyran-4-yl)methoxy)benzenesulfonamide 1474110-21-8 C25H35NO5S
Epacadostat (INCB024360) Epacadostat (INCB024360) 1204669-58-8 C11H13BrFN7O4S
5'-Methoxy-6'-[3-(1-pyrrolidinyl)propoxy]spiro[cyclobutane-1,3'-[3H]indol]-2'-amine 5'-Methoxy-6'-[3-(1-pyrrolidinyl)propoxy]spiro[cyclobutane-1,3'-[3H]indol]-2'-amine 1527503-11-2 C19H27N3O2
ML346 ML346 100872-83-1 C14H12N2O4
IN00076730 IN00076730 1454700-89-0 C17H21BrO2
JH-II-127 JH-II-127 1700693-08-8 C19H21ClN6O3
A-196 A-196 1982372-88-2 C18H16Cl2N4
ODM-201 ODM-201 1297538-32-9 C19H19ClN6O2
GSK-2881078 GSK-2881078 1539314-06-1 C14H13F3N2O2S
Acamprosate calcium Acamprosate calcium 77337-73-6 C10H20CaN2O8S2
JNJ 63533054 JNJ 63533054 1802326-66-4 C17H17ClN2O2
mk-1064 mk-1064 1207253-08-4 C24H20ClN5O3
EPZ031686 EPZ031686 1808011-22-4 C26H34ClF3N4O4S
RSL3 RSL3 1219810-16-8 C23H21ClN2O5
MS049 MS049 1502816-23-0 C15H24N2O
PIK-III PIK-III 1383716-40-2 C17H17N7
ALS-8176 ALS-8176 1445385-02-3 C18H25ClFN3O6
SBI-0640756 SBI-0640756 1821280-29-8 C23H14ClFN2O2
SirReal2 SirReal2 709002-46-0 C22H20N4OS2
9-Propenyladenine 9-Propenyladenine 1446486-33-4 C8H9N5
SRT3025 SRT3025 1231952-55-8 C31H31N5O2S2
BI-9564 BI-9564 1883429-22-8 C20H23N3O3
CFMTI CFMTI 864864-17-5 C19H16FN5O
N-(4-((1R,3S,5S)-3-amino-5-methylcyclohexyl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide N-(4-((1R,3S,5S)-3-amino-5-methylcyclohexyl)pyridin-3-yl)-6-(2,6-difluorophenyl)-5-fluoropicolinamide 1210608-43-7 C24H23F3N4O
APS-2-79 hydrochloride APS-2-79 hydrochloride 2002381-31-7 C23H22ClN3O3
ml390 ml390 2029049-79-2 C21H21F3N2O3
Amiselimod(MT-1303) free base Amiselimod(MT-1303) free base 942399-20-4 C19H30F3NO3
NMS-P118 NMS-P118 1262417-51-5 C20H24F3N3O2
HDAC-IN-4 HDAC-IN-4 934828-12-3 C24H29N5O
MX-69 MX-69 1005264-47-0 C27H26N2O4S
ASK1-IN-1 ASK1-IN-1 1262041-49-5 C23H21N7O
BAY41-4109  Racemic BAY41-4109 Racemic 298708-79-9 C18H13ClF3N3O2
MELK-8a MELK-8a 1922153-17-0 C25H32N6O
1-(3,6-DIBROMO-9H-CARBAZOL-9-YL)-3-(DIMETHYLAMINO)PROPAN-2-OL 1-(3,6-DIBROMO-9H-CARBAZOL-9-YL)-3-(DIMETHYLAMINO)PROPAN-2-OL 253449-04-6 C17H18Br2N2O
RO 31-8220 METHANESULFONATE RO 31-8220 METHANESULFONATE 125314-64-9 C25H23N5O2S
Deoxythymidine triphosphate Deoxythymidine triphosphate 18423-43-3 C10H18N2NaO14P3
Testolactone Testolactone 968-93-4 C19H24O3
O-304 O-304 1261289-04-6 C16H11Cl2N3O2S
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