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Agonist Inhibitors

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Structure Chemical Name CAS MF
Calcitetrol Calcitetrol 72203-93-1 C27H44O4
Regorafenib (Hydrochloride) Regorafenib (Hydrochloride) 835621-07-3 C21H16Cl2F4N4O3
VTP-27999 (Hydrochloride) VTP-27999 (Hydrochloride) 1264191-73-2 C26H42Cl2N4O5
Phenol, 4-chloro-3-[5-Methyl-3-[[4-[2-(1-pyrrolidinyl)ethoxy]phenyl]aMino]-1,2,4-benzotriazin-7-yl]- Phenol, 4-chloro-3-[5-Methyl-3-[[4-[2-(1-pyrrolidinyl)ethoxy]phenyl]aMino]-1,2,4-benzotriazin-7-yl]- 867334-05-2 C26H26ClN5O2
1alpha-Hydroxy VD4 1alpha-Hydroxy VD4 143032-85-3 C28H46O2
2,4-IMidazolidinedione, 5-[(7-chloro-1H-indol-3-yl)Methyl]-3-Methyl-, (5R)- 2,4-IMidazolidinedione, 5-[(7-chloro-1H-indol-3-yl)Methyl]-3-Methyl-, (5R)- 852391-19-6 C13H12ClN3O2
ACTB-1003 ACTB-1003 939805-30-8 C27H26F5N7O3
AM-095 AM-095 1345614-59-6 C27H25N2NaO5
Anagliptin Anagliptin 739366-20-2 C19H25N7O2
ATB 346 ATB 346 1226895-20-0 C21H19NO3S
AUZ 454 AUZ 454 853299-07-7 C24H26F3N7O2
BenzaMide, 3-[[4-[(5-hydroxy-2-Methylphenyl)aMino]-2-pyriMidinyl]aMino]- BenzaMide, 3-[[4-[(5-hydroxy-2-Methylphenyl)aMino]-2-pyriMidinyl]aMino]- 944795-06-6 C18H17N5O2
Vipadenant Vipadenant 442908-10-3 C16H15N7O
CBB 1007 CBB 1007 1379573-92-8 C27H34N8O4
Eliglustat Eliglustat 491833-29-5 C23H36N2O4
GSK 189254A GSK 189254A 720690-73-3 C21H25N3O2
LY 450108 LY 450108 376594-67-1 C19H22F2N2O3S
MethanesulfonaMide, N-[5-[4-[5-[[(2R,6S)-2,6-diMethyl-4-Morpholinyl]Methyl]-2-oxazolyl]-1H-indazol-6-yl]-2-Methoxy-3-pyridinyl]-, rel- MethanesulfonaMide, N-[5-[4-[5-[[(2R,6S)-2,6-diMethyl-4-Morpholinyl]Methyl]-2-oxazolyl]-1H-indazol-6-yl]-2-Methoxy-3-pyridinyl]-, rel- 1254036-66-2 C24H28N6O5S
SSR 240612 SSR 240612 464930-42-5 C42H53ClN4O7S
AZD-7687 AZD-7687 1166827-44-6 C21H25N3O3
AG 7352 Hydrochloride AG 7352 Hydrochloride 175519-16-1 C18H20ClN5O4S
11-Piperazinyldibenzo[b,e][1,4]diazepine 11-Piperazinyldibenzo[b,e][1,4]diazepine 56296-18-5 C17H18N4
J 147 J 147 1146963-51-0 C18H17F3N2O2
PCI-27483 PCI-27483 871266-63-6 C26H24N6O9S
SGI-110 SGI-110 929901-49-5 C18H24N9O10P
(S)-3-(3-fluoro-4-(6-(2-Methyl-2H-tetrazol-5-yl)pyridin-3-yl)phenyl)-5-(hydroxyMethyl)oxazolidin-2-one (S)-3-(3-fluoro-4-(6-(2-Methyl-2H-tetrazol-5-yl)pyridin-3-yl)phenyl)-5-(hydroxyMethyl)oxazolidin-2-one 1431699-67-0 C17H15FN6O3
BMN 673 (8R,9S) BMN 673 (8R,9S) 1207456-00-5 C19H14F2N6O
GRT6005 GRT6005 863513-91-1 C24H27FN2O
NVP BGJ398 phosphate NVP BGJ398 phosphate 1310746-10-1 C26H34Cl2N7O7P
SDZ 220-581 (AMMoniuM salt) SDZ 220-581 (AMMoniuM salt) 179411-94-0 C16H20ClN2O5P
NSP989 NSP989 304853-42-7 C16H15N3OS
TAK-593 TAK-593 1005780-62-0 C23H23N7O3
UNC0646 UNC0646 1320288-17-2 C36H59N7O2
Ripasudil hydrochloride dihydrate Ripasudil hydrochloride dihydrate 887375-67-9 C15H21ClFN3O3S
TAS-102 TAS-102 733030-01-8 C19H23Cl2F3N6O7
2-Acetylfuro-1,4-naphthoquinone 2-Acetylfuro-1,4-naphthoquinone 83280-65-3 C14H8O4
TPT-260 TPT-260 769856-81-7 C8H12N4S3
Leukadherin 1 Leukadherin 1 344897-95-6 C22H15NO4S2
BenzaMide, N-[3-[3-[4-[(diMethylaMino)Methyl]phenyl]pyrazolo[1,5-a]pyriMidin-7-yl]phenyl]-3-(trifluoroMethyl)- BenzaMide, N-[3-[3-[4-[(diMethylaMino)Methyl]phenyl]pyrazolo[1,5-a]pyriMidin-7-yl]phenyl]-3-(trifluoroMethyl)- 950736-05-7 C29H24F3N5O
GSK 2801 GSK 2801 1619994-68-1 C20H21NO4S
JNJ-38431055 JNJ-38431055 897732-93-3 C21H29N5O6S
2-Methyl-3-furoic acid iMidazolide 2-Methyl-3-furoic acid iMidazolide 1415238-77-5 C9H8N2O2
RGB-286638 (free base) RGB-286638 (free base) 784210-88-4 C29H35N7O4
Piribedil-d8 Piribedil-d8 1398044-45-5 C16H18N4O2
MK-8033 (hydrochloride) MK-8033 (hydrochloride) 1283000-43-0 C25H22ClN5O3S
Arginase inhibitor 1 Arginase inhibitor 1 1345808-25-4 C13H27BN2O4
LY3039478 LY3039478 1421438-81-4 C22H23F3N4O4
Brexpiprazole Brexpiprazole 913611-97-9 C25H27N3O2S
Setipiprant Setipiprant 866460-33-5 C24H19FN2O3
APY29 APY29 1216665-49-4 C17H16N8
4-Methyl-2-(1-piperidinyl)-quinoline 4-Methyl-2-(1-piperidinyl)-quinoline 5465-86-1 C15H18N2
DAA-1106 DAA-1106 220551-92-8 C23H22FNO4
N,N'-(Dithiodi-2,1-ethanediyl)bis[2,5-dichloro-benzenesulfonaMide N,N'-(Dithiodi-2,1-ethanediyl)bis[2,5-dichloro-benzenesulfonaMide 927822-86-4 C16H16Cl4N2O4S4
AZD-5069 AZD-5069 878385-84-3 C18H22F2N4O5S2
GSK-2269557 GSK-2269557 1254036-77-5 C26H29ClN6O
CDDO-EA CDDO-EA 932730-51-3 C33H46N2O3
GDC-0834 (RaceMate) GDC-0834 (RaceMate) 1133432-46-8 C33H36N6O3S
ITD-1 ITD-1 1099644-42-4 C27H29NO3
Afobazole (hydrochloride) Afobazole (hydrochloride) 173352-39-1 C15H22ClN3O2S
CDK7-IN-1 CDK7-IN-1 1604810-84-5 C31H28ClN7O2
JW 642 JW 642 1416133-89-5 C21H20F6N2O3
CUDC-427 CUDC-427 1446182-94-0 C29H36N6O4S
OTSSP167HCL OTSSP167HCL 1431698-10-0 C25H29Cl3N4O2
BMS-983970 BMS-983970 1584713-87-0 C26H26F4N4O3
AZD-5582 AZD-5582 1258392-53-8 C58H78N8O8
SUN11602 SUN11602 704869-38-5 C26H37N5O2
Bucladesine (calciuM salt) Bucladesine (calciuM salt) 938448-87-4 C18H26CaN5O8P
PF-06447475 PF-06447475 1527473-33-1 C17H15N5O
EPZ011969 EPZ011969 1598383-40-4 C35H51N5O4
MCC950 MCC950 210826-40-7 C20H24N2O5S
6-amino-4-(2,5-dimethoxyphenyl)-1,4-dihydro-3-(2-naphthalenyl)-pyrano[2,3-c]pyrazole-5-carbonitrile 6-amino-4-(2,5-dimethoxyphenyl)-1,4-dihydro-3-(2-naphthalenyl)-pyrano[2,3-c]pyrazole-5-carbonitrile 361185-42-4 C25H20N4O3
WZB117 WZB117 1223397-11-2 C20H13FO6
Csn-B Csn-B 321661-62-5 C18H26O5
2-[1-PIPERAZINYL]QUINOLINE MALEATE SALT 2-[1-PIPERAZINYL]QUINOLINE MALEATE SALT 5786-68-5 C17H19N3O4
Bis(4-cyanophenyl)methanol Bis(4-cyanophenyl)methanol 134521-16-7 C15H10N2O
CDKI-73 CDKI-73 1421693-22-2 C15H15FN6O2S2
3,6-Dichlorotrimellitic anhydride 3,6-Dichlorotrimellitic anhydride 81742-10-1 C9H2Cl2O5
E6446 (dihydrochloride) E6446 (dihydrochloride) 1345675-25-3 C27H36ClN3O3
PDE1-IN-1 (phosphate) PDE1-IN-1 (phosphate) 1642303-38-5 C29H29FN7O5P
RSV604 RSV604 676128-63-5 C22H17FN4O2
AZD 3759 AZD 3759 1626387-80-1 C22H23ClFN5O3
Nampt-IN-1 Nampt-IN-1 1698878-14-6 C20H25N3O5S
DASA-58 DASA-58 1203494-49-8 C19H23N3O6S2
GR148672X GR148672X 263890-70-6 C15H11F3N2O2S
PLX7904 PLX7904 1393465-84-3 C24H22F2N6O3S
XEN907 XEN907 912656-34-9 C21H21NO4
Naquotinib Naquotinib 1448232-80-1 C30H42N8O3
TASP0415914 TASP0415914 1292300-75-4 C13H17N5O3S
GPRP (acetate) GPRP (acetate) 157009-81-9 C20H35N7O7
NSC5844 NSC5844 140926-75-6 C20H16Cl2N4
Upadacitinib Upadacitinib 1310726-60-3 C17H19F3N6O
jnj39758979 jnj39758979 1046447-90-8 C11H19N5
DG172 (dihydrochloride) DG172 (dihydrochloride) 1361504-77-9 C20H21BrClN3
HLCL-61 (hydrochloride) HLCL-61 (hydrochloride) 1158279-20-9 C23H25ClN2O
TA-01 TA-01 1784751-18-3 C20H12F3N3
BI-7273 BI-7273 1883429-21-7 C20H23N3O3
SHP099 SHP099 1801747-42-1 C16H19Cl2N5
Lu AF21934 Lu AF21934 1445605-23-1 C14H16Cl2N2O2
BLU-554 BLU-554 1707289-21-1 C24H24Cl2N4O4
Elacestrant dihydrochloride Elacestrant dihydrochloride 1349723-93-8 C30H40Cl2N2O2
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