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Agonist Inhibitors

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Structure Chemical Name CAS MF
Bupropion Bupropion 34911-55-2 C13H18ClNO
6-THIO-2'-DEOXYGUANOSINE 6-THIO-2'-DEOXYGUANOSINE 789-61-7 C10H13N5O3S
Linaprazan Linaprazan 248919-64-4 C21H26N4O2
CHLORPHENOXAMINE CHLORPHENOXAMINE 77-38-3 C18H22ClNO
CYCLO(-ARG-GLY-ASP-D-TYR-LYS) CYCLO(-ARG-GLY-ASP-D-TYR-LYS) 217099-14-4 C27H41N9O8
2,3,4-TRIMETHOXYBENZYL ALCOHOL 2,3,4-TRIMETHOXYBENZYL ALCOHOL 71989-96-3 C10H14O4
GW843682,  5-(5,6-Dimethoxy-1H-benzimidazol-1-yl)-3-{[2-(trifluoromethyl)-benzyl]oxy}thiophene-2-carboxamide GW843682, 5-(5,6-Dimethoxy-1H-benzimidazol-1-yl)-3-{[2-(trifluoromethyl)-benzyl]oxy}thiophene-2-carboxamide 660868-91-7 C22H18F3N3O4S
Atrasentan hydrochloride Atrasentan hydrochloride 195733-43-8 C29H38N2O6.ClH
Talaporfin sodium Talaporfin sodium 220201-34-3 C38H42N5NaO9
4-Methylpyrazole 4-Methylpyrazole 7554-65-6 C4H6N2
Zacopride hydrochloride Zacopride hydrochloride 101303-98-4 C15H21Cl2N3O2
CP-547632 CP-547632 252003-65-9 C20H24BrF2N5O3S
1-(4-Fluorophenyl)-N-[3-fluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-1,2-dihydro-2-oxo-3-pyridinecarboxamide 1-(4-Fluorophenyl)-N-[3-fluoro-4-(1H-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-1,2-dihydro-2-oxo-3-pyridinecarboxamide 888719-03-7 C25H16F2N4O3
3-[3-[2-(1-Piperidinyl)ethoxy]phenyl]-5-(1H-1,2,4-triazol-5-yl)-1H-indazole 3-[3-[2-(1-Piperidinyl)ethoxy]phenyl]-5-(1H-1,2,4-triazol-5-yl)-1H-indazole 395104-30-0 C22H24N6O
N-[2,4-Difluoro-3-[[5-(3-pyridinyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]carbonyl]phenyl]-2-propanesulfonamide N-[2,4-Difluoro-3-[[5-(3-pyridinyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]carbonyl]phenyl]-2-propanesulfonamide 918505-61-0 C22H18F2N4O3S
Nsc66811 Nsc66811 6964-62-1 C23H20N2O
VCH-916 VCH-916 1200133-34-1 C26H36KNO4S
GW791343 dihydrochloride GW791343 dihydrochloride 1019779-04-4 C20H24F2N4O
Vaniprevir Vaniprevir 923590-37-8 C38H55N5O9S
1-(4-Methoxyphenyl)-2-methyl-3-nitro-1H-indol-6-ol 1-(4-Methoxyphenyl)-2-methyl-3-nitro-1H-indol-6-ol 147591-46-6 C16H14N2O4
Losartan-d4 Carboxylic Acid Losartan-d4 Carboxylic Acid 1246820-62-1 C22H21ClN6O2
Delamanid Delamanid 681492-22-8 C25H25F3N4O6
MK-8998 MK-8998 953778-58-0 C20H23F3N2O2
Amg 517 Amg 517 659730-32-2 C20H13F3N4O2S
AC-55541 AC-55541 916170-19-9 C25H20BrN5O3
Unii-950o97nupo Unii-950o97nupo 377727-87-2 C25H29N9O3
N-[trans-4-[2-(6-Cyano-3,4-dihydro-2(1H)-isoquinolinyl)ethyl]cyclohexyl]-4-quinolinecarboxamide N-[trans-4-[2-(6-Cyano-3,4-dihydro-2(1H)-isoquinolinyl)ethyl]cyclohexyl]-4-quinolinecarboxamide 215803-78-4 C28H30N4O
BML-210 BML-210 537034-17-6 C20H25N3O2
FIPI FIPI 939055-18-2 C23H24FN5O2
2-Amino-6-[2-(cyclopropylmethoxy)-6-hydroxyphenyl]-4-(4-piperidinyl)-3-pyridinecarbonitrile hydrochloride 2-Amino-6-[2-(cyclopropylmethoxy)-6-hydroxyphenyl]-4-(4-piperidinyl)-3-pyridinecarbonitrile hydrochloride 406209-26-5 C21H25ClN4O2
SCH-900776 SCH-900776 891494-64-7 C15H18BrN7
AnaMorelin hydrochloride AnaMorelin hydrochloride 861998-00-7 C31H43ClN6O3
BN-2629 BN-2629 232931-57-6 C31H32N4O6
ARRY-520 ARRY-520 885060-09-3 C20H22F2N4O2S
KN-92 (hydrochloride) KN-92 (hydrochloride) 1431698-47-3 C24H26Cl2N2O3S
PSN632408 PSN632408 857652-30-3 C18H24N4O4
CEP-32496 CEP-32496 1227678-26-3 C24H23ClF3N5O5
A 804598 A 804598 1125758-85-1 C19H17N5
NDT 9513727 NDT 9513727 439571-48-9 C36H35N3O4
(E)-1-(3-chloro-4-fluorophenyl)-4-((5-nitrofuran-2-yl)Methylene)pyrazolidine-3,5-dione (E)-1-(3-chloro-4-fluorophenyl)-4-((5-nitrofuran-2-yl)Methylene)pyrazolidine-3,5-dione 423148-78-1 C14H7ClFN3O5
GAP 27 GAP 27 198284-64-9 C60H101N15O17
AST-1306 AST-1306 897383-62-9 C24H18ClFN4O2
GSK-25 GSK-25 874119-56-9 C24H16Cl2F2N6O
1alpha, 24, 25-Trihydroxy VD2 1alpha, 24, 25-Trihydroxy VD2 457048-34-9 C28H44O4
BAY 61-3606 (dihydrochloride) BAY 61-3606 (dihydrochloride) 648903-57-5 C20H20Cl2N6O3
BIX02189 BIX02189 1265916-41-3 C27H28N4O2
PDK1 inhibitor PDK1 inhibitor 1001409-50-2 C28H22F2N4O4
Belumosudil Belumosudil 911417-87-3 C26H24N6O2
5-PyriMidinecarboxaMide, 2-[[2-(3-chloro-4-hydroxyphenyl)ethyl]aMino]-4-[(phenylMethyl)aMino]- 5-PyriMidinecarboxaMide, 2-[[2-(3-chloro-4-hydroxyphenyl)ethyl]aMino]-4-[(phenylMethyl)aMino]- 919486-40-1 C20H20ClN5O2
BAY-57-1293 BAY-57-1293 348086-71-5 C18H18N4O3S2
BenzenesulfonaMide, 5-(phenylsulfonyl)-N-4-piperidinyl-2-(trifluoroMethyl)- BenzenesulfonaMide, 5-(phenylsulfonyl)-N-4-piperidinyl-2-(trifluoroMethyl)- 915759-45-4 C18H19F3N2O4S2
ELN 441958 ELN 441958 913064-47-8 C29H29ClN4O2
GeMigliptin GeMigliptin 911637-19-9 C18H19F8N5O2
GLI1-Mediated transcription inhibitor GLI1-Mediated transcription inhibitor 496794-70-8 C24H23ClN4O3
LOR 253 LOR 253 916151-99-0 C22H14FN5
MibaMpator MibaMpator 375345-95-2 C21H30N2O4S2
N3PT N3PT 13860-66-7 C13H19Cl2N3OS
Opicapone Opicapone 923287-50-7 C15H10Cl2N4O6
PPQ-102 PPQ-102 931706-15-9 C26H22N4O3
Repertaxin Repertaxin 266359-83-5 C14H21NO3S
XL647 XL647 781613-23-8 C24H25Cl2FN4O2
PF 04447943 PF 04447943 1082744-20-4 C20H25N7O2
Hederagenin 3-O-α-L-rhaMnopyranosyl(1→2)-(β-D-glucopyranosyl(1→4))-α-L-arabinopyranoside Hederagenin 3-O-α-L-rhaMnopyranosyl(1→2)-(β-D-glucopyranosyl(1→4))-α-L-arabinopyranoside 68027-15-6 C47H76O17
L 2-401 L 2-401 883050-24-6 C16H13FN2O2S
Roniciclib Roniciclib 1223498-69-8 C18H21F3N4O3S
(2S)-Methyl 2-(2-chlorophenyl)-2-(2-oxo-7,7a-dihydrothieno[3,2-c]pyridin-5(2H,4H,6H)-yl)acetate (2S)-Methyl 2-(2-chlorophenyl)-2-(2-oxo-7,7a-dihydrothieno[3,2-c]pyridin-5(2H,4H,6H)-yl)acetate 1147350-75-1 C16H16ClNO3S
AT 7867 dihydrochloride AT 7867 dihydrochloride 1431697-86-7 C20H21Cl2N3
CC401 HCl CC401 HCl 1438391-30-0 C22H25ClN6O
c-Met inhibitor 1 c-Met inhibitor 1 1357072-61-7 C17H14N8S
XR9576 XR9576 625375-83-9 C39H42N4O9S
QNZ-46 QNZ-46 1237744-13-6 C24H17N3O6
LH-846 LH-846 639052-78-1 C16H13ClN2OS
PF 4618433 PF 4618433 1166393-85-6 C24H27N7O2
Pyrido[2,3-d]pyriMidin-7(8H)-one, 6-(2,4-dichlorophenyl)-8-ethyl-2-[[3-fluoro-4-(1-piperazinyl)phenyl]aMino]- Pyrido[2,3-d]pyriMidin-7(8H)-one, 6-(2,4-dichlorophenyl)-8-ethyl-2-[[3-fluoro-4-(1-piperazinyl)phenyl]aMino]- 1232030-35-1 C25H23Cl2FN6O
LY 2606368 LY 2606368 1234015-52-1 C18H19N7O2
ADH 1 ADH 1 229971-81-7 C22H34N8O6S2
LY2334737 LY2334737 892128-60-8 C17H25F2N3O5
ML281 ML281 1404437-62-2 C22H19N3O2S
O-Propargyl-PuroMycin O-Propargyl-PuroMycin 1416561-90-4 C24H29N7O5
20-O-Acetylingenol-3-angelate 20-O-Acetylingenol-3-angelate 82425-35-2 C27H36O7
AICAR (phosphate) AICAR (phosphate) 681006-28-0 C9H17N4O9P
LHW090-A7 LHW090-A7 1308256-94-1 C20H22ClNO4
ZLN005 ZLN005 49671-76-3 C17H18N2
AdipoRon AdipoRon 924416-43-3 C27H28N2O3
LEE011 (hydrochloride) LEE011 (hydrochloride) 1211443-80-9 C23H31ClN8O
ML314 ML314 1448895-09-7 C24H28N4O3
Emixustat hydrochloride Emixustat hydrochloride 1141934-97-5 C16H26ClNO2
1-tert-butyl-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyriMidin-4-aMine hydrochloride 1-tert-butyl-3-(naphthalen-1-yl)-1H-pyrazolo[3,4-d]pyriMidin-4-aMine hydrochloride 956025-47-1 C19H20ClN5
Atglistatin Atglistatin 1469924-27-3 C17H21N3O
PCI-32765 (RaceMate) PCI-32765 (RaceMate) 936563-87-0 C25H24N6O2
GNE-7915 (tosylate) GNE-7915 (tosylate) 2070015-00-6 C26H29F4N5O6S
4EGI-1 4EGI-1 315706-13-9 C18H12Cl2N4O4S
2-AMino-6-chloro-α-cyano-3-(ethoxycarbonyl)-4H-1-benzopyran-4-acetic Acid Ethyl Ester 2-AMino-6-chloro-α-cyano-3-(ethoxycarbonyl)-4H-1-benzopyran-4-acetic Acid Ethyl Ester 305834-79-1 C17H17ClN2O5
Thiazolidine-4-carboxylic acid Thiazolidine-4-carboxylic acid 444-27-9 C4H7NO2S
RO5126766(CH5126766) RO5126766(CH5126766) 946128-88-7 C21H18FN5O5S
I-CBP112 I-CBP112 1640282-31-0 C27H36N2O5
IWP-3 IWP-3 687561-60-0 C22H17FN4O2S3
Cerdulatinib Cerdulatinib 1198300-79-6 C20H27N7O3S
HG-14-10-04 HG-14-10-04 1356962-34-9 C29H34ClN7O
kb-NB77-78 kb-NB77-78 1350622-33-1 C18H25NO3Si
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