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Agonist Inhibitors

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Structure Chemical Name CAS MF
Flunisolide Flunisolide 3385-03-3 C24H31FO6
4-AMINO-1-TERT-BUTYL-3-(1'-NAPHTHYL)PYRAZOLO[3,4-D]PYRIMIDINE 4-AMINO-1-TERT-BUTYL-3-(1'-NAPHTHYL)PYRAZOLO[3,4-D]PYRIMIDINE 221243-82-9 C19H19N5
CANDESARTAN-D4 CANDESARTAN-D4 1346604-70-3 C24H16D4N6O3
RGX-104 free Acid RGX-104 free Acid 610318-54-2 C34H33ClF3NO3
Moricizine Moricizine 31883-05-3 C22H25N3O4S
OSI-420 OSI-420 183321-86-0 C21H21N3O4
2-ACETAMIDO-1,2,5-TRIDEOXY-1,5-IMINO-D-G LUCITOL 2-ACETAMIDO-1,2,5-TRIDEOXY-1,5-IMINO-D-G LUCITOL 105265-96-1 C8H16N2O4
6-CARBOXYFLUORESCEIN DIACETATE 6-CARBOXYFLUORESCEIN DIACETATE 3348-03-6 C25H16O9
BENZOTRIAZOL-1-YL-(2,4-DICHLORO-PHENYL)-METHANONE BENZOTRIAZOL-1-YL-(2,4-DICHLORO-PHENYL)-METHANONE 200626-61-5 C13H7Cl2N3O
KNK437 KNK437 218924-25-5 C13H11NO4
LFM-A13 LFM-A13 62004-35-7 C11H8Br2N2O2
5-METHOXY-3-(1,2,5,6-TETRAHYDRO-4-PYRIDINYL)-1H-INDOLE HEMISUCCINATE 5-METHOXY-3-(1,2,5,6-TETRAHYDRO-4-PYRIDINYL)-1H-INDOLE HEMISUCCINATE 107008-28-6 C18H22N2O5
Diloxanide furoate Diloxanide furoate 3736-81-0 C14H11Cl2NO4
1-(2-DIPHENYLMETHOXYETHYL)-4-(3-PHENYL-2-PROPENYL)-PIPERAZINE DIHYDROCHLORIDE 1-(2-DIPHENYLMETHOXYETHYL)-4-(3-PHENYL-2-PROPENYL)-PIPERAZINE DIHYDROCHLORIDE 67469-57-2 C28H32N2O
AC-ARG-CYS-GLY-VAL-PRO-ASP-NH2 AC-ARG-CYS-GLY-VAL-PRO-ASP-NH2 158841-76-0 C27H46N10O9S
U0126 U0126 109511-58-2 C18H16N6S2
CLOZAPINE N-OXIDE CLOZAPINE N-OXIDE 34233-69-7 C18H19ClN4O
TETRAETHYLENEPENTAMINE PENTAHYDROCHLORIDE TETRAETHYLENEPENTAMINE PENTAHYDROCHLORIDE 4961-41-5 C8H24ClN5
2',3'-DIDEOXY-3'-FLUORO-GUANOSINE 2',3'-DIDEOXY-3'-FLUORO-GUANOSINE 92562-88-4 C10H12FN5O3
alfa1-[[1,1-Dimethylethylamino]methyl]-4-hydroxy-1-(S),3-benzene dimethanol Hydrochlorid alfa1-[[1,1-Dimethylethylamino]methyl]-4-hydroxy-1-(S),3-benzene dimethanol Hydrochlorid 50293-90-8 C13H22ClNO3
Tacalcitol Tacalcitol 57333-96-7 C27H44O3
2,3,4,9-tetrahydro-2-methyl-1H-dibenzo[3,4:6,7]cyclohepta[1,2-c]pyridyl maleate 2,3,4,9-tetrahydro-2-methyl-1H-dibenzo[3,4:6,7]cyclohepta[1,2-c]pyridyl maleate 85650-57-3 C23H23NO4
7-CHLORO-4-INDANOL 7-CHLORO-4-INDANOL 145-94-8 C9H9ClO
Efaproxiral sodium Efaproxiral sodium 170787-99-2 C20H24NNaO4
ALEGLITAZAR ALEGLITAZAR 475479-34-6 C24H23NO5S
NUTLIN-3 NUTLIN-3 548472-68-0 C30H30Cl2N4O4
celgosivir celgosivir 121104-96-9 C12H21NO5
Tafenoquine Tafenoquine 106635-80-7 C24H28F3N3O3
Azacosterol dihydrochloride Azacosterol dihydrochloride 1249-84-9 C25H45ClN2O
Avermectin A1a, 25-cyclohexyl-4-O-de(2,6-dideoxy-3-O-methyl-.alpha.-L-arabino-hexopyranosyl)-5-demethoxy-25-de(1-methylpropyl)-22,23-dihydro-5-(hydroxyimino)- Avermectin A1a, 25-cyclohexyl-4-O-de(2,6-dideoxy-3-O-methyl-.alpha.-L-arabino-hexopyranosyl)-5-demethoxy-25-de(1-methylpropyl)-22,23-dihydro-5-(hydroxyimino)- 165108-07-6 C43H63NO11
[2-(4-chlorophenyl)quinolin-4-yl]-(2-piperidyl)methanol [2-(4-chlorophenyl)quinolin-4-yl]-(2-piperidyl)methanol 5428-80-8 C21H21ClN2O
10-Methoxycamptothecin 10-Methoxycamptothecin 19685-10-0 C21H18N2O5
SR 58611A SR 58611A 121524-09-2 C22H27Cl2NO4
DMP 777 DMP 777 157341-41-8 C31H40N4O6
doxorubicin(6-maleimidocaproyl)hydrazone doxorubicin(6-maleimidocaproyl)hydrazone 151038-96-9 C37H42N4O13
AS1975063 AS1975063 955925-61-8 C24H22N2O4.Na
2(BIS-(HYDROXYETHYL)AMINO)-6-(4-METHOXYBENZYLAMINO)-9-ISOPROPYL-PURINE 2(BIS-(HYDROXYETHYL)AMINO)-6-(4-METHOXYBENZYLAMINO)-9-ISOPROPYL-PURINE 199986-75-9 C20H28N6O3
VERATRYLCURCUMINOID VERATRYLCURCUMINOID 160096-59-3 C23H24O6
Rucaparib Rucaparib 283173-50-2 C19H18FN3O
3-[[3-[(DIMETHYLAMINO)CARBONYL]-2-HYDROXYPHENYL]AMINO]-4-[[(R)-1-(4-ISOPROPYLFURAN-2-YL)PROPYL]AMINO]CYCLOBUT-3-ENE-1,2-DIONE 3-[[3-[(DIMETHYLAMINO)CARBONYL]-2-HYDROXYPHENYL]AMINO]-4-[[(R)-1-(4-ISOPROPYLFURAN-2-YL)PROPYL]AMINO]CYCLOBUT-3-ENE-1,2-DIONE 473728-58-4 C23H27N3O5
adoprazine adoprazine 222551-17-9 C24H24FN3O2
inolitazone inolitazone 223132-37-4 C27H26N4O4S
Talarozole Talarozole 870093-23-5 C21H23N5S
Methylprednisolone sodium succinate Methylprednisolone sodium succinate 2375-03-3 C26H33O8.Na
Z-FL-COCHO Z-FL-COCHO 1373215-15-6 C25H29FN4O5
IB-MECA IB-MECA 152918-18-8 C18H19IN6O4
3-(3-oxo-4-propyl-quinoxalin-2-yl)propyl N-methylcarbamate 3-(3-oxo-4-propyl-quinoxalin-2-yl)propyl N-methylcarbamate 135779-82-7 C16H21N3O3
(-)-JASMONIC ACID (-)-JASMONIC ACID 6894-38-8 C12H18O3
(SCD1 inhibitor) (SCD1 inhibitor)
Azeliragon Azeliragon 603148-36-3 C32H38ClN3O2
Cephalothin Cephalothin 153-61-7 C16H16N2O6S2
Levobupivacaine Levobupivacaine 27262-47-1 C18H28N2O
Bis[(4-chlorophenyl)methylene]carbonimidic dihydrazide hydrochloride Bis[(4-chlorophenyl)methylene]carbonimidic dihydrazide hydrochloride 25875-51-8 C15H13Cl2N5
TANDUTINIB TANDUTINIB 228266-40-8 C27H43N3O4
2-Aminothiazole 2-Aminothiazole 96-50-4 C3H4N2S
DL-KYNURENINE DL-KYNURENINE 343-65-7 C10H12N2O3
IDAZOXAN HYDROCHLORIDE IDAZOXAN HYDROCHLORIDE 79944-56-2 C11H13ClN2O2
(S,S)-Hydroxy Bupropion (S,S)-Hydroxy Bupropion 192374-14-4 C13H18ClNO2
Prasugrel Hydrochloride Prasugrel Hydrochloride 389574-19-0 C20H20FNO3S.ClH
(R)-4-(2-(2-(2-METHYLPYRROLIDIN-1-YL)ETHYL)BENZOFURAN-5-YL)BENZONITRILE (R)-4-(2-(2-(2-METHYLPYRROLIDIN-1-YL)ETHYL)BENZOFURAN-5-YL)BENZONITRILE 460746-46-7 C22H22N2O
Dexrazoxane hydrochloride Dexrazoxane hydrochloride 149003-01-0 C11H16N4O4.ClH
5ALPHA-CHOLESTAN-3-ONE 5ALPHA-CHOLESTAN-3-ONE 566-88-1 C27H46O
N-(4-piperidinyl)-4-(2,6-dichlorobenzoylamino)-1H-pyrazole-3-carboxamide  Hcl N-(4-piperidinyl)-4-(2,6-dichlorobenzoylamino)-1H-pyrazole-3-carboxamide Hcl 902135-91-5 C16H18Cl3N5O2
CJ-42794 CJ-42794 847728-01-2 C22H17ClFNO4
N3-(7-Cyclobutyl-3-phenyl-1,2,4-triazolo[4,3-b]pyridazin-6-yl)-N1,N1,2,2-tetramethyl-1,3-propanediamine N3-(7-Cyclobutyl-3-phenyl-1,2,4-triazolo[4,3-b]pyridazin-6-yl)-N1,N1,2,2-tetramethyl-1,3-propanediamine 473382-39-7 C22H30N6
Tafamidis Tafamidis 594839-88-0 C14H7Cl2NO3
PIK-75 PIK-75 372196-67-3 C16H14BrN5O4S
Thiamet GDiscontinuedThiamet G Discontinued 1009816-48-1 C9H16N2O4S
Acotiamide hydrochloride trihydrate Acotiamide hydrochloride trihydrate 773092-05-0 C21H31ClN4O5S
MP-412 MP-412 451492-95-8 C27H28ClFN6O
XL-765,SAR245409 XL-765,SAR245409 1123889-87-1 C31H29N5O6S
LX-4211 LX-4211 1018899-04-1 C21H25ClO5S
MK-8617 MK-8617 1187990-87-9 C24H21N5O4
SU14813 SU14813 627908-92-3 C23H27FN4O4
3-Cyano-4-phenyl-6-(3-bromo-6-hydroxy)phenyl-2(1H)-pyridone 3-Cyano-4-phenyl-6-(3-bromo-6-hydroxy)phenyl-2(1H)-pyridone 491871-58-0 C18H11BrN2O2
2-(Hydroxymethyl)-2-(methoxymethyl)-1-azabicyclo[2.2.2]octan-3-one 2-(Hydroxymethyl)-2-(methoxymethyl)-1-azabicyclo[2.2.2]octan-3-one 5291-32-7 C10H17NO3
4,5-Dihydro-3-phenyl-5-isoxazoleaceticacid 4,5-Dihydro-3-phenyl-5-isoxazoleaceticacid 6501-72-0 C11H11NO3
2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl-benzoicacid 2-Cyclopentyl-4-(5-phenyl-1H-pyrrolo[2,3-b]pyridin-3-yl-benzoicacid 890842-28-1 C25H22N2O2
N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl-2-pyrrolidinedicarboxamide N-[1,1'-Biphenyl]-2-yl-1-[2-[(1-methyl-1H-benzimidazol-2-yl)thio]acetyl-2-pyrrolidinedicarboxamide 916141-36-1 C27H26N4O2S
Atopaxar Atopaxar 751475-53-3 C29H38FN3O5
Iron Chelator, Dp44mT Iron Chelator, Dp44mT 152095-12-0 C14H15N5S
4E1RCat 4E1RCat 328998-25-0 C28H18N2O6
TC-O 9311 TC-O 9311 444932-31-4 C20H19N3O4
TC-H 106 TC-H 106 937039-45-7 C20H25N3O2
Azilsartan-d5 Azilsartan-d5 1346599-45-8 C25H20N4O5
Tofogliflozin Tofogliflozin 903565-83-3 C22H26O6
Narlaprevir Narlaprevir 865466-24-6 C36H61N5O7S
Des(benzylpyridyl) Atazanavir Des(benzylpyridyl) Atazanavir 1192224-24-0 C26H43N5O7
ATN-224 ATN-224 649749-10-0 C5H14MoNOS4-
4-[3-Oxo-3-(2-oxo-2,3-dihydrobenzoxazol-6-yl)propyl]piperazine-1-carboxylic acid 3,5-dichlorobenzyl ester 4-[3-Oxo-3-(2-oxo-2,3-dihydrobenzoxazol-6-yl)propyl]piperazine-1-carboxylic acid 3,5-dichlorobenzyl ester 1144035-53-9 C22H21Cl2N3O5
trans-4-[4-(7-Aminopyrazolo[1,5-a]pyrimidin-6-yl)phenyl]cyclohexaneacetic acid trans-4-[4-(7-Aminopyrazolo[1,5-a]pyrimidin-6-yl)phenyl]cyclohexaneacetic acid 1031336-60-3 C20H22N4O2
GW 627368X GW 627368X 439288-66-1 C30H28N2O6S
SR 1001 SR 1001 1335106-03-0 C15H13F6N3O4S2
(R)-2-(4'-(4-(((1-(2-chlorophenyl)ethoxy)carbonyl)aMino)-3-Methylisoxazol-5-yl)-[1,1'-biphenyl]-4-yl)acetic acid (R)-2-(4'-(4-(((1-(2-chlorophenyl)ethoxy)carbonyl)aMino)-3-Methylisoxazol-5-yl)-[1,1'-biphenyl]-4-yl)acetic acid 1228690-19-4 C27H23ClN2O5
N,N'-Bis(2-bromoethyl)phosphorodiamidic acid (1-methyl-2-nitro-1H-imidazol-5-yl)methyl ester N,N'-Bis(2-bromoethyl)phosphorodiamidic acid (1-methyl-2-nitro-1H-imidazol-5-yl)methyl ester 918633-87-1 C9H16Br2N5O4P
6-Fluoro-2-[4-(pyridin-2-yl)-3-butynyl]imidazo[1,2-a]pyridine 6-Fluoro-2-[4-(pyridin-2-yl)-3-butynyl]imidazo[1,2-a]pyridine 872363-17-2 C16H12FN3
Nesbuvir Nesbuvir 691852-58-1 C22H23FN2O5S
(alphaR)-3,5-Difluoro-alpha-hydroxybenzeneacetic acid 2-(2-ethyl-4-hydroxy-3-methylbenzoyl)hydrazide (alphaR)-3,5-Difluoro-alpha-hydroxybenzeneacetic acid 2-(2-ethyl-4-hydroxy-3-methylbenzoyl)hydrazide 1184940-47-3 C18H18F2N2O4
BMS-911543 BMS-911543 1271022-90-2 C23H28N8O
NIBR-17 NIBR-17 944396-88-7 C18H20N8O2
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